SCOPUS 정보 검색 플랫폼

Volumn 58, Issue 11, 2002, Pages 2147-2153

Regioselective 4-amino-de-chlorination of trichloro- and dichloro-pyrimidines with N-sodium carbamates

(8) Montebugnoli, Dario a Bravo, Pierfrancesco a,b Corradi, Eleonora a Dettori, Giovanna c Mioskowski, Charles c Volonterio, Alessandro b Wagner, Alain c Zanda, Matteo a

a POLITECNICO DI MILANO (Italy)

b CNR (Italy)

c UNIVERSITÉ DE STRASBOURG (France)

Author keywords

Amination; Carbamates; Pyrimidines; Regioselection

Indexed keywords

2,4 DICHLOROPYRIMIDINE; 2,4,6 TRICHLOROPYRIMIDINE; 4 N ALKOXYCARBONYLAMINO 2,6 CHLOROPYRIMIDINE; 4 N ALKOXYCARBONYLAMINO 2,6 DICHLOROPYRIMIDINE; 4,6 DICHLOROPYRIMIDINE; CARBAMIC ACID DERIVATIVE; PYRIMIDINE DERIVATIVE; UNCLASSIFIED DRUG;

ARTICLE; CHEMICAL STRUCTURE; DECHLORINATION; PRIORITY JOURNAL; PROTON NUCLEAR MAGNETIC RESONANCE; STRUCTURE ANALYSIS; SYNTHESIS; X RAY DIFFRACTION;

EID: 0037060945 PISSN: 00404020 EISSN: None Source Type: Journal
DOI: 10.1016/S0040-4020(02)00084-4 Document Type: Article

Times cited : (12)

References (49)

1
- 0029915494
- (1996) J. Med. Chem. , vol.39 , pp. 4358-4360
- Chen, C.¹ Dagnino Jr., R.² De Souza, E.B.³ Grigoriadis, D.E.⁴ Huang, C.Q.⁵ Kim, K.-I.⁶ Liu, Z.⁷ Moran, T.⁸ Webb, T.R.⁹ Whitten, J.P.¹⁰ Xie, Y.F.¹¹ McCarthy, J.R.¹²

2
- 0023943817
- and references therein
- (1987) Farmaco, Ed. Sci. , vol.43 , pp. 277-291
- Maggiali, C.¹ Morini, G.² Mossini, F.³ Morini, G.⁴ Barocelli, E.⁵ Impicciatore, M.⁶

3
- 0033529014
- (1999) J. Med. Chem. , vol.42 , pp. 1481-1500
- Williams, M.¹ Kowaluk, E.A.² Arneric, S.P.³

4
- 0031694835
- (1998) Bioorg. Med. Chem. , vol.6 , pp. 1057-1068
- Ban, M.¹ Taguchi, H.² Katsushima, T.³ Aoki, S.⁴ Watanabe, A.⁵

5
- 0030956592
- (1997) Drugs Fut. , vol.22 , pp. 208-210

6
- 0026652620
- (1992) J. Org. Chem. , vol.57 , pp. 3218-3225
- Taylor, E.C.¹ Gillespie, P.² Patel, M.³

7
- 0027074583
- (1992) J. Med. Chem. , vol.35 , pp. 4809-4812
- Temple, C.¹ Rener, G.A.²

8
- 0008594585
- (1977) Chem. Heterocycl. Compd. (Engl. Transl.) , vol.13 , pp. 1006-1009
- Boldyrev, I.V.¹ Vladimirtsev, I.F.² Romanenko, E.A.³ Korzhenevskaya, N.G.⁴ Titov, E.V.⁵ Cherkasov, V.M.⁶

9
- 0034635799
- (2000) Tetrahedron Lett. , vol.41 , pp. 1757-1761
- Zanda, M.¹ Talaga, P.² Wagner, A.³ Mioskowski, C.⁴

