-
1
-
-
0017236348
-
Bestatin, an inhibitor of aminopeptidase B, produced by actinomycetes
-
Umezawa, H., Aoyagi, T., Suda, H., Hamada, M., and Takeuchi, T., Bestatin, an inhibitor of aminopeptidase B, produced by actinomycetes. J. Antibiot., 29, 97-101 (1976).
-
(1976)
J. Antibiot.
, vol.29
, pp. 97-101
-
-
Umezawa, H.1
Aoyagi, T.2
Suda, H.3
Hamada, M.4
Takeuchi, T.5
-
2
-
-
0017596420
-
Synthesis and structure-activity relationships of bestatin analogues, inhibitors of aminopeptidase B
-
Nishizawa, R., Saino, T., Takita, T., Suda, H., Aoyagi, T., and Umezawa, H., Synthesis and structure-activity relationships of bestatin analogues, inhibitors of aminopeptidase B. J. Med. Chem., 20, 510-515 (1977)
-
(1977)
J. Med. Chem.
, vol.20
, pp. 510-515
-
-
Nishizawa, R.1
Saino, T.2
Takita, T.3
Suda, H.4
Aoyagi, T.5
Umezawa, H.6
-
3
-
-
0017131813
-
Inhibition of aminopeptidase B and leucine aminopeptidase by bestatin and its stereoisomer
-
Suda, H., Aoyagi, T., Takeuchi, T., and Umezawa, H., Inhibition of aminopeptidase B and leucine aminopeptidase by bestatin and its stereoisomer. Arch. Biochem. Biophys., 177, 196-200 (1976)
-
(1976)
Arch. Biochem. Biophys.
, vol.177
, pp. 196-200
-
-
Suda, H.1
Aoyagi, T.2
Takeuchi, T.3
Umezawa, H.4
-
4
-
-
0020577840
-
Identification and properties of the cell membrane bound leucine aminopeptidase interacting with the potential immunostimulant and chemotherapeutic agent bestatin
-
Leyhausen, G., Schuster, D. K., Vaith, P., Zahn, R. K., Umezawa, H., Falke, D., and Mueller, W. E. G., Identification and properties of the cell membrane bound leucine aminopeptidase interacting with the potential immunostimulant and chemotherapeutic agent bestatin. Biochem. Pharmacol., 32, 1051-1057 (1983).
-
(1983)
Biochem. Pharmacol.
, vol.32
, pp. 1051-1057
-
-
Leyhausen, G.1
Schuster, D.K.2
Vaith, P.3
Zahn, R.K.4
Umezawa, H.5
Falke, D.6
Mueller, W.E.G.7
-
5
-
-
0018815111
-
Regio- and stereospecific synthesis of threo-3-amino-2-hydroxy-acids, novel amino acids containing aminopeptidase inhibitors of microbial origin
-
Kato, K., Sino, T., Nishizawa, R., Takita, T., and Umezawa, H., Regio- and stereospecific synthesis of threo-3-amino-2-hydroxy-acids, novel amino acids containing aminopeptidase inhibitors of microbial origin. J. Chem. Soc., Perkin Trans. I, 1618-1621 (1980)
-
(1980)
J. Chem. Soc., Perkin Trans. I
, pp. 1618-1621
-
-
Kato, K.1
Sino, T.2
Nishizawa, R.3
Takita, T.4
Umezawa, H.5
-
6
-
-
0020112101
-
Stereo and regioselective openings of chiral 2,3-epoxy alcohols, versatile routes to optically pure natural products and drugs, unusual kinetic resolutions
-
Sharpless, K. B., Behrens, C. H., Katsuki, T., Lee, A. W. M., Martin, V. S., Takatani, M., Viti, S. M., Walker, F. J., and Woodard, S. S., Stereo and regioselective openings of chiral 2,3-epoxy alcohols, versatile routes to optically pure natural products and drugs, unusual kinetic resolutions. Pure Appl. Chem., 55, 589-604 (1983)
-
(1983)
Pure Appl. Chem.
, vol.55
, pp. 589-604
-
-
Sharpless, K.B.1
Behrens, C.H.2
Katsuki, T.3
Lee, A.W.M.4
Martin, V.S.5
Takatani, M.6
Viti, S.M.7
Walker, F.J.8
Woodard, S.S.9
-
7
-
-
0021181831
-
A stereocontrolled synthesis of (—)-bestatin from an acyclic allylamine by iodocyclocarbamation
-
Kobayashi, S., Isobe, T., and Ohno, M., A stereocontrolled synthesis of (—)-bestatin from an acyclic allylamine by iodocyclocarbamation. Tetrahedron Lett., 25, 5079-5082 (1984);
-
(1984)
Tetrahedron Lett.
, vol.25
, pp. 5079-5082
-
-
Kobayashi, S.1
Isobe, T.2
Ohno, M.3
-
8
-
-
0024450764
-
Synthesis of β-Amino-α-hydroxy Acids via Aldol Condensation of a Chiral Glycolate Enolate. Synthesis of (—)-Bestatin
-
Pearson, W. H. and Hines, J. V., Synthesis of β-Amino-α-hydroxy Acids via Aldol Condensation of a Chiral Glycolate Enolate. Synthesis of (—)-Bestatin. J. Org. Chem., 54, 4235-4237 (1989)
-
(1989)
J. Org. Chem.
, vol.54
, pp. 4235-4237
-
-
Pearson, W.H.1
Hines, J.V.2
-
9
-
-
0025006910
-
An improved one-pot method for stereoselective synthesis of the (2S',3R)-3-amino-2-hydroxy acids: Key intermediates for bestatin and amastatin
-
Herranz, R., Castro-Pichel, J., Vinuesa, S., and Garciα-Lopez, T., An improved one-pot method for stereoselective synthesis of the (2S',3R)-3-amino-2-hydroxy acids: key intermediates for bestatin and amastatin. J. Org. Chem., 55, 2232-2234 (1990)
-
(1990)
J. Org. Chem.
, vol.55
, pp. 2232-2234
-
-
Herranz, R.1
Castro-Pichel, J.2
Vinuesa, S.3
Garciα-Lopez, T.4
-
10
-
-
0026607899
-
A stereocontrolled synthesis of the (2R,3S)- and (2S,3R)-3-amino-2-hydrox-ybutyric acid derivatives, the key components of a renin inhibitor and bestatin
-
Kobayashi, Y., Takemoto, Y., Kamijo, T., Harada, H., Ito, Y., and Terashima, S., A stereocontrolled synthesis of the (2R,3S)- and (2S,3R)-3-amino-2-hydrox-ybutyric acid derivatives, the key components of a renin inhibitor and bestatin. Tetrahedron, 48, 1853-1868 (1992)
-
(1992)
Tetrahedron
, vol.48
, pp. 1853-1868
-
-
Kobayashi, Y.1
Takemoto, Y.2
Kamijo, T.3
Harada, H.4
Ito, Y.5
Terashima, S.6
-
11
-
-
0026471808
-
A stereospecific synthesis of (—)-bestatin from L-malic acid
-
Norman, B. H. and Morris, M. L., A stereospecific synthesis of (—)-bestatin from L-malic acid. Tetrahedron Lett., 33, 6803-6806 (1992)
-
(1992)
Tetrahedron Lett.
, vol.33
, pp. 6803-6806
-
-
Norman, B.H.1
Morris, M.L.2
-
12
-
-
0027272436
-
An enantio-divergent synthesis of threo-β-amino alcohols: Preparation of key intermediates for bestatin and the related peptides
-
Kawabata, T., Kiryu, Y., Sugiura, Y., and Fuji, K., An enantio-divergent synthesis of threo-β-amino alcohols: preparation of key intermediates for bestatin and the related peptides. Tetrahedron Lett., 34, 5127-5130 (1993).
-
(1993)
Tetrahedron Lett.
, vol.34
, pp. 5127-5130
-
-
Kawabata, T.1
Kiryu, Y.2
Sugiura, Y.3
Fuji, K.4
-
13
-
-
0025799274
-
Chemistry of aspartic acid and its application to drug-synthesis
-
Matsumoto, K. and Seki, M., Chemistry of aspartic acid and its application to drug-synthesis. J. Syn. Org. Chem. Jpn, (in Japanese), 49, 26-41 (1991)
-
(1991)
J. Syn. Org. Chem. Jpn, (In Japanese)
, vol.49
, pp. 26-41
-
-
Matsumoto, K.1
Seki, M.2
-
14
-
-
0008481013
-
Chemistry of amino acids and its application to drug synthesis
-
Seki, M. and Matsumoto, K., Chemistry of amino acids and its application to drug synthesis. Bioindustry, (in Japanese), 1995, 5-19 (1995).
-
(1995)
Bioindustry, (In Japanese)
, vol.1995
, pp. 5-19
-
-
Seki, M.1
Matsumoto, K.2
-
15
-
-
85009552278
-
A novel synthesis of allophenylnor-statine from (I?)-aspartic acid
-
(in press)
-
Seki, M. and Matsumoto, K., A novel synthesis of allophenylnor-statine from (i?)-aspartic acid. Synthesis (in press).
-
Synthesis
-
-
Seki, M.1
Matsumoto, K.2
|