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Volumn 45, Issue 14, 2002, Pages 3022-3031

Further characterization of structural requirements for ligands at the dopamine D2 and D3 receptor: Exploring the thiophene moiety

(6) Dijkstra, Durk a Rodenhuis, Nienke a Vermeulen, Erik S a Pugsley, Thomas A b Wise, Lawrence D b Wikström, Håkan V a

a UNIVERSITY OF GRONINGEN (Netherlands)

b PFIZER INC (United States)

Author keywords

[No Author keywords available]

Indexed keywords

2 AMINOTETRALIN DERIVATIVE; 2,3,4A,5,6,9B HEXAHYDRO 4H THIANAPHTH[4,5E][1,4]OXAZINE; 5 (N DI N PROPYL)AMINO 4,5,6,7 TETRAHYDROBENZO[B]THIOPHENE; 6 (N DI N PROPYL)AMINO 4,5,6,7 TETRAHYDROBENZO[B]THIOPHENE; DOPAMINE 2 RECEPTOR; DOPAMINE 3 RECEPTOR; DOPAMINE RECEPTOR STIMULATING AGENT; HEXAHYDROTHIANAPHTHOXAZINE DERIVATIVE; N PROPYL 2,3,4A,5,6,9B HEXAHYDRO 4H THIANAPHTH[4,5E][1,4]OXAZINE; ROTIGOTINE; THIOPHENE DERIVATIVE; UNCLASSIFIED DRUG;

ANIMAL CELL; ANIMAL EXPERIMENT; ARTICLE; BINDING AFFINITY; DOPAMINERGIC SYSTEM; DRUG BIOAVAILABILITY; DRUG RECEPTOR BINDING; DRUG STRUCTURE; DRUG SYNTHESIS; LIGAND BINDING; MICRODIALYSIS; NONHUMAN; PHARMACOPHORE; RAT;

ANIMALS; BINDING, COMPETITIVE; BIOLOGICAL AVAILABILITY; CHO CELLS; CRICETINAE; DOPAMINE AGONISTS; HUMANