Synthesis and antituberculous activity of fluorinated 3-r-hydrazino-2-benzoylacrylates and their cyclization products

Pharmaceutical Chemistry Journal

Volumn 36, Issue 11, 2002, Pages 585-587

  Nosova, E V ^a   Kravchenko, M A ^b   Lipunova, G N ^a   Chasovskikh, O M ^a   Sokolov, V A ^b   Charushin, V N ^a  

^a URAL FEDERAL UNIVERSITY   (Russian Federation)

^b N N BLOKHIN NATIONAL MEDICAL RESEARCH CENTER OF ONCOLOGY   (Russian Federation)

Author keywords

[No Author keywords available]

Indexed keywords

2 [5' (2'',3'',5'',6'' TETRAFLUOROPHENYL) 4' ETHOXYCARBONYLPYRAZOL 1' YL]BENZOTHIAZOLE DERIVATIVE; 3 ETHOXYCARBONYL 5,7 DIFLUORO 6 (PYRROLIDIN 1 YL)BENZIMIDAZOL[1,2 A]PYRAZOLO[1,5 C]QUINAZOLINE; 3 HYDRAZIDOPYRIDINE 2 POLYFLUOROBENZOYLACRYLATIC ACID DERIVATIVE; BENZIMIDAZO[1,2 A]PYRAZOLO[1,5 C]QUINAZOLINE DERIVATIVE; BENZOXAZOLE DERIVATIVE; DIFLUOROBENZIMIDAZOLE DERIVATIVE; HYDRAZINO 2 BENZOYLACRYLATIC ACID DERIVATIVE; ISONIAZID; QUINOLINE DERIVED ANTIINFECTIVE AGENT; TUBERCULOSTATIC AGENT; UNCLASSIFIED DRUG;

ARTICLE; BACTERIAL STRAIN; CONTROLLED STUDY; CYCLIZATION; DRUG ACTIVITY; DRUG SCREENING; DRUG SYNTHESIS; FLUORINATION; MINIMUM INHIBITORY CONCENTRATION; MYCOBACTERIUM TUBERCULOSIS; NONHUMAN;

EID: 0038366919     PISSN: 0091150X     EISSN: None     Source Type: Journal    
DOI: 10.1023/A:1022657029905     Document Type: Article

References (7)

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