10
- 0035808966
- (2001) Tetrahedron Lett. , vol.42 , pp. 1033-1035
- Zucca, C.¹ Bravo, P.² Volonterio, A.³ Zanda, M.⁴ Wagner, A.⁵ Mioskowski, C.⁶

11
- 0003000662
- and references therein
- (1990) Adv. Heterocycl. Chem. , vol.49 , pp. 117-192
- Vorbruggen, H.¹

12
- 84986446957
- (1982) J. Heterocycl. Chem. , vol.19 , pp. 917-921
- Ladd, D.L.¹

13
- 21844497570
- and references therein
- (1995) Pol. J. Chem. , vol.69 , pp. 1409-1416
- Zawadzki, H.¹ Penkowski, M.²

14
- 84945096445
- (1901) Chem. Ber. , vol.34 , pp. 3362-3366
- Gabriel, S.¹

15
- 84943952094
- (1903) Chem. Ber. , vol.36 , pp. 2227-2235
- Büttner, E.¹

16
- 0021354529
- (1984) Farmaco, Ed. Sci. , vol.39 , pp. 189-199
- Mossini, F.¹ Maggiali, C.² Morini, G.³ Impicciatore, M.⁴ Morini, G.⁵ Molina, E.⁶

17
- 84993899438
- (1995) J. Heterocycl. Chem. , vol.32 , pp. 1177-1180
- Delia, T.J.¹ Stark, D.² Glenn, S.K.³

18
- 0034491926
- (2000) J. Heterocycl. Chem. , vol.37 , pp. 1457-1462
- Schomaker, J.M.¹ Delia, T.J.²

19
- 0032763257
- (1999) J. Heterocycl. Chem. , vol.36 , pp. 1259-1261
- Delia, T.J.¹ Meltsner, B.R.² Schomaker, J.M.³

20
- 0008596607
- (1995) J. Indian Chem. Soc. , vol.72 , pp. 413-416
- Ramesh, A.¹ Sundar, B.S.² Murti, P.S.R.³

21
- 0021746725
- (1984) J. Med. Chem. , vol.27 , pp. 1621-1629
- D'Atri, G.¹ Gomarasca, P.² Resnati, G.³ Tronconi, G.⁴ Scolastico, C.⁵ Sirtori, C.R.⁶

22
- 0027051983
- (1992) J. Heterocycl. Chem. , vol.29 , pp. 1741-1747
- Koga, M.¹ Schneller, S.W.²

23
- 0041037814
- (2000) J. Comb. Chem. , vol.2 , pp. 195-214
- Franzén, R.G.¹

24
- 0031040133
- (1997) Helv. Chem. Acta , vol.80 , pp. 65-72
- Obrecht, D.¹ Abrecht, C.² Grieder, A.³ Villalgordo, J.M.⁴

25
- 0032785521
- (1999) Chem. Eur. J. , vol.5 , pp. 3450-3458
- Guiller, F.¹ Roussel, P.² Moser, H.³ Kane, P.⁴ Bradley, M.⁵

26
- 0034183890
- (2000) J. Comb. Chem. , vol.2 , pp. 249-253
- Di Lucrezia, R.¹ Gilbert, I.H.² Floyd, C.D.³

27
- 0024507397
- (1989) J. Med. Chem. , vol.32 , pp. 663-671
- Bagley, J.R.¹ Wynn, R.L.² Rudo, F.G.³ Doorley, B.M.⁴ Spencer, H.K.⁵ Spaulding, T.⁶

28
- 0008618732
- (1987) J. Med. Chem. , vol.30 , pp. 1794-1798
- Campbell, S.F.¹ Plews, R.M.²

29
- 15144354135
- (1998) J. Med. Chem. , vol.41 , pp. 3727-3735
- Tucker, J.A.¹ Allwine, D.A.² Grega, K.C.³ Barbachyn, M.R.⁴ Klock, J.L.⁵ Adamski, J.L.⁶ Brickner, S.J.⁷ Hutchinson, D.K.⁸ Ford, C.W.⁹ Zurenko, G.E.¹⁰ Conradi, R.A.¹¹ Burton, P.S.¹² Jensen, R.M.¹³

