SCOPUS 정보 검색 플랫폼

Volumn 45, Issue 9, 2002, Pages 1845-1852

5′-deoxy congeners of 9-(3-amido-3-deoxy-β-D-xylofuranosyl)-N6-cyclopentyladenine: New adenosine A1 receptor antagonists and inverse agonists

(10) Van Calenbergh, Serge a Link, Andreas b Fujikawa, Shelly c De Ligt, Rianne A F c Vanheusden, Veerle a Golisade, Abolfasl b Blaton, Norbert M d Rozenski, Jef e IJzerman, Adriaan P c Herdewijn, Piet a,e

a GHENT UNIVERSITY (Belgium)

b UNIVERSITY OF HAMBURG (Germany)

c LEIDEN UNIVERSITY (Netherlands)

d UNIVERSITY OF LEUVEN (Belgium)

e REGA INSTITUTE FOR MEDICAL RESEARCH (Belgium)

Author keywords

[No Author keywords available]

Indexed keywords

9 (3 AMIDO 3 DEOXY BETA DEXTRO XYLOFURANOSYL) N6 CYCLOPENTYLADENINE; ADENINE DERIVATIVE; ADENOSINE A1 RECEPTOR ANTAGONIST; ADENOSINE RECEPTOR; ADENOSINE RECEPTOR STIMULATING AGENT; UNCLASSIFIED DRUG; CYCLIC AMP; DEOXYADENOSINE DERIVATIVE;

ARTICLE; CYTOTOXICITY; HIGH PERFORMANCE LIQUID CHROMATOGRAPHY; LIGAND BINDING; MOLECULAR INTERACTION; PROTON NUCLEAR MAGNETIC RESONANCE; RECEPTOR AFFINITY; STRUCTURE ACTIVITY RELATION; STRUCTURE ANALYSIS; SYNTHESIS; X RAY ANALYSIS; X RAY CRYSTALLOGRAPHY; ANIMAL; BINDING COMPETITION; BIOSYNTHESIS; CHEMICAL STRUCTURE; CHEMISTRY; CHO CELL; DRUG ANTAGONISM; DRUG POTENTIATION; HAMSTER; HUMAN; IN VITRO STUDY; METABOLISM; RADIOASSAY; RAT;

ANIMALS; BINDING, COMPETITIVE; CHO CELLS; CRICETINAE; CRYSTALLOGRAPHY, X-RAY; CYCLIC AMP; DEOXYADENOSINES; HUMANS; MODELS, MOLECULAR; RADIOLIGAND ASSAY; RATS; RECEPTORS, PURINERGIC P1; STRUCTURE-ACTIVITY RELATIONSHIP;

EID: 0037171438 PISSN: 00222623 EISSN: None Source Type: Journal
DOI: 10.1021/jm0110439 Document Type: Article

Times cited : (15)

References (21)

1
- 0033545638
- 1 receptor antagonist with potent diuretic activity
- (1999) J. Med. Chem. , vol.42 , pp. 779-783
- Akahane, A.¹ Katayama, H.² Mitsunaga, T.³ Kato, T.⁴ Kinoshita, T.⁵ Kita, Y.⁶ Kusunoki, T.⁷ Terai, T.⁸ Yoshida, K.⁹ Shiokawa, Y.¹⁰

2
- 0027097122
- Adenosine A1 antagonists; A new therapeutic approach to cognitive deficits and acute renal failure
- (1992) Drug News Perspect. , vol.5 , pp. 587-591
- Suzuki, F.¹

3
- 0008920845
- Respirable Antisense Oligonucleotides (RASONS)
- Crooke, S. T., Ed.; Marcel Dekker: New York
- (2001) Antisense Drug Technology. Principles, Strategies, and Applications , pp. 679-685
- Nyce, J.W.¹

4
- 0033524916
- 1 adenosine receptor
- and references therein
- (1999) J. Biol. Chem. , vol.274 , pp. 3617-3621
- Rivkees, S.A.¹ Barbhaiya, H.² IJzerman, A.P.³

5
- 0022629566
- Ribose-modified adenosine analogues as adenosine receptor agonists
- (1986) J. Med. Chem. , vol.29 , pp. 346-353
- Taylor, M.D.¹ Moos, W.H.² Szotek, D.S.³ Patt, W.C.⁴ Badger, E.W.⁵ Bristol, J.A.⁶ Bruns, R.F.⁷ Heffner, T.G.⁸ Mertz, T.E.⁹

6
- 0028859493
- Ribose-modified adenosine analogues as potential partial agonists for the adenosine receptor
- (1995) J. Med. Chem. , vol.38 , pp. 4000-4006
- Van der Wenden, E.M.¹ Von Frijtag Drabbe Künzel, J.K.² Mathôt, R.A.A.³ Danhof, M.⁴ IJzerman, A.P.⁵ Soudijn, W.⁶

