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Volumn 18, Issue 1, 2003, Pages 71-79

Transdermal delivery of zidovudine: Effect of vehicles on permeation across rat skin and their mechanism of action

Author keywords

Thermogravimetric analysis; Transdermal permeation; Vehicle effect; Zidovudine

Indexed keywords

CELLS; DIFFUSION; SOLUBILITY; THERMOGRAVIMETRIC ANALYSIS; WATER;

EID: 0037243753     PISSN: 09280987     EISSN: None     Source Type: Journal    
DOI: 10.1016/S0928-0987(02)00242-7     Document Type: Article
Times cited : (92)

References (32)
  • 1
    • 0025118816 scopus 로고
    • Contributions of drug solubilization, partitioning, barrier disruption, and solvent permeation to the enhancement of skin permeation of various compounds with fatty acids and amines
    • Aungst B.J., Blake J.A., Hussain M.A. Contributions of drug solubilization, partitioning, barrier disruption, and solvent permeation to the enhancement of skin permeation of various compounds with fatty acids and amines. Pharm. Res. 7:1990;712-718.
    • (1990) Pharm. Res. , vol.7 , pp. 712-718
    • Aungst, B.J.1    Blake, J.A.2    Hussain, M.A.3
  • 2
    • 0023597397 scopus 로고
    • Mode of action of penetration enhancers in human skin
    • Barry B.W. Mode of action of penetration enhancers in human skin. J. Controlled Release. 6:1987;85-97.
    • (1987) J. Controlled Release , vol.6 , pp. 85-97
    • Barry, B.W.1
  • 3
    • 0025785005 scopus 로고
    • Examination of the effect of ethanol on human stratum corneum in vivo using infrared spectroscopy
    • Bommannan D., Potts R.O., Guy R.H. Examination of the effect of ethanol on human stratum corneum in vivo using infrared spectroscopy. J. Controlled Release. 16:1991;299-304.
    • (1991) J. Controlled Release , vol.16 , pp. 299-304
    • Bommannan, D.1    Potts, R.O.2    Guy, R.H.3
  • 4
    • 0018228927 scopus 로고
    • Factors influencing the percutaneous absorption of drugs
    • Chandrasekaran S.K., Shaw J.E. Factors influencing the percutaneous absorption of drugs. Curr. Probl. Dermatol. 7:1978;142-155.
    • (1978) Curr. Probl. Dermatol. , vol.7 , pp. 142-155
    • Chandrasekaran, S.K.1    Shaw, J.E.2
  • 5
    • 0032581199 scopus 로고    scopus 로고
    • Enhancement of percutaneous absorption of ketoprofen: Effect of vehicles and adhesive matrix
    • Cho Y.J., Choi H.-K. Enhancement of percutaneous absorption of ketoprofen: effect of vehicles and adhesive matrix. Int. J. Pharm. 169:1998;95-104.
    • (1998) Int. J. Pharm. , vol.169 , pp. 95-104
    • Cho, Y.J.1    Choi, H.-K.2
  • 7
    • 0023606009 scopus 로고
    • The effect of ethanol on the transport of B-estradiol and other permeants in hairless mouse skin. II. A new quantitative approach
    • Ghanem A.H., Rohr U., Higuchi W.I., Fox J.L., Liu P., Good W.R., Mahmoud H. The effect of ethanol on the transport of B-estradiol and other permeants in hairless mouse skin. II. A new quantitative approach. J. Controlled Release. 6:1987;75-83.
    • (1987) J. Controlled Release , vol.6 , pp. 75-83
    • Ghanem, A.H.1    Rohr, U.2    Higuchi, W.I.3    Fox, J.L.4    Liu, P.5    Good, W.R.6    Mahmoud, H.7
  • 8
    • 0033037654 scopus 로고    scopus 로고
    • Passive enhancement strategies in topical and transdermal drug delivery
    • Hadgraft J. Passive enhancement strategies in topical and transdermal drug delivery. Int. J. Pharm. 184:1999;1-6.
