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Bioorganic and Medicinal Chemistry Letters

Volumn 12, Issue 16, 2002, Pages 2113-2116

Pyrrolylquinoxalinediones carrying a piperazine residue represent highly potent and selective ligands to the homomeric kainate receptor GluR5

(7) Lubisch, W a Behl, B a Henn, C a Hofmann, H P a Reeb, J a Regner, F a Vierling, M a

a ABBOTT GMBH AND CO KG (Germany)

Author keywords

[No Author keywords available]

Indexed keywords

KAINIC ACID RECEPTOR; LIGAND; PIPERAZINE; PROTEIN GLUR5; PROTEIN GLUR6; PROTEIN GLUR7; PYRROLYLQUINOXALINEDIONE; RECOMBINANT PROTEIN; UNCLASSIFIED DRUG; ALPHA AMINO 3 HYDROXY 5 METHYL 4 ISOXAZOLEPROPIONIC ACID; AMINO ACID RECEPTOR BLOCKING AGENT; GLUR5 KAINATE RECEPTOR; N METHYLASPARTIC ACID; PIPERAZINE DERIVATIVE; QUINOXALINE DERIVATIVE;

ARTICLE; BINDING AFFINITY; CHEMICAL ANALYSIS; PROTEIN BINDING; ANIMAL; BINDING SITE; CHEMICAL STRUCTURE; CHEMICALLY INDUCED DISORDER; CHEMISTRY; DOSE RESPONSE; DRUG ANTAGONISM; ENZYME SPECIFICITY; METABOLISM; MOUSE; SEIZURE; STRUCTURE ACTIVITY RELATION; SYNTHESIS;

ALPHA-AMINO-3-HYDROXY-5-METHYL-4-ISOXAZOLEPROPIONIC ACID; ANIMALS; BINDING SITES; DOSE-RESPONSE RELATIONSHIP, DRUG; EXCITATORY AMINO ACID ANTAGONISTS; LIGANDS; MICE; MOLECULAR STRUCTURE; N-METHYLASPARTATE; PIPERAZINES; QUINOXALINES; RECEPTORS, KAINIC ACID; SEIZURES; STRUCTURE-ACTIVITY RELATIONSHIP; SUBSTRATE SPECIFICITY;

EID: 0037135991 PISSN: 0960894X EISSN: None Source Type: Journal
DOI: 10.1016/S0960-894X(02)00335-9 Document Type: Article

Times cited : (9)

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