Simple and convenient preparation of new highly protected aziridines fused with pyrroline rings

Synlett

Volumn , Issue 7, 2003, Pages 995-996

  Attanasi, Orazio A ^a   Favi, Gianfranco ^a   Filippone, Paolino ^a   Stanovnik, Branko ^b   Svete, Jurij ^b  

^a UNIVERSITY OF URBINO   (Italy)

^b UNIVERSITY OF LJUBLJANA   (Slovenia)

Author keywords

1,2 diaza 1,3 butadienes; Aziridines; Bicyclic compounds; Michael additions; Regioselectivity

Indexed keywords

1,3 BUTADIENE DERIVATIVE; ACRYLIC ACID DERIVATIVE; AZIRIDINE DERIVATIVE; METHYL 2 BENZOYLAMINO 3 DIMETHYLAMINOPROPENOATE; PYRROLINE DERIVATIVE; UNCLASSIFIED DRUG;

ARTICLE; CHEMICAL REACTION; SYNTHESIS; TECHNIQUE;

EID: 0037899695     PISSN: 09365214     EISSN: None     Source Type: Journal    
DOI: None     Document Type: Article

References (19)

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11. For the synthesis and application of this and related compounds see: (a) Hvala, A.; Simonic, I.; Stanovnik, B.; Svete, J.; Tisler, M.; Zorz, L. Heterocycles 1988, 27, 903. (b) Èadež, Z.; Stanovnik, B.; Svete, J.; Tišler, M. Synthesis 1990, 70. (c) Stanovnik, B. J. Heterocycl. Chem. 1999, 36, 1581. (d) Stanovnik, B.; Svete, J. Synlett 2000, 1077. (e) Stanovnik, B.; Svete, J. Targets in Heterocyclic Systems 2000, 4, 105.
12. For the synthesis and application of this and related compounds see: (a) Hvala, A.; Simonic, I.; Stanovnik, B.; Svete, J.; Tisler, M.; Zorz, L. Heterocycles 1988, 27, 903. (b) Èadež, Z.; Stanovnik, B.; Svete, J.; Tišler, M. Synthesis 1990, 70. (c) Stanovnik, B. J. Heterocycl. Chem. 1999, 36, 1581. (d) Stanovnik, B.; Svete, J. Synlett 2000, 1077. (e) Stanovnik, B.; Svete, J. Targets in Heterocyclic Systems 2000, 4, 105.
13. For the synthesis and application of this and related compounds see: (a) Hvala, A.; Simonic, I.; Stanovnik, B.; Svete, J.; Tisler, M.; Zorz, L. Heterocycles 1988, 27, 903. (b) Èadež, Z.; Stanovnik, B.; Svete, J.; Tišler, M. Synthesis 1990, 70. (c) Stanovnik, B. J. Heterocycl. Chem. 1999, 36, 1581. (d) Stanovnik, B.; Svete, J. Synlett 2000, 1077. (e) Stanovnik, B.; Svete, J. Targets in Heterocyclic Systems 2000, 4, 105.
14. For the synthesis and application of this and related compounds see: (a) Hvala, A.; Simonic, I.; Stanovnik, B.; Svete, J.; Tisler, M.; Zorz, L. Heterocycles 1988, 27, 903. (b) Èadež, Z.; Stanovnik, B.; Svete, J.; Tišler, M. Synthesis 1990, 70. (c) Stanovnik, B. J. Heterocycl. Chem. 1999, 36, 1581. (d) Stanovnik, B.; Svete, J. Synlett 2000, 1077. (e) Stanovnik, B.; Svete, J. Targets in Heterocyclic Systems 2000, 4, 105.
15. 7: C, 55.53; H, 4.92; N, 10.79. Found: C, 55.45; H, 4.98; N, 10.66.
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