Supercritical fluids applications in the pharmaceutical industry

S.T.P. Pharma Sciences

Volumn 13, Issue 2, 2003, Pages 83-91

  Perrut, M ^a,b  

^a Lavipharm Laboratories   (United States)

^b Separex   (France)

Author keywords

Drug formulation; Extraction; Micronization; Purification; Supercritical fluid

Indexed keywords

ALCOHOL; ANTIBODY; BOVINE SERUM ALBUMIN; BUFFER; CARBON DIOXIDE; CATALASE; CELECOXIB; CERAMIDE; DIACYLGLYCEROL; DIMETHYL ETHER; ENZYME; EXCIPIENT; GLYCOLIPID; INSULIN; LACTASE; LIPID; MEVINOLIN; MONOACYLGLYCEROL; ORGANIC SOLVENT; POLOXAMER; POLYMER; POLYUNSATURATED FATTY ACID; SORBITOL; SURFACTANT; TOCOPHEROL; TRIACYLGLYCEROL; TRYPSIN; UNINDEXED DRUG; VALINE; WATER;

CHROMATOGRAPHY; CONTROLLED RELEASE FORMULATION; DRUG ACTIVITY; DRUG BIOAVAILABILITY; DRUG FORMULATION; DRUG INDUSTRY; DRUG SOLUBILITY; EXTRACTION; FRACTIONATION; MICROENCAPSULATION; PARTICLE SIZE; PURIFICATION; REVIEW; SUPERCRITICAL FLUID; TABLET; X RAY DIFFRACTION;

EID: 0037346659     PISSN: 11571489     EISSN: None     Source Type: Journal    
DOI: None     Document Type: Review

References (57)

