A direct introduction of the mercaptoacetic acid unit into amino acid esters

Synthesis

Volumn , Issue 1, 2003, Pages 19-20

  Kraus, George A ^a   Bae, Jaehoon ^a   Choudhury, Prabir K ^a  

^a IOWA STATE UNIVERSITY   (United States)

Author keywords

Acylations; Amines; Amino acids; Combinatorial chemistry; Esters; Ligands; Thiols

Indexed keywords

AMINO ACIDS; ESTERS;

MERCAPTOACETIC ACID;

SYNTHESIS (CHEMICAL);

AMINO ACID DERIVATIVE; ESTER DERIVATIVE; THIOGLYCOLIC ACID;

ACYLATION; ARTICLE; CHEMICAL REACTION; ENVIRONMENTAL TEMPERATURE; NUCLEAR MAGNETIC RESONANCE SPECTROSCOPY; RACEMIC MIXTURE;

EID: 0037244843     PISSN: 00397881     EISSN: None     Source Type: Journal    
DOI: 10.1055/s-2003-36252     Document Type: Article

References (8)

1. (a) Baidoo, K. E.; Lever, S. Z. Bioconjugate Chem. 1990, 1, 132.
2. (b) Bryson, N.; Dewan, J. C.; Lister-James, J.; Jones, A. G.; Davison, A. Inorg. Chem. 1988, 27, 2154.
3. Bell, R. A.; Dickson, K. C.; Valliant, J. F. Can. J. Chem. 1999, 77, 146.
4. Higashiya, S.; Narizuka, S.; Konno, A.; Maeda, T.; Momota, K.; Fuchigami, T. J. Org. Chem. 1999, 64, 133.
5. The diphenylsilyl analog has been reported: Molt, K. R.; Hechenbleikner, I.; Homberg, O. A U.S. 3305573, 1967.
6. (a) Compound 3a: Johannsen, B.; Noll, B.; Leibnitz, G.; Reck, G.; Noll, St.; Spies, H. Radiochim. Acta 1993, 63, 133.
7. (b) Compound 3d: Davidovich, Y. A.; Semenova, N. N.; Babievskii, K. K.; Rogozhin, S. V. Izv. Akad. Nauk., Ser. Khim. 1986, 2139.
8. MTPA ester: Dale, J. A.; Mosher, H. S. J. Am. Chem. Soc. 1973, 95, 512.