Synthesis and analgesic activity of stereoisomers of cis-fluoro-ohmefentanyl

Pharmazie

Volumn 58, Issue 5, 2003, Pages 300-302

  Yong, Zou ^b   Hao, Wu ^a   Weifang, Yuan ^a   Qiyuan, Dai ^a   Xinjian, Chen ^a   Wenqiao, Jin ^a   Youcheng, Zhu ^a  

^a SHANGHAI INSTITUTE OF MATERIA MEDICA   (China)

^b GUANGZHOU INSTITUTE OF CHEMISTRY   (China)

Author keywords

[No Author keywords available]

Indexed keywords

BETA HYDROXYMEFENTANYL; FLUOROHYDROXYMEFENTANYL; MORPHINE; MU OPIATE RECEPTOR; N [1 [2 HYDROXY 2 (4' FLUOROPHENYLETHYL)] 3 METHYL 4 PIPERIDYL] N PHENYLPROPANAMIDE; UNCLASSIFIED DRUG;

ANALGESIC ACTIVITY; ANIMAL EXPERIMENT; ARTICLE; BINDING KINETICS; CONTROLLED STUDY; DRUG CONFORMATION; DRUG DOSE; DRUG POTENCY; DRUG RECEPTOR BINDING; DRUG SYNTHESIS; HOT PLATE TEST; MOUSE; NONHUMAN; STEREOCHEMISTRY; STEREOISOMERISM; STRUCTURE ANALYSIS; X RAY ANALYSIS;

ANALGESICS, OPIOID; ANIMALS; CHEMISTRY, PHYSICAL; CRYSTALLOGRAPHY, X-RAY; FENTANYL; INDICATORS AND REAGENTS; MAGNETIC RESONANCE SPECTROSCOPY; MICE; MOLECULAR CONFORMATION; MORPHINE; STEREOISOMERISM; STRUCTURE-ACTIVITY RELATIONSHIP;

EID: 0037568184     PISSN: 00317144     EISSN: None     Source Type: Journal    
DOI: None     Document Type: Article

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