Halogenated boldine derivatives with enhanced monoamine receptor selectivity

Journal of Natural Products

Volumn 63, Issue 4, 2000, Pages 480-484

  Sobarzo Sánchez, Eduardo M ^a   Arbaoui, Jeannette ^b   Protais, Philippe ^b   Cassels, Bruce K ^a  

^a UNIVERSITY OF CHILE   (Chile)

^b UNIVERSITÉ DE ROUEN   (France)

Author keywords

[No Author keywords available]

Indexed keywords

BOLDINE;

ARTICLE; DRUG RECEPTOR BINDING; DRUG SELECTIVITY; DRUG STRUCTURE; HALOGENATION; LIGAND BINDING;

(R)-2,3,4,5-TETRAHYDRO-8-CHLORO-3-METHYL-5-PHENYL-1H-3-BENZAZEPIN-7-OL; ACETIC ACIDS; ANIMALS; ANTI-INFLAMMATORY AGENTS, NON-STEROIDAL; APORPHINES; BINDING, COMPETITIVE; BRAIN CHEMISTRY; CHLORIDES; NEOSTRIATUM; RACLOPRIDE; RADIOLIGAND ASSAY; RATS; RATS, WISTAR; RECEPTORS, BIOGENIC AMINE; RECEPTORS, DOPAMINE D1; RECEPTORS, DOPAMINE D2;

EID: 0037649227     PISSN: 01633864     EISSN: None     Source Type: Journal    
DOI: 10.1021/np990433j     Document Type: Article

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