7
- 0023723881
- 6-cyclohexyladenosine: An adenosine derivative with antagonist properties at adenosine receptors
- (1988) Eur. J. Pharmacol. , vol.156 , pp. 157-160
- Lohse, M.J.¹ Klotz, K.-N.² Diekmann, E.³ Friedrich, K.⁴ Schwabe, U.⁵

8
- 0031558658
- 1 receptor antagonists
- (1997) J. Med. Chem. , vol.40 , pp. 3765-3772
- Van Calenbergh, S.¹ Von Frijtag Drabbe Künzel, J.K.² Blaton, N.M.³ Peeters, O.M.⁴ Rozenski, J.⁵ Van Aerschot, A.⁶ De Bruyn, A.⁷ De Keukeleire, D.⁸ IJzerman, A.P.⁹ Herdewijn, P.¹⁰

9
- 0026009348
- 6-cyclopentyl-5′-deoxyadenosine
- (1991) Nucleosides Nucleotides , vol.10 , pp. 1477-1483
- Davidson, J.G.¹ Fiore, P.J.²

10
- 0014820904
- Halo sugar nucleosides. I. Iodination of the primary hydroxyl groups of nucleosides with methyltriphenoxyphosphonium iodide
- (1970) J. Org. Chem. , vol.35 , pp. 2319-2326
- Verheyden, J.P.H.¹ Moffatt, J.G.²

11
- 0015922292
- Reactions of 2-acyloxyisobutyryl halides with nucleosides. II. Reactions of adenosine
- (1973) J. Am. Chem. Soc. , vol.95 , pp. 4025-4030
- Russel, A.F.¹ Greenberg, S.² Moffatt, J.G.³

12
- 0022374989
- Regiospecific and stereoselective conversion of ribonucleotides to 3′-deoxynucleotides. A high yield three-stage synthesis of cordyceptin from adenosine
- (1985) Tetrahedron Lett. , vol.26 , pp. 4295-4298
- Hansske, F.¹ Robins, M.J.²

13
- 0000246280
- Carbon-carbon bond-forming methods on solid support. Utilization of Kenner's "safety-catch" linker
- (1994) J. Am. Chem. Soc. , vol.116 , pp. 11171-11172
- Backes, B.J.¹ Ellman, J.A.²

14
- 0001176887
- Activation method to prepare a highly reactive acylsulfonamide "safety-catch" linker for solid-phase synthesis
- (1996) J. Am. Chem. Soc. , vol.118 , pp. 3055-3056
- Backes, B.J.¹ Virgilio, A.A.² Ellman, J.A.³

15
- 0031777856
- 1 adenosine receptors stably expressed in Chinese hamster ovary cells
- (1998) Mol. Pharmacol. , vol.53 , pp. 886-892
- Shryock, J.C.¹ Ozeck, M.J.² Belardinelli, L.³

16
- 0024438160
- 6-(-aminoalkyl)-adenosines on adenosine receptor affinity and intrinsic activity
- (1989) Eur. J. Pharmacol. , vol.172 , pp. 185-193
- Pirovano, I.M.¹ IJzerman, A.P.² Van Galen, P.J.M.³ Soudijn, W.⁴

17
- 0024854441
- 2 receptors in rat brain
- (1989) J. Pharmacol. Exp. Ther. , vol.251 , pp. 888-893
- Jarvis, M.F.¹ Schultz, R.² Hutchison, A.J.³ Hoi Do, U.⁴ Sills, M.⁵ Williams, M.⁶

18
- 0028179205
- 3 adenosine receptor
- (1994) Mol. Pharmacol. , vol.45 , pp. 978-982
- Olah, M.E.¹ Gallo-Rodriguez, C.² Jacobson, K.A.³ Stiles, G.⁴

19
- 0028337831
- 3 adenosine receptor
- (1994) Mol. Pharmacol. , vol.45 , pp. 1101-1111
- Van Galen, P.J.M.¹ Van Bergen, A.² Gallo-Rodriguez, C.³ Melman, N.⁴ Olah, M.E.⁵ IJzerman, A.P.⁶ Stiles, G.L.⁷ Jacobson, K.A.⁸

20
- 0000604488
- SIR92 - A program for automatic solution of crystal structures by direct methods
- (1994) J. Appl. Crystallogr. , vol.27 , pp. 435
- Altomare, A.¹ Cascarano, G.² Giacovazzo, C.³ Guagliardi, A.⁴

21
- 0004150157
- University of Göttingen: Germany
- (1993) SHELXL97, Program for the Refinement of Crystal Structures
- Sheldrick, G.M.¹

* 이 정보는 Elsevier사의 SCOPUS DB에서 KISTI가 분석하여 추출한 것입니다.