SCOPUS 정보 검색 플랫폼

Volumn , Issue 11, 2003, Pages 1699-1704

Concise synthesis of cyclothialidine analogues with ring sizes from 12 to 15: Novel macrocyclization protocol involving reductive thiolation

(3) Geiwiz, J a,b Goetschi, E a Hebeisen, P a

a F HOFFMANN LA ROCHE LTD (Switzerland)

b Ciba Grenzach GmbH (Germany)

Author keywords

Antibacterials; Cyclothialidine; DNA gyrase inhibitor; Macrocyclization; Reductive thiolation

Indexed keywords

BACTERIA; DNA; ENZYME INHIBITION; ENZYMES; SYNTHESIS (CHEMICAL);

CONGENERS;

ORGANIC COMPOUNDS;

ANTIINFECTIVE AGENT; BENZILIC ACID DERIVATIVE; BENZYLIC SULFIDE; CYCLOTHIALIDINE DERIVATIVE; GYRASE INHIBITOR; LACTONE; MACROCYCLIC COMPOUND; THIOL DERIVATIVE; UNCLASSIFIED DRUG;

ACYLATION; ANTIBACTERIAL ACTIVITY; ARTICLE; CYCLIZATION; DRUG STRUCTURE; DRUG SYNTHESIS; INFRARED SPECTROSCOPY; MASS SPECTROMETRY; MITSUNOBU REACTION; PROTON NUCLEAR MAGNETIC RESONANCE; REDUCTION; STRUCTURE ACTIVITY RELATION;

EID: 0041737756 PISSN: 00397881 EISSN: None Source Type: Journal
DOI: 10.1055/s-2003-40877 Document Type: Article

Times cited : (9)

References (7)

1
- 0028013120
- Watanabe, J.; Nakada, N.; Sawairi, S.; Shimada, H.; Ohshima, S.; Kamiyama, T.; Arisawa, M. J. Antibiotics 1994, 47, 32.
- (1994) Antibiotics , vol.47 , pp. 32
- Watanabe, J.¹ Nakada, N.² Sawairi, S.³ Shimada, H.⁴ Ohshima, S.⁵ Kamiyama, T.⁶ Arisawa, M.J.⁷

2
- 0041946902
- European Patent App. EP 675122, 1995
- Geiwiz, J.; Goetschi, E.; Hebeisen, P.; Link, H.; Luebbers, T. European Patent App. EP 675122, 1995; Chem. Abstr. 1996, 124, 146213.
- (1996) Chem. Abstr. , vol.124 , pp. 146213
- Geiwiz, J.¹ Goetschi, E.² Hebeisen, P.³ Link, H.⁴ Luebbers, T.⁵

3
- 0037767712
- Yamazaki, M., Ed.; Blackwell: Oxford
- Goetschi, E.; Angehrn, P.; Gmuender, H.; Hebeisen, P.; Link, H.; Masciadri, R.; Reindl, P.; Ricklin, F. In Today and Tomorrow, Proceedings of AIMECS 95, Tokyo, September 1995; Yamazaki, M., Ed.; Blackwell: Oxford, 1996, 263-270.
- (1996) Today and Tomorrow, Proceedings of AIMECS 95, Tokyo, September 1995 , pp. 263-270
- Goetschi, E.¹ Angehrn, P.² Gmuender, H.³ Hebeisen, P.⁴ Link, H.⁵ Masciadri, R.⁶ Reindl, P.⁷ Ricklin, F.⁸

4
- 0042948520
- in press
- Angehrn, P.; Buchmann, S.; Goetschi, E.; Gmuender, H.; Hebeisen, P.; Kostrewa, D.; Link, H.; Luebbers, T.; Masciadri, R.; Nielsen, J.; Reindl, P.; Ricklin, F.; Schmitt-Hoffmann, A., Theil, F.-P. J. Med. Chem., in press.
- J. Med. Chem.
- Angehrn, P.¹ Buchmann, S.² Goetschi, E.³ Gmuender, H.⁴ Hebeisen, P.⁵ Kostrewa, D.⁶ Link, H.⁷ Luebbers, T.⁸ Masciadri, R.⁹ Nielsen, J.¹⁰ Reindl, P.¹¹ Ricklin, F.¹² Schmitt-Hoffmann, A.¹³ Theil, F.-P.¹⁴

5
- 0042447611
- PCT Int. Appl. WO 9218490, 1992
- Arisawa, M.; Goetschi, E.; Kamiyama, T.; Masciadri, R.; Shimada, H.; Watanabe, J.; Hebeisen, P.; Link, H. PCT Int. Appl. WO 9218490, 1992; Chem. Abstr. 1993, 119, 117285.
- (1993) Chem. Abstr. , vol.119 , pp. 117285
- Arisawa, M.¹ Goetschi, E.² Kamiyama, T.³ Masciadri, R.⁴ Shimada, H.⁵ Watanabe, J.⁶ Hebeisen, P.⁷ Link, H.⁸

6
- 0029956650
- Götschi, E.; Jenny, Ch. J.; Reindl, P.; Ricklin, F. Helv. Chim. Acta 1996, 79, 2219.
- (1996) Helv. Chim. Acta , vol.79 , pp. 2219
- Götschi, E.¹ Jenny, Ch.J.² Reindl, P.³ Ricklin, F.⁴

7
- 0028204031
- Richter, L. S.; Marsters, J. C. Jr.; Gadek, T. R. Tetrahedron Lett. 1994, 35, 1631.
- (1994) Tetrahedron Lett. , vol.35 , pp. 1631
- Richter, L.S.¹ Marsters J.C., Jr.² Gadek, T.R.³

* 이 정보는 Elsevier사의 SCOPUS DB에서 KISTI가 분석하여 추출한 것입니다.