Antibacterial effect of some substituted tricyclic quinazolines and their synthetic precursors

Folia Microbiologica

Volumn 44, Issue 2, 1999, Pages 187-190

  Jantova S ^a   Spirkova K ^a   Stankovsky S ^a   Duchonova P ^a  

^a SLOVAK UNIVERSITY OF TECHNOLOGY   (Slovakia)

Author keywords

[No Author keywords available]

Indexed keywords

BACILLUS SUBTILIS; PSEUDOMONAS; PSEUDOMONAS AERUGINOSA;

ANTIINFECTIVE AGENT; QUINAZOLINE DERIVATIVE;

ARTICLE; BACILLUS SUBTILIS; BACTERIUM; CHEMISTRY; DRUG EFFECT; ESCHERICHIA COLI; MICROBIOLOGICAL EXAMINATION; PSEUDOMONAS AERUGINOSA; STAPHYLOCOCCUS AUREUS; SYNTHESIS;

ANTI-BACTERIAL AGENTS; BACILLUS SUBTILIS; BACTERIA; ESCHERICHIA COLI; MICROBIAL SENSITIVITY TESTS; PSEUDOMONAS AERUGINOSA; QUINAZOLINES; STAPHYLOCOCCUS AUREUS;

EID: 0041622212     PISSN: 00155632     EISSN: None     Source Type: Journal    
DOI: 10.1007/BF02816240     Document Type: Article

References (16)

1. ABDELMEGEED M.F., YASSIN S.M., ELSHANSHOUR A.R., ELBADAWI M.: Synthesis of some new chloro derivatives of quinazolino(4,3-β)quinazolin-8-one and s-tetrazolo (4,3-c)quinazoline with expected antifungicidal and antibacterial activities. Rev.Roum.Chim. 39, 189-197 (1994).
2. BODAJLA M., STANKOVSKÝ Š., ŠPIRKOVÁ K., JANTOVÁ S., HUDECOVÁ D.: Azolylquinazolines, synthesis and biological activity. Chem.Papers 48, 432-436 (1994).
3. ELZOHRY M.F., ELHAMED A., AHMED N., OMAR F.A., ABDALLA M.A.: Synthesis and antibacterial activity of certain quinoline and quinazoline derivatives containing sulfide and sulfone moieties. J.Chem.Technol.Biotechnol. 53, 329-336 (1992).
4. FARGHALY A.M., CHAABAN I., KHALIL M.A., BEKHIT A.A.: Nonsteroidal antiinflammatory agents. Synthesis of novel 2-pyrazolyl-4(3H)-quinazolines. Arch.Pharm. 323, 833-836 (1990).
5. FARGHALY A.M., MONSEN A., OMAR M.E., KHALIL M.A., GABER M.A.: Synthesis of 3-aryl-2-substituted-4(3H)-quinazolines as potential antimicrobial agents. Farmaco 45, 431-438 (1990).
6. GOTTASOVÁ R., KUBÍKOVÁ J., ČIPÁK L'.: Antibacterial effect of some 2,6-substituted 4-anilinoquinazolines. Folia Microbiol. 43, 679-682 (1998).
7. GURSOY A., KARALI N.: Synthesis and anticovulsant activity of new acylthiosemicarbazides and thiazolidones. Farmaco 50, 857-866 (1995).
8. JANTOVÁ S., HUDECOVÁ D., ŠPIRKOVÁ K., STANKOVSKÝ Š.: Structure-activity relationships of some 4 quinazolylthiosemicarbazides and their triazolo derivatives. Folia Microbiol. 39, 471-474 (1994).
9. JANTOVÁ S., HUDECOVÁ D., STANKOVSKÝ Š., ŠPIRKOVÁ K., RUŽEKOVÁ L'.: Antibacterial effect of substituted 4-quinazolylhydrazines and their arylhydrazones determined by modified microdilution method. Folia Microbiol. 40, 611-614 (1995).
10. JANTOVÁ S., BALÁŽ Š., STANKOVSKÝ Š., ŠPIRKOVÁ K., LUKÁČOVÁ V.: Relationships between the structure, cytotoxicity and hydrophobicity of quinazoline derivatives by quantitative structure-activity relationship. Folia Biol. 43, 83-89 (1997).
11. KUROGI Y., INOUE Y., TSUTSUMI K., NAKAMURA S., NAGAO K., YOSHITSUGU H., TSUDA Y.: Synthesis and hypolipidemis activities of novel 2-(4-((diethoxyphosphoryl)methyl)phenyl)quinazolines and 4(3H)-quinazolinones. J.Med.Chem. 39, 1433-1437 (1996).
12. PEET N.P., BAUGH L.E., LEWIS J.E., MATTHEWS E.H., OLBERDING E.L., SHAN D.N., SUNDER S.: Chemistry and antiallergic activity of 3-(1H-tetrazol-5-yl)-4-(3H)-quinazoline sodium-salt (MDL-427). Abstr.Pap.Amer.Chem.Soc. 192, 13 (1986).
13. POMARNACKA E., ANGIELSKI S., HOPPE A.: Derivatives of 4-chloro-5-sulfanoyl-benzoic acid. 8. Synthesis and diuretic activity of pyrazole (3,2-)quinazoline and 1-benzoylpyrazole derivatives. Acta Polon.Pharm. 41, 141-151 (1984).
14. SAKSENA R.K., KANT P.: Synthesis and antibacterial activity of azomethines and thiazolidinones derived from 2-phenyl-3-(p-aminodiphenyl)-4-quinazolones. J.Indian Chem.Soc. 61, 722-724 (1984).
15. ŠPIRKOVÁ K., STANKOVSKÝ Š., ZAHRADNÍK M.: Annelation to the quinazoline ring. Preparation and utilization of 3-quinazolyl-carboxylates in the synthesis of Fused Systems. Chem.Papers 51, 403-407 (1997).
16. TAKEMURA Y., JACKMAN A.L.: Folate-based thymidylate synthase inhibitors in cancer chemotherapy. Anti-Cancer Drugs 8, 3-16 (1997).