Estimation of the solubility of sulfonamides in aqueous media from partition coefficients and entropies of fusion

Physics and Chemistry of Liquids

Volumn 40, Issue 4, 2002, Pages 411-420

  Martínez, Fleming ^a   Gómez, Alfredo ^a  

^a UNIVERSIDAD NACIONAL DE COLOMBIA   (Colombia)

Author keywords

Partition coefficient; Solubility; Sulfonamides; Yalkowsky Valvani and Jain Yalkowsky equations

Indexed keywords

MELTING; SOLUBILITY;

AQUEOUS MEDIA;

SULFUR COMPOUNDS;

ENTROPY; EQUATION; LIQUID-LIQUID MIXING; MATHEMATICAL ANALYSIS; SOLUBILITY;

EID: 0041648745     PISSN: 00319104     EISSN: None     Source Type: Journal    
DOI: 10.1080/0031910021000017735     Document Type: Article

References (36)

1. S.C. Valvani and S.H. Yalkowsky (1980). In: S.H. Yalkowsky, A.A. Sinkula and S.C. Valvani (Eds.), Physical Chemical Properties of Drugs, Chap. 6, pp. 201-229. Marcel Dekker, Inc., New York.
2. S.H. Yalkowsky and S.C. Valvani (1980). J. Pharm. Sci., 69, 912.
3. M.M. Morelock, L.L. Choi, G.L. Bell and J.L. Wright (1994). J. Pharm. Sci., 83, 948.
4. G.L. Amidon and S.T. Anik (1976). J. Pharm. Sci., 65, 801.
5. D.E. Leahy (1986). J. Pharm. Sci., 75, 629.
6. R.M. Soler-Roca, G.M. Anton-Fos, R. Garcia-Domenech and J. Galvez-Alvarez (1991). Anal. Real Acad. Farm., 57, 563.
7. J. Huuskonen, M. Salo and J. Taskinen (1997). J. Pharm. Sci., 86, 450.
8. W.L. Jorgensen and E.M. Duffy (2000). Bioorg. Med. Chem. Letters, 10, 1155.
9. N. Bodor and M.J. Huang (1992). J. Pharm. Sci., 81, 954.
10. M.H. Abraham and J.E. Le (1999). J. Pharm. Sci., 88, 868.
11. P. Ruelle, C. Rey-Memert, M. Buchmann, H. Nam-Tran, U.W. Kesselring and P.L. Huyskens (1991). Pharm. Res., 8, 840.
12. A. Martin and P. Bustamante (1989). Anal. Real Acad. Farm., 55, 175.
13. A. Regosz, T. Pelplinska, P. Kowalsky and Z. Thiel (1992). Int. J. Pharm., 88, 437.
14. C. Hansch, J.E. Quinlan and G.L. Lawrence (1968). J. Org. Chem., 33, 347.
15. S.H. Yalkowsky (1999). Solubility and Solubilization in Aqueous Media. American Chemical Society and Oxford University Press, New York, pp. 61-70.
16. F. Martínez and A. Gómez (2001). J. Solution Chem., 30, 909.
17. R.M. Dannenfelser and S.H. Yalkowsky (1999). J. Pharm. Sci., 88, 722.
18. R.J. Prankerd and R.H. McKeown (1994). Int. J. Pharm., 112, 1.
19. A. Kristl (1999). J. Pharm. Sci., 88, 109.
20. N. Jain and S.H. Yalkowsky (2001). J. Pharm. Sci., 90, 234.
21. USP23 - NF18: The United States Pharmacopeia and the National Formulary (The United States Pharmacopeial Convention, Inc., Easton, U.S.A., 1995), 23rd Edn., pp. 1449-1467.
22. S.A. McCauley and H.G. Brittain (1995). In: H.G. Brittain (Ed.), Physical Characterization of Pharmaceutical Solids, Chap. 8, pp. 235-243. Marcel Dekker, Inc., New York.
23. J.W. Mauger, A.N. Paruta and R.J. Gerraugthty (1972). J. Pharm. Sci., 61, 94.
24. F. Martínez and J.H. Rojas (1999). Rev. Col. Cienc. Quim. Farm., 28, 45.
25. G. Best and N. Taylor (1961). The Physiological Basis of Medical Practice, 7th Edn., pp. 600-601. Williams and Williams, Baltimore, Md.
26. A.N. Martin, P. Bustamante and A.H.C. Chun (1993). Physical Pharmacy, Physical Chemical Principles in the Pharmaceutical Sciences, 4th Edn., Chap. 7, pp. 160-161. Lea and Febiger, Philadelphia.
27. P.H. Bell and R.O. Roblin (1942). J. Am. Chem. Soc., 64, 2905.
28. S. Budavari, M.J. O'Neil, A. Smith and P.E. Heckelman (1989). The Merck Index, an Encyclopedia of Chemicals, Drugs, and Biologicals, 11th Edn., p. 1403. Merck & Co., Inc., Rahway, N.J., U.S.A.
29. A.C. Moffat, J.V. Jackson, M.S. Moss and B. Widdop (1986). Clarke's Isolation and Identification of Drugs in Pharmaceuticals, Body Fluids, and Post-mortem Material, 2nd Edn., pp. 981-989. The Pharmaceutical Press, London.
30. E.C. Foernzler and A.N. Martin (1967). J. Pharm. Sci., 56, 608.
31. A.T. Florence and D. Attwood (1998). Physicochemical Principles of Pharmacy, 3rd Edn., Chap. 3, pp. 80-96. MacMillan Press Ltd, London.
32. S.S. Yang and J.K. Guillory (1972). J. Pharm. Sci., 61, 26.
33. C. Sunwoo and H. Eisen (1971). J. Pharm. Sci., 60, 238.
34. L. Maury, J. Rambaud, B. Pauvert, G. Berge, Y. Lasserre and M. Audian (1986). Farmaco Ed. Prat., 41, 25.
35. A. Kristl and G. Vesnaver (1995). J. Chem. Soc. Faraday Trans., 91, 995.
36. F. Martínez and A. Gómez (2001). Rev. Col. Quím., In press.