1. STAHL E., QUIRIN K.-W., GERARD D. - Dense Gases for Extraction and Refining. - Springer-Verlag, 1987.
2. RIZVI S.S.H. - Supercritical Fluid Processing of Food and Biomaterials. - Ed. Blackie A&P, 1994.
3. KING M. B., LIST T. R. - Extraction of Natural Products Using Near-Critical Solvents. - Ed. Blackie A&P, 1996.
4. PERRUT M., SUBRA P. -In: Proc. 5th Meeting on Supercritical Fluids, Nice, 23-25 March 1998.
5. POLIAKOFF M., GEORGE M.W., HOWDLE S.M. - In: Proc. 6th Meeting on Supercritical Fluids, Nottingham, 10-13 April 1999.
6. PERRUT M., REVERCHON E. - In: Proc. 7th Meeting on Supercritical Fluids, Antibes, 6-8 December 2000.
7. BESNARD M., CANSELL F. - In: Proc. 8th Meeting on Supercritical Fluids, Bordeaux, 14-17 April 2002.
8. BRUNNER G. - Gas Extraction. - Springer Verlag, 1994.
9. PERRUT M. - Supercritical fluid applications: industrial developments and economic issues. - Ind. Eng. Chem. Res., 39, 4531-4535, 2000.
10. 2 for bone delipidation. - Biomaterials, 15, 650-656, 1994.
11. FAGES J., MATHON D., POIRIER B., AUTEFAGE A., LARZUL D., JEAN E., FRAYSSINET P. - Supercritical processing enhances viral safety and functionality of bone allografts. - In: Proc. 4th International Symposium on Supercritical Fluids, Sendai, S. Saito & K. Arai Eds., 1997, pp. 383-386.
12. PERRUT M., MAJEWSKI W., BREIVIK H. - Purifying polyunsaturated fatty acid glycerides. - US Patent 6,204,401, 2001.
13. BRUNNER G. - Gas Extraction. - Springer Verlag, 1994, pp. 278-290.
14. BRUNNER G. - Gas Extraction. - Springer Verlag, 1994, pp. 290-299.
15. DESCHAMPS F., MAJEWSKI W., CHAMINADE P., LAIMAY F., BAILLET A., PERRUT M. - A new concept in continuous supercritical fluid fractionation of lipids. - In: Proc. 7th Meeting on Supercritical Fluids, Antibes, M. Perrut & E. Reverchon Eds., 2000, pp. 573-578.
16. BRUNNER G. - Gas Extraction. - Springer Verlag, 1994, pp. 358-377.
17. CLAVIER J.Y., NICOUD R.M., PERRUT M. - A new efficient fractionation process: the simulated moving bed with supercritical eluent. - In: High Pressure Chemical Engineering, R. von Rohr & C. Trepp Eds., Elsevier, 1996, pp. 429-434.
18. DENET F., HAUCK W., NICOUD R.M., DI GIOVANI O., MAZZOTTI M., MORBIDELLI M. - Supercritical fluid simulated moving bed for chiral separation. - Proc. 7th Meeting on Supercritical Fluids, Antibes, M. Perrut & E. Reverchon Eds., 2000, pp. 821-826
19. HUTCHENSON K.W. - Organic chemical reactions and catalysis in supercritical fluid media. - In: Supercritical Fluid Technology in Materials Science and Engineering, Ya-Ping Sun Ed., Marcel Dekker, pp. 87-187.
20. HERKEY C. - Homogeneous catalysis in supercritical carbon dioxide. - In: Supercritical Fluid Technology in Materials Science and Engineering, Ya-Ping Sun Ed., Marcel Dekker, 2002, pp. 189-226.
21. GIDNER A., STENMARK L. - Recycling of precious metals by supercritical water oxidation. - In: High Pressure in Venice, Chemical Engineering Transactions, A. Bertucco Ed., AIDIC, 2002, pp. 753-758.
22. KOMPELLA U.D., KOUSHIK K. - Preparation of drug delivery systems using supercritical fluids. - Crit. Rev. Therapeutic Carrier Systems, 18 (2), 173-199, 2001.
23. JUNG J., PERRUT M. - Particle design using supercritical fluids: literature and patent review. - J. Supercritical Fluids, 20, 179-219, 2001.
24. PALAKODATY S., SLOAN R., KORDIKOWSKI A., YORK P. - Pharmaceutical and biological materials processing with supercritical fluids. - In: Supercritical Fluid Technology in Materials Science and Engineering, Ya-Ping Sun Ed. Marcel Dekker, 2002, pp. 439-490.
25. WEBER M., THIES M.C. - Understanding the RESS process. - In: Supercritical Fluid Technology in Materials Science and Engineering, Ya-Ping Sun Ed., Marcel Dekker, 2002, pp. 387-437.
26. PERRUT M., JUNG J., LEBOEUF F. - Process for preparation of amorphous particles. - French Patent Application, FR-02 05046, 2002.
27. PERRUT M., JUNG J., LEBOEUF F. - Solid state morphology of particles prepared by a supercritical fluid process. - In: High Pressure in Venice, Chemical Engineering Transactions. A. Bertucco Ed., AIDIC, Vol. 2., 2002, pp. 711-716.
28. LEBOEUF F., JUNG J., PERRUT M. - Process of manufacture of very fine particles from at least one water-soluble compound. - French Patent Application, FR-01.06403, 2001.
29. KRUKONIS V. - Method for drying water-borne materials. - US Patent Application, 60/359,665, 2002.
30. KNEZ Z. - Micronization of pharmaceuticals using supercritical fluids. - In: Proc. 7th Meeting on Supercritical Fluids, Antibes, M. Perrut & E. Reverchon Eds., 2000, pp. 21-26.
31. PERRUT M. - Process for encapsulation of fine particles in form of microcapsules. - French Patent FR 2 811 913, 2000, World Patent WO 02/05944, 2001.
32. DEBENEDETTI P., TOM J.W., YEO S.D., LIM G.B. - Application of supercritical fluids for the production of sustained delivery devices. - J. Controlled Release, 24, 27-44, 1993.