    • (1999) Int. J. Pharm. , vol.184 , pp. 1-6
    • Hadgraft, J.1
  • 9
    • 0002086622 scopus 로고
    • Physical chemical analysis of percutaneous absorption process from creams and ointments
    • Higuchi T. Physical chemical analysis of percutaneous absorption process from creams and ointments. J. Soc. Cosmet. Chem. 11:1960;85-97.
    • (1960) J. Soc. Cosmet. Chem. , vol.11 , pp. 85-97
    • Higuchi, T.1
  • 10
    • 0037133255 scopus 로고    scopus 로고
    • Transdermal drug delivery of imipramine hydrochloride. I. Effect of terpenes
    • Jain A.K., Thomas N.S., Panchagnula R. Transdermal drug delivery of imipramine hydrochloride. I. Effect of terpenes. J. Controlled Release. 79:2002;93-101.
    • (2002) J. Controlled Release , vol.79 , pp. 93-101
    • Jain, A.K.1    Thomas, N.S.2    Panchagnula, R.3
  • 11
    • 0033998593 scopus 로고    scopus 로고
    • Effect of application volume of ethanol-isopropyl myristate mixed solvent system on permeation of zidovudine and probenecid through rat skin
    • Jin Y., Seki T., Morimoto Y., Juni K. Effect of application volume of ethanol-isopropyl myristate mixed solvent system on permeation of zidovudine and probenecid through rat skin. Drug Dev. Ind. Pharm. 26:2000;193-198.
    • (2000) Drug Dev. Ind. Pharm. , vol.26 , pp. 193-198
    • Jin, Y.1    Seki, T.2    Morimoto, Y.3    Juni, K.4
  • 12
    • 0030017412 scopus 로고    scopus 로고
    • Permeation of zidovudine and probenecid from oily bases containing alcohols through rat skin
    • Jin Y., Toeda C., Kawaguchi T., Seki T., Juni K. Permeation of zidovudine and probenecid from oily bases containing alcohols through rat skin. Drug Dev. Ind. Pharm. 22:1996;653-658.
    • (1996) Drug Dev. Ind. Pharm. , vol.22 , pp. 653-658
    • Jin, Y.1    Toeda, C.2    Kawaguchi, T.3    Seki, T.4    Juni, K.5
  • 14
    • 0030058510 scopus 로고    scopus 로고
    • Transdermal delivery of dideoxynucleoside-type anti-HIV drugs. 2. The effect of vehicle and enhancer on skin permeation
    • Kim D.D., Chien Y.W. Transdermal delivery of dideoxynucleoside-type anti-HIV drugs. 2. The effect of vehicle and enhancer on skin permeation. J. Pharm. Sci. 85:1996;214-219.
    • (1996) J. Pharm. Sci. , vol.85 , pp. 214-219
    • Kim, D.D.1    Chien, Y.W.2
  • 15
    • 0033972550 scopus 로고    scopus 로고
    • Effect of vehicles and pressure sensitive adhesives on the permeation of tacrine across hairless mouse skin
    • Kim J., Cho Y., Choi H. Effect of vehicles and pressure sensitive adhesives on the permeation of tacrine across hairless mouse skin. Int. J. Pharm. 196:2000;105-113.
    • (2000) Int. J. Pharm. , vol.196 , pp. 105-113
    • Kim, J.1    Cho, Y.2    Choi, H.3
  • 16
    • 0026503846 scopus 로고
    • Short chain alkanols as transport enhancers for lipophilic and polar/ionic permeants in hairless mouse skin: Mechanism(s) of action
    • Kim Y.H., Ghanem A.H., Mahmoud H., Higuchi W.I. Short chain alkanols as transport enhancers for lipophilic and polar/ionic permeants in hairless mouse skin: mechanism(s) of action. Int. J. Pharm. 80:1992;17-31.
    • (1992) Int. J. Pharm. , vol.80 , pp. 17-31
    • Kim, Y.H.1    Ghanem, A.H.2    Mahmoud, H.3    Higuchi, W.I.4
  • 17
    • 0023091771 scopus 로고
    • Plasma and cerebrospinal fluid pharmacokinetics of 3′-azido-3′-deoxythymidine: A novel pyrimidine analog with potential application for the treatment of patients with AIDS and related diseases
