SCOPUS 정보 검색 플랫폼

Volumn 45, Issue 17, 2002, Pages 3579-3582

Synthesis, biological properties, and molecular modeling investigation of the first potent, selective, and water-soluble human A3 adenosine receptor antagonist

(11) Maconi, Anna a Moro, Stefano a Pastorin, Giorgia a Da Ros, Tatiana a Spalluto, Giampiero b Gao, Zhan guo b Jacobson, Kenneth A c Baraldi, Pier Giovanni c Cacciari, Barbara c Varani, Katia d Andrea Borea, Pier c

a UNIVERSITY OF TRIESTE (Italy)

b NATIONAL INSTITUTE OF DIABETES AND DIGESTIVE AND KIDNEY DISEASES (United States)

c UNIVERSITY OF FERRARA (Italy)

d UNIVERSITY OF PADOVA (Italy)

Author keywords

[No Author keywords available]

Indexed keywords

5 [[(4 PYRIDYL)AMINO]CARBONYL]AMINO 8 METHYL 2 (2 FURYL)PYRAZOLO[4,3 E] 1,2,4 TRIAZOLO[1,5 C]PYRIMIDINE; ADENOSINE A3 RECEPTOR ANTAGONIST; UNCLASSIFIED DRUG;

ANIMAL CELL; ARTICLE; BINDING AFFINITY; CHO CELL; DRUG ACTIVITY; DRUG BINDING; DRUG POTENCY; DRUG SELECTIVITY; DRUG SOLUBILITY; DRUG STRUCTURE; DRUG SYNTHESIS; MOLECULAR MODEL; NONHUMAN;

ANIMALS; CELL LINE; CRICETINAE; HUMANS; MODELS, MOLECULAR; PYRIMIDINES; RECEPTOR, ADENOSINE A3; RECEPTORS, PURINERGIC P1; SOLUBILITY; STRUCTURE-ACTIVITY RELATIONSHIP; TRIAZOLES;

EID: 0037103340 PISSN: 00222623 EISSN: None Source Type: Journal
DOI: 10.1021/jm020974x Document Type: Article

Times cited : (74)

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