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Volumn 12, Issue 6, 2002, Pages 879-881
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Dermorphin and deltorphin heptapeptide analogues: Replacement of Phe residue by Dmp greatly improves opioid receptor affinity and selectivity
a a a a a a |
Author keywords
[No Author keywords available]
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Indexed keywords
2,6 DIMETHYLPHENYLALANINE;
DELTA OPIATE RECEPTOR;
DELTORPHIN;
DERMORPHIN DERIVATIVE;
HEPTAPEPTIDE;
MU OPIATE RECEPTOR;
OPIATE RECEPTOR;
PHENYLALANINE DERIVATIVE;
UNCLASSIFIED DRUG;
2',6' DIMETHYLPHENYLALANINE;
2',6'-DIMETHYLPHENYLALANINE;
DERMORPHIN;
DRUG DERIVATIVE;
NARCOTIC ANALGESIC AGENT;
OLIGOPEPTIDE;
OPIATE PEPTIDE;
PHENYLALANINE;
ANIMAL TISSUE;
ARTICLE;
BIOASSAY;
CONTROLLED STUDY;
DRUG POTENCY;
DRUG PROTEIN BINDING;
DRUG RESEARCH;
DRUG SYNTHESIS;
IN VITRO STUDY;
NONHUMAN;
RECEPTOR AFFINITY;
ANIMAL;
CHEMISTRY;
DRUG ANTAGONISM;
DRUG EFFECT;
GUINEA PIG;
IC 50;
METABOLISM;
MUSCLE CONTRACTION;
PHYSIOLOGY;
PROTEIN BINDING;
SMOOTH MUSCLE;
STRUCTURE ACTIVITY RELATION;
SYNTHESIS;
ANALGESICS, OPIOID;
ANIMALS;
GUINEA PIGS;
INHIBITORY CONCENTRATION 50;
MUSCLE CONTRACTION;
MUSCLE, SMOOTH;
OLIGOPEPTIDES;
OPIOID PEPTIDES;
PHENYLALANINE;
PROTEIN BINDING;
RECEPTORS, OPIOID;
STRUCTURE-ACTIVITY RELATIONSHIP;
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EID: 0037170786
PISSN: 0960894X
EISSN: None
Source Type: Journal
DOI: 10.1016/S0960-894X(02)00035-5 Document Type: Article |
Times cited : (16)
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References (27)
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