Brevetoxin derivatives act as partial agonists at neurotoxin site 5 on the voltage-gated Na+ channel

Brain Research

Volumn 959, Issue 1, 2003, Pages 120-127

  LePage, K T ^a   Baden, D G ^b   Murray, T F ^a  

^a UNIVERSITY OF GEORGIA   (United States)

^b UNIVERSITY OF NORTH CAROLINA WILMINGTON   (United States)

Author keywords

Brevetoxins; Voltage gated Na+ channel

Indexed keywords

BREVETOXIN; BREVETOXIN PBTX 1; BREVETOXIN PBTX 2; BREVETOXIN PBTX 3; BREVETOXIN PBTX 3ALPHA NAPHTHOYL; BREVETOXIN PBTX 3BETA NAPHTHOYL; NEUROTOXIN; SODIUM CHANNEL; UNCLASSIFIED DRUG;

ANIMAL CELL; ARTICLE; BINDING SITE; CALCIUM TRANSPORT; CELL CULTURE; CONCENTRATION RESPONSE; CONTROLLED STUDY; FLUORESCENCE; GRANULE CELL; NERVE CELL LESION; NERVE CELL NECROSIS; NONHUMAN; PRIORITY JOURNAL; RAT; SYNAPTIC TRANSMISSION;

ANIMALS; BINDING, COMPETITIVE; CALCIUM; CELLS, CULTURED; CEREBELLUM; DOSE-RESPONSE RELATIONSHIP, DRUG; MARINE TOXINS; NEURONS; NEUROTOXINS; OXOCINS; RATS; RATS, SPRAGUE-DAWLEY; SODIUM CHANNELS;

EID: 0037414734     PISSN: 00068993     EISSN: None     Source Type: Journal    
DOI: 10.1016/S0006-8993(02)03737-X     Document Type: Article

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