30
- 0007398924
- (1996) Med. Chem. Res. , pp. 61-68
- Basha, A.¹ Ratajczyk, J.D.² Dyer, R.D.³ Young, P.⁴ Carter, G.W.⁵ Brooks, C.D.W.⁶

31
- 0000033492
- (1981) Tetrahedron , vol.37 , pp. 1787-1794
- Tomazic, A.¹ Tisler, M.² Stanovnik, B.³

32
- 0024596112
- (1989) J. Med. Chem. , vol.32 , pp. 562-568
- Arrowsmith, J.E.¹ Campbell, S.F.² Cross, P.E.³ Burges, R.A.⁴ Gardiner, D.G.⁵

33
- 0030042625
- (1996) J. Med. Chem. , vol.39 , pp. 570-581
- Klein, J.T.¹ Davis, L.² Olsen, G.E.³ Wong, G.S.⁴ Huger, F.P.⁵ Smith, C.P.⁶ Petko, W.W.⁷ Cornfeldt, M.⁸ Wilker, J.C.⁹ Blitzer, R.D.¹⁰ Landau, E.¹¹ Haroutunian, V.¹² Martin, L.L.¹³ Effland, R.C.¹⁴

34
- 0028238212
- (1994) J. Org. Chem. , vol.59 , pp. 2473-2481
- Edstrom, E.D.¹ Wei, Y.² Gordon, M.³

35
- 4243584163
- (1996) Collect. Czech. Chem. Commun. , vol.61
- Sharkin, Y.¹

36
- 0019076502
- (1980) Farmaco, Ed. Sci. , vol.35 , pp. 879-886
- Giovanninetti, G.¹ Garuti, L.² Cavrini, V.³ Roveri, P.⁴ Mannini Palenzona, A.⁵ Sinibaldi, P.⁶ Fusco, P.A.⁷

37
- 0025077664
- (1990) J. Heterocycl. Chem. , vol.27 , pp. 1527-1536
- Bridges, A.J.¹ Sanchez, J.P.²

38
- 0008554853
- Note

39
- 0008584763
- Note

40
- 0002432140
- (1998) J. Chem. Soc., Chem Commun. , pp. 891-892
- Steiner, T.¹ Desiraju, G.R.²

41
- 1842763826
- (1997) J. Chem. Soc., Chem. Commun. , pp. 727-734
- Steiner, T.¹

42
- 0343953413
- (2000) Tetrahedron Lett. , vol.41 , pp. 5827-5831
- Mazik, M.¹ Blaser, D.² Boese, R.³

43
- 0000216832
- (1996) Acc. Chem. Res. , vol.29 , pp. 441-449
- Desiraju, G.R.¹

44
- 11344284526
- (1987) J. Chem. Soc., Perkin Trans. 2
- Allen, F.M.¹ Kennard, O.² Watson, D.G.³ Brammer, L.⁴ Orpen, A.G.⁵ Taylor, R.J.⁶

45
- 0003467672
- Wiley: New York
- (1992) Advanced Organic Chemistry; 4th ed. , pp. 278-286
- March, J.¹

46
- 0008551249
- Note

47
- 0001109555
- (1989) J. Appl. Crystallogr. , vol.22 , pp. 389-393
- Burla, M.C.¹ Camalli, M.² Cascarano, G.³ Giacovazzo, C.⁴ Polidori, G.⁵ Spagna, R.⁶ Viterbo, D.⁷

48
- 0011713836
- Nónius, B.V.: Delft, The Netherlands
- (1997) LSFM OpenMoleN, Interactive Intelligent Structure Solution

49
- 84944438568
- (1983) Acta Crystallogr. , vol.A39 , pp. 876-880
- Flack, H.D.¹

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