Structure-based analysis of GPCR function: Conformational adaptation of both agonist and receptor upon leukotriene B4 binding to recombinant BLT1

Journal of Molecular Biology

Volumn 329, Issue 4, 2003, Pages 801-814

  Baneres, Jean Louis ^a   Martin, Aimée ^a   Hullot, Pierre ^a   Girard, Jean Pierre ^a   Rossi, Jean Claude ^a   Parello, Joseph ^a  

^a UNIV MONTPELLIER   (France)

Author keywords

Antagonistic effects; Bacterial expression; Conformational adaptation; Leukotriene B4 receptor; Recombinant GPCR

Indexed keywords

BINDING CELL SURFACE LEUKOTRIENE 1; CELL SURFACE RECEPTOR; G PROTEIN COUPLED RECEPTOR; LEUKOTRIENE B4; LEUKOTRIENE DERIVATIVE; MEMBRANE PROTEIN; RECEPTOR; TRYPTOPHAN DERIVATIVE; UNCLASSIFIED DRUG;

AGONIST; ARTICLE; COMPLEX FORMATION; CONJUGATION; CYTOPLASM; DNA HELIX; ENVIRONMENT; NONHUMAN; PRIORITY JOURNAL; PROTEIN CONFORMATION; STRUCTURE ANALYSIS;

BACTERIA (MICROORGANISMS); ESCHERICHIA COLI;

EID: 0037648337     PISSN: 00222836     EISSN: None     Source Type: Journal    
DOI: 10.1016/S0022-2836(03)00438-8     Document Type: Article

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