33. BENOIT J.P., ROLLAND H., THIES C., VAN DE VELDE V. - Method of coating particles and coated spherical particles. - Patent EP 0 706 821, 1996, WO 96/11055, 1996.
34. RICHARD J., RIBERO Dos SANTOS I., PECH B., THIES C., BENOIT J.P. - Coating protein particles with lipids using a novel supercritical fluid process. - 13th Int. Symp. on Micro-encapsulation, Angers, 2001.
35. FISCHER W., MULLER B.W. - Method and apparatus for the manufacture of a product having a substance embedded in a carrier. - Patent DE 3744329, 1987, US 5,043,280, 1991.
36. HANNA M., YORK P. - Method and apparatus for the formation of particles. - World Patent WO 95/01221, 1994.
37. CHOU Y.-H., TOMASKO D. - Gas crystallization of polymerpharmaceutical composite particles. - In: Proc. 4th International Symposium on Supercritical Fluids, Sendai, S. Saito & K. Arai Eds., 1997, pp. 55-57.
38. GHADERI R., ARTURSSON P., CALFORS J. - Preparation of biodegradable micro-particles using compressed anti-solvents for use in controlled release applications. - In: Proc. Int. Symp. Control. Rel. Bioact. Mater., 26, 1999, pp. 701-702.
39. ELVASSORE N., DAMINATO M., BERTUCCO A., CALICETI P. - Proteins and polymers processing by compressed gas anti-solvent techniques. - In: Proc. 6th Conference on Supercritical Fluids, Maiori, E. Reverchon Ed., 2001, pp. 313-318.
40. TAKI S., BADENS E., CHARBIT G. - Controlled-release system formed by supercritical anti-solvent coprecipitation of a herbicide and a biodegradable polymer. - J. Supercritical Fluids, 21, 61-70, 2001.
41. SUBRAMANIAM B., SAIM S., RAJEWSKI R.A., STELLA V. - Methods for a particle precipitation and coating using nearcritical and supercritical antisolvents. - US Patent 5,833,891, 1998.
42. BENOIT J.P., RICHARD J., THIES C. - Method for preparing microcapsules comprising active materials coated with a polymer and novel microcapsules in particular obtained according to the method. - Patent FR 2 753 639, 1996, WO 96/13136, 1998.
43. PERRUT M. - Process for collection and encapsulation of fine particles formed by a process using a fluid at supercritical pressure. - French Patent FR 2 803 539, 2000, World Patent WO 01/49407, 2001.
44. BUISSON B., FRANÇAIS E., LANNE J.Y., PERRUT M. - Film coating method for tablets. - French Patent FR-2800613, 1999.
45. WAKAYAMA H., FUKUSHIMA Y., TATSUDA N., KOJIMA Y., KAMIGAITO O., GOTO Y., NAGAKI S., SUZUKI K., SASAKI M., HAYASHI H., HIGUCHI K., SETOYAMA N. - Coated object and process for producing the same. - US Patent 6,194,650, 2001.
46. FILARDO G., GALIA A., PIERRO P. - Polymerisation of vinyl monomers in presence of solutes: new route for preparation of drug delivery sytems. - In: Proc. 7th Meeting on Supercritical Fluids, Antibes, M. Perrut & E. Reverchon Eds., 2000, pp. 161-166.
47. FILARDO G., GALIA A., PIERRO P. - Chain free radical dispersion copolymerisation of vinyl monomers in presence of solutes for the preparation of controlled release systems. - In: Proc. 6th Conf. on Supercritical Fluids, Maiori, E. Everchon Ed., 2001, pp. 221-224.
48. 2. A way of preparing controlled drug delivery systems. - Proc. 6th Meeting on Supercritical Fluids, Nottingham, Poliakoff M., George M.W., Howdle S.M. Eds., 1999, pp.101-107.
49. LANGELAAN H.C., LITJENS M.J.J., POORTIER E., HARMSEN P.F.H., VINGERHOEDS M.H. - Microencapsulation for food applications using supercritical fluids. - 13th International Symposium on Microencapsulation, Angers, 2001.
50. MAJEWSKI W., PERRUT M. - On-line direct impregnation of natural extracts. - In: Proc. 7th Meeting on Supercritical Fluids, Antibes, M. Perrut & E. Reverchon Eds., 2000, pp. 779-780.
51. WEIDNER E. - Powder generation by high pressure spray processes. - GVC-Fachausschuss «High Pressure Chemical Engineering», Karlsruhe (Germany), 1999, pp. 225-230.
52. CASTOR T.P., HONG G.T. - Critical fluid disruption of microbial cells. - In: Proc. 2nd International Symposium on Supercritical Fluids, Boston, M. Mc Hugh Ed., 1991, pp.139-142.
53. STAHL E., QUIRIN K.-W., GERARD D. - Dense Gases for Extraction and Refining. - Springer Verlag, 1987, pp. 218-221.
54. FOSTER N., DILLOW A., LANGER R., HRKACH J. - Supercritical fluid sterilization method. - US Patent 6,149,864, 2000.
55. CASTOR T.P., LANDER A.D., COSMAN M.D., D'ENTREMONT P.R., PELLETIER M.R. - Viral inactivation method using near critical, critical or supercritical fluids. - US Patent 5,877,005, 1999.
56. BOUZIDI A., PERRUT M., MAJEWSKI W. - Viral inactivation and delipidation of plasma and plasma products: new developments and experience of supercritical fluids. - In: Proc. 4th International Symposium on Supercritical Fluids, Sendaï, S. Saito & K. Arai Eds., 1997, Vol. A, pp. 387-390.
57. BOUZIDI A., MAJEWSKI W., HOBER D., PERRUT M. - Supercritical fluids improve tolerance and viral safety of fresh frozen plasma. - In: Proc. 5th Meeting on Supercritical Fluids, Nice, 1998, M. Perrut & E. Reverchon Eds., pp. 717-722.