    • Klecker R.W. Jr., Collins J.M., Yarchoan R., Thomas R., Jenkins J.F., Broder S., Myers C.E. Plasma and cerebrospinal fluid pharmacokinetics of 3′-azido-3′-deoxythymidine: a novel pyrimidine analog with potential application for the treatment of patients with AIDS and related diseases. Clin. Pharmacol. Ther. 41:1987;407-412.
    • (1987) Clin. Pharmacol. Ther. , vol.41 , pp. 407-412
    • Klecker R.W., Jr.1    Collins, J.M.2    Yarchoan, R.3    Thomas, R.4    Jenkins, J.F.5    Broder, S.6    Myers, C.E.7
  • 18
    • 12244265114 scopus 로고
    • Solvent mediates alternation of the stratum corneum
    • Knuston K., Krill S.L., Zang J. Solvent mediates alternation of the stratum corneum. J. Controlled Release. 11:1990;93-103.
    • (1990) J. Controlled Release , vol.11 , pp. 93-103
    • Knuston, K.1    Krill, S.L.2    Zang, J.3
  • 19
    • 0033045943 scopus 로고    scopus 로고
    • Safety and pharmacokinetics of abacavir (1592U89) following oral administration of escalating single doses in human immunodeficiency virus type 1-infected adults
    • Kumar P.N., Sweet D.E., McDowell J.A., Symonds W., Lou Y., Hetherington S., LaFon S. Safety and pharmacokinetics of abacavir (1592U89) following oral administration of escalating single doses in human immunodeficiency virus type 1-infected adults. Antimicrob. Agents Chemother. 43:1999;603-608.
    • (1999) Antimicrob. Agents Chemother. , vol.43 , pp. 603-608
    • Kumar, P.N.1    Sweet, D.E.2    McDowell, J.A.3    Symonds, W.4    Lou, Y.5    Hetherington, S.6    LaFon, S.7
  • 20
    • 0025032458 scopus 로고
    • Percutaneous absorption enhancement of an ionic molecule by ethanol-water systems in human skin
    • Kurihara-Bergstrom T., Knutson K., DeNoble L.J., Goates C.Y. Percutaneous absorption enhancement of an ionic molecule by ethanol-water systems in human skin. Pharm. Res. 7:1990;762-766.
    • (1990) Pharm. Res. , vol.7 , pp. 762-766
    • Kurihara-Bergstrom, T.1    Knutson, K.2    DeNoble, L.J.3    Goates, C.Y.4
  • 21
    • 0024458218 scopus 로고
    • Infrared spectroscopic study of ethanol-induced changes in rat liver plasma membrane
    • Lewis E.N., Levin I.W., Steer C.J. Infrared spectroscopic study of ethanol-induced changes in rat liver plasma membrane. Biochim. Biophys. Acta. 986:1989;161-166.
    • (1989) Biochim. Biophys. Acta , vol.986 , pp. 161-166
    • Lewis, E.N.1    Levin, I.W.2    Steer, C.J.3
  • 22
    • 85056062854 scopus 로고    scopus 로고
    • Experimental methods to evaluate diffusion coefficients and investigate transport processes of pharmaceutical interest
    • G.L. Amidon, P.I. Lee, & E.M. Topp. New York: Marcel Dekker
    • Mauger J.W. Experimental methods to evaluate diffusion coefficients and investigate transport processes of pharmaceutical interest. Amidon G.L., Lee P.I., Topp E.M. Transport Processes in Pharmaceutical Systems. 2000;87-108 Marcel Dekker, New York.
    • (2000) Transport Processes in Pharmaceutical Systems , pp. 87-108
    • Mauger, J.W.1
  • 23
    • 0021017126 scopus 로고
    • Vehicle effect on topical drug delivery. II. Concurrent skin transport of drugs and vehicle components
    • Mollgaard B., Hoelgaard A. Vehicle effect on topical drug delivery. II. Concurrent skin transport of drugs and vehicle components. Acta Pharm. Suec. 20:1983;443-450.
    • (1983) Acta Pharm. Suec. , vol.20 , pp. 443-450
    • Mollgaard, B.1    Hoelgaard, A.2
  • 24
