Synthesis of 1,4-diazines by ring expansion of 1,3-diazines

Journal of Organic Chemistry

Volumn 68, Issue 6, 2003, Pages 2334-2337

  Zaleska, Barbara ^a   Socha, Robert ^a   Karelus, Marcin ^a   Szneler, Edward ^a   Grochowski, Jacek ^b   Serda, Paweł ^b  

^a Regl Lab Physicochemical Analyses   (Poland)

^b JAGIELLONIAN UNIVERSITY   (Poland)

Author keywords

[No Author keywords available]

Indexed keywords

CARBOXYLIC ACIDS; DERIVATIVES; SYNTHESIS (CHEMICAL);

RING EXPANSION;

KETONES;

2 ANILINO 2 ETHOXY 3 OXOTHIOBUTANOIC ACID; BUTYRIC ACID; PIPERAZINE DERIVATIVE; QUINOXALINE DERIVATIVE; UNCLASSIFIED DRUG;

ARTICLE; CHIRALITY; CYCLIZATION; DRUG SYNTHESIS; MELTING POINT; NUCLEAR MAGNETIC RESONANCE SPECTROSCOPY; REACTION ANALYSIS; STEREOCHEMISTRY; X RAY DIFFRACTION;

EID: 0037459688     PISSN: 00223263     EISSN: None     Source Type: Journal    
DOI: 10.1021/jo026756t     Document Type: Article

References (18)

1. Dinsmore, C. J.; Hutchinson, J. H.; Williams, T. M. PCT Int. Appl. WO 99 09,985 (Cl. A61K31/495), Mar 4, 1999; GB Appl. 98/975, Jan 16, 1998.
2. Baudoin, B.; Dereu, N.; El-Ahmad, Y.; Jimonet, P.; Le Brun, A. PCT Int. Appl. WO 99 41,242 (Cl. C07D241/08), Aug 19, 1999; U.S. Appl. PV 81,602, Apr 14, 1998.
3. Anthony, N. J.; Ciccarone, T. M.; Dinsmore, C. J.; Gomez, R. P.; Williams, T. M.; Hartman, G. D. U.S. 5,856,326 (Cl. 514-252; A61 K31/ 495), Jan 5, 1999; U.S. Appl. 470,690, Jun 6, 1995.
4. Burkholder, T. P.; Kudlacz, M. E.; Le Tieu-Binh PCT Int. Appl. WO 96 28,441 (Cl. C07D403/06), Sep 19, 1996; U.S. Appl. 404,788, Mar 15, 1995.
5. Matsuo, M.; Hagiwara, D.; Miyake, H. PCT Int. Appl. WO 96 37,488 (Cl. C07D403/06), Nov 28, 1996; GB Appl 95/10,600, May 25, 1995.
6. Burkholder, T. P.; Le Tieu-Binh; Kudlacz, E. M. PCT Int. Appl. WO 96 32,385 (Cl. C07D241/04), Oct 17, 1996; U.S. Appl. 421,719, Apr 13, 1995.
7. Farmitalia, C. E. Jpn. Kokai Tokkyo Koho JP 61,167,686 [86,167,686] (Cl. C07D457/02), Jul 29, 1986; GB Appl. 85/1,078, Jan 16, 1985.
8. Schoenafinger, K.; Beyerle, R.; Schindler, W. Eur. Pat. Appl. 3,817,198, May 20, 1988.
9. Lumma, W. C.; Saari, W. S. U.S. 4,163,849 (Cl. 544-357; A61 K31/495), Aug 07, 1979; Appl. 887,693, Mar 17, 1978.
10. Shiozawa, A.; Inubushi, A.; Narita, K.; Shimada, K.; Hosono, M. Jpn. Kokai Tokkyo Koho JP 08 27,154 [9627,154] (Cl. C07D491/ 052), Jan 30, 1996; Appl. 94/198,080, Jul 20, 1994.
11. Kosinski, L.; Raymond E. Eur. Pat. Appl. EP 448,037 (Cl. C08K5/3492), Sep 25, 1991; U.S. Appl. 495,665, Mar 19, 1990.
12. Jennings, E. Can. Pat. Appl. CA 2,019,285 (Cl. C08L47/00), Dec 21, 1990; U.S. Appl. 369,573, Jun 21, 1989.
13. Kletecka, G.; Lai, J. T.; Son, P. N. U.S. 5,098,944 (Cl. 524-100; C08K5/3492), Mar 24, 1992; Appl. 580,727, Sep 11, 1990.
14. Hayakawa, H.; Morimoto, K.; Fujimoto, H. Jpn. Kokai Tokkyo, Koho JP 06,148,840 [94,148,840] (Cl. G03C7/407), May 27, 1994; Appl. 92/293,515, Oct 30, 1992.
15. Zaleska, B.; Socha, R.; Ciechanowicz-Rutkowska, M.; Pilati, T. Monatsh. Chem. 2000, 131, 1151-1160.
16. Zaleska, B.; Socha, R. Monatsh. Chem. 2000, 131, 1061-1066.
17. Zaleska, B.; Bazanek, T.; Socha, R.; Karelus, M.; Grochowski, J.; Serda, P. J. Org. Chem. 2002, 67, 4526-4529.
18. Belleney, J.; Bui, C.; Carriere, F. J. Magn. Reson Chem. 1990, 28, 606.