In vivo and in vitro peripheral-type benzodiazepine receptor polymerization: Functional significance in drug ligand and cholesterol binding

Biochemistry

Volumn 42, Issue 15, 2003, Pages 4506-4519

  Delavoie, Franck ^a,b   Li, Hua ^a,c   Hardwick, Matthew ^a,d   Robert, Jean Claude ^b   Giatzakis, Christoforos ^a   Péranzi, Gabriel ^b   Yao, Zhi Xing ^a   Maccario, Jean ^b   Lacapère, Jean Jacques ^b   Papadopoulos, Vassilios ^a  

^a GEORGETOWN UNIVERSITY MEDICAL CENTER   (United States)

^b INSERM   (France)

^c Analytical Sciences   (United States)

^d JOHNS HOPKINS HOSPITAL   (United States)

Author keywords

[No Author keywords available]

Indexed keywords

CHOLESTEROL; CROSSLINKING; DRUG PRODUCTS; ELECTRON MICROSCOPY; OXYGEN; POLYMERIZATION; PROTEINS; ULTRAVIOLET RADIATION;

DRUG LIGANDS;

BIOCHEMISTRY;

BENZODIAZEPINE RECEPTOR; CHOLESTEROL; CHORIONIC GONADOTROPIN; FREE RADICAL; LIGAND; MONOMER; N SEC BUTYL 1 (2 CHLOROPHENYL) N METHYL 3 ISOQUINOLINECARBOXAMIDE; PERIPHERAL TYPE BENZODIAZEPINE RECEPTOR; POLYMER; REACTIVE OXYGEN METABOLITE; RECOMBINANT RECEPTOR; STEROID; TYROSINE DERIVATIVE; UNCLASSIFIED DRUG;

ANIMAL CELL; ARTICLE; BINDING AFFINITY; BREAST CANCER; CANCER CELL; CELL FUNCTION; CELL SPECIFICITY; CHOLESTEROL TRANSPORT; CONTROLLED STUDY; COVALENT BOND; CROSS LINKING; DRUG BINDING; DRUG RECEPTOR BINDING; ELECTRON MICROSCOPY; FREEZE FRACTURE; HUMAN; HUMAN CELL; IN VITRO STUDY; IN VIVO STUDY; LEYDIG CELL; LIGHT; MOLECULAR WEIGHT; MOUSE; NONHUMAN; PARTICLE SIZE; POLYACRYLAMIDE GEL ELECTROPHORESIS; PRIORITY JOURNAL; PROTEIN ANALYSIS; PROTEIN FUNCTION; PROTEIN POLYMERIZATION; PROTEOLIPOSOME; SPECTROSCOPY; STEROIDOGENESIS; ULTRAVIOLET RADIATION;

ANIMALS; CHOLESTEROL; DIMERIZATION; LIGANDS; MICE; PROTEIN BINDING; PROTEOLIPIDS; REACTIVE OXYGEN SPECIES; RECEPTORS, GABA-A; SPECTROPHOTOMETRY; ULTRAVIOLET RAYS;

ANIMALIA;

EID: 0037461325     PISSN: 00062960     EISSN: None     Source Type: Journal    
DOI: 10.1021/bi0267487     Document Type: Article

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