    • 0031416704 scopus 로고    scopus 로고
    • Transdermal delivery of azidothymidine (AZT) through rat skin ex-vivo
    • Panchagnula R., Patel J.R. Transdermal delivery of azidothymidine (AZT) through rat skin ex-vivo. Pharm. Sci. 3:1997;83-87.
    • (1997) Pharm. Sci. , vol.3 , pp. 83-87
    • Panchagnula, R.1    Patel, J.R.2
  • 25
    • 0035927221 scopus 로고    scopus 로고
    • Transdermal delivery of naloxone: Effect of water, propylene glycol, ethanol and their binary combinations on permeation through rat skin
    • Panchagnula R., Salve P.S., Thomas N.S., Jain A.K., Ramarao P. Transdermal delivery of naloxone: effect of water, propylene glycol, ethanol and their binary combinations on permeation through rat skin. Int. J. Pharm. 219:2001;95-105.
    • (2001) Int. J. Pharm. , vol.219 , pp. 95-105
    • Panchagnula, R.1    Salve, P.S.2    Thomas, N.S.3    Jain, A.K.4    Ramarao, P.5
  • 26
    • 0015454316 scopus 로고
    • Diffusion of drugs from topical vehicles: An analysis of vehicle effects
    • Poulsen B.J. Diffusion of drugs from topical vehicles: an analysis of vehicle effects. Adv. Biol. Skin. 12:1972;495-509.
    • (1972) Adv. Biol. Skin , vol.12 , pp. 495-509
    • Poulsen, B.J.1
  • 27
    • 33845549925 scopus 로고
    • Lipid chain-length and temperature-dependence of ethanol phsphatidylcholine interactions
    • Rowe E.S. Lipid chain-length and temperature-dependence of ethanol phsphatidylcholine interactions. Biochemistry. 22:1983;3299-3305.
    • (1983) Biochemistry , vol.22 , pp. 3299-3305
    • Rowe, E.S.1
  • 28
    • 0022424889 scopus 로고
    • Thermodynamic reversibility of phase transitions. Specific effects of alcohols on phosphatidylcholines
    • Rowe E.S. Thermodynamic reversibility of phase transitions. Specific effects of alcohols on phosphatidylcholines. Biochim. Biophys. Acta. 813:1985;321-330.
    • (1985) Biochim. Biophys. Acta , vol.813 , pp. 321-330
    • Rowe, E.S.1
  • 29
    • 0022619484 scopus 로고
    • In vitro percutaneous absorption experiments. A technique for production of intact epidermal membrane from rat skin
    • Scott R.C., Walker M., Dugard P.H. In vitro percutaneous absorption experiments. A technique for production of intact epidermal membrane from rat skin. J. Soc. Cosmet. Chem. 37:1986;35-41.
    • (1986) J. Soc. Cosmet. Chem. , vol.37 , pp. 35-41
    • Scott, R.C.1    Walker, M.2    Dugard, P.H.3
  • 31
    • 0035991649 scopus 로고    scopus 로고
    • Prediction of steady-state skin permeabilities of polar and nonpolar permeants across excised pig skin based on measurements of transient diffusion: Characterization of hydration effects on the skin porous pathway
    • Tang H., Blankschtein D., Langer R. Prediction of steady-state skin permeabilities of polar and nonpolar permeants across excised pig skin based on measurements of transient diffusion: Characterization of hydration effects on the skin porous pathway. J. Pharm. Sci. 91:2002;1891-1907.
    • (2002) J. Pharm. Sci. , vol.91 , pp. 1891-1907
    • Tang, H.1    Blankschtein, D.2    Langer, R.3
  • 32
    • 0024245440 scopus 로고
    • Membrane-solvent-solute interaction in a model permeation system
    • Twist J.N., Zatz J.L. Membrane-solvent-solute interaction in a model permeation system. J. Pharm. Sci. 77:1988;536-540.
    • (1988) J. Pharm. Sci. , vol.77 , pp. 536-540
    • Twist, J.N.1    Zatz, J.L.2


* 이 정보는 Elsevier사의 SCOPUS DB에서 KISTI가 분석하여 추출한 것입니다.