Characterization of some novel α1-adrenoceptor antagonists in human hyperplastic prostate

European Journal of Pharmacology

Volumn 445, Issue 1-2, 2002, Pages 125-131

  Chueh, Shih Chieh ^a   Chern, Ji Wang ^a   Choong, Chee Min ^a   Guh, Jih Hwa ^a   Teng, Che Ming ^a  

^a NATIONAL TAIWAN UNIVERSITY   (Taiwan)

Author keywords

Hyperplastic prostate, human; 1 Adrenoceptor antagonist; 1 Adrenoceptor subtype

Indexed keywords

15 HYDROXY 11ALPHA,9ALPHA EPOXYMETHANOPROSTA 5,13 DIENOIC ACID; 2 [4 [4 (2 METHOXYPHENYL)PIPERAZINYL]BUTYL]AMINO 4 CYCLOHEXYAMINOQUINAZOLIN; 4 [3 [4 (2 METHOXYPHENYL)PIPERAZINYL]PROPYL]AMINOQUINAZOLIN 2 CARBOXAMIDE; ALPHA 1 ADRENERGIC RECEPTOR; ALPHA 1A ADRENERGIC RECEPTOR; ALPHA 1B ADRENERGIC RECEPTOR; ALPHA ADRENERGIC RECEPTOR BLOCKING AGENT; ETHYL 4 [3 [4 (2 METHOXYPHENYL)PIPERAZINYL]AMINOQUINAZOLIN 2 CARBOXYLATE]; EW 154; EW 65; FH 71; PHENYLEPHRINE; POTASSIUM ION; UNCLASSIFIED DRUG;

ADULT; AGED; AORTA CONSTRICTION; ARTICLE; CONTROLLED STUDY; DRUG ACTIVITY; DRUG CYTOTOXICITY; DRUG EFFECT; DRUG MECHANISM; DRUG POTENCY; DRUG SCREENING; DRUG SELECTIVITY; DRUG SYNTHESIS; HUMAN; HUMAN TISSUE; MALE; PRIORITY JOURNAL; PROSTATE; PROSTATE HYPERTROPHY; SMOOTH MUSCLE CONTRACTION; SMOOTH MUSCLE FIBER; SPLEEN; VAS DEFERENS;

ADRENERGIC ALPHA-ANTAGONISTS; ANIMALS; AORTA; CELL SURVIVAL; CELLS, CULTURED; DOSE-RESPONSE RELATIONSHIP, DRUG; HUMANS; MALE; PIPERAZINES; PIPERIDINES; PROSTATIC HYPERPLASIA; QUINAZOLINES; RATS; RECEPTORS, ADRENERGIC, ALPHA-1; SPLEEN; VAS DEFERENS;

EID: 0037036238     PISSN: 00142999     EISSN: None     Source Type: Journal    
DOI: 10.1016/S0014-2999(02)01717-X     Document Type: Article

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