Preparation of β-fluoro- and ββ-difluoro-histidinols

Journal of Fluorine Chemistry

Volumn 123, Issue 1, 2003, Pages 95-99

  Dolensky, Bohumil ^a   Narayanan, Jayan ^a   Kirk, Kenneth L ^a  

^a NATIONAL INSTITUTE OF DIABETES AND DIGESTIVE AND KIDNEY DISEASES   (United States)

Author keywords

"FBr" addition; Histidine biosynthesis; Imidazole analogues; Solvent effects on halogen mobility

Indexed keywords

AZIDE; CARBOXYLIC ACID; HISTIDINOL; ORGANOFLUORINE DERIVATIVE; SOLVENT; TRITYL DERIVATIVE;

ARTICLE; CHEMICAL BOND; CHEMICAL REACTION; CHEMICAL STRUCTURE; CONTROLLED STUDY; DRUG SYNTHESIS; FLUORINATION; REACTION ANALYSIS; REDUCTION; SOLVENT EFFECT;

EID: 0041784646     PISSN: 00221139     EISSN: None     Source Type: Journal    
DOI: 10.1016/S0022-1139(03)00096-4     Document Type: Article

References (12)

1. Correa J.F. Cabeza M.I. Sardina F.J. Tetrahedron Lett. 37 1996 9259-9262
2. Warrington R.C. Fang W.D. Zhang L. Shieh M. Saier M.H. Jr. Anticancer Res. 16 1996 3629-3634
3. Warrington R.C. Fang W.D. Zhang L. Anticancer Res. 16 1996 3641-3646
4. Stolfi R.L. Martin D.S. Chemotherapy 36 1990 435-440
5. Percy E. Singh M. Takahashi T. Takeuchi Y. Kirk K.L. J. Fluorine Chem. 91 1998 5-7
6. Dolensky B. Kirk K.L. J. Org. Chem. 67 2002 3468-3473
7. Dolensky B. Kirk K.L. J. Org. Chem. 66 2001 4687-4691
8. Deng W.-P. Nam G. Fan J. Kirk K.L. J. Org. Chem. 68 2003 2798-2802
9. B.E. Smart, Characteristics of C-F Systems, in: R.E. Banks, B.E. Smart, J.C. Tatlow (Eds.), Organofluorine Chemistry, Principles and Commercial Applications, Plenum Press, New York, 1994, pp. 57-82.
10. Haufe G. Alvernhe G. Laurent A. Ernet T. Goj O. Kröger S. Sattler A. Org. Synth. 76 1999 159
11. Kremlev M.M. Haufe G. J. Fluorine Chem. 90 1998 121
12. Malik A.A. Tzeng D. Cheng P. Baum K. J. Org. Chem. 56 1991 3043-3044