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-
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12244259004
-
-
note
-
3L form (Scheme 5) by the repulsive interaction between the protonated side chain and the diprotonated cyclen ring.
-
-
-
-
53
-
-
12244281452
-
-
note
-
+) (see the Supporting Information).
-
-
-
-
54
-
-
12244267635
-
-
note
-
3).
-
-
-
-
55
-
-
12244274280
-
-
note
-
1 in pH 7.4 buffer were estimated to be <7.
-
-
-
-
56
-
-
12244306851
-
-
note
-
2+ contents were determined to be 7.5 ± 0.2 mg/capsule and 2.0 ± 0.3 mg/tablet, values agreeing with the indicated values (7.5 mg/capsule and 2 mg/tablet, respectively).
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12244290249
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note
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1 caused colorless precipitations.
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76
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