Glutamic acid as a new linker for attachment of alcohols to solid support

Tetrahedron Letters

Volumn 43, Issue 50, 2002, Pages 9221-9223

  Subra, Gilles ^a   Amblard, Muriel ^a   Martinez, Jean ^a  

^a UNIVERSITÉ DE MONTPELLIER   (France)

Author keywords

Combinatorial chemistry; Glutamic acid; Linker; Solid phase synthesis

Indexed keywords

3,3' DIAMINODIPHENYLMETHANOL; ALCOHOL DERIVATIVE; DIMER; GLUTAMIC ACID; METHANOL DERIVATIVE; UNCLASSIFIED DRUG;

ARTICLE; CYCLIZATION; DEPROTECTION REACTION; MASS SPECTROMETRY; SYNTHESIS;

EID: 0037049205     PISSN: 00404039     EISSN: None     Source Type: Journal    
DOI: 10.1016/S0040-4039(02)02209-8     Document Type: Article

References (8)

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3. Subra, G. Synthese d'agonistes et d'antagonistes du TGF-β, Ph.D., Université de Montpellier I, France, 1999; pp. 73-76.
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6. While the writing of this paper, we were advised of a poster communication presented at the 27th European Peptide Symposium in Sorrento (Italy) August 31, September 6, 2002, by T. Wakamiya et al. about the use of glutamic acid linker.
7. Kaiser E., Collescot R.L., Bossinger C.D., Cook P.I. Anal. Biochem. 40:1967;2164-2167.
8. Purity was estimated by HPLC analysis at 220 nm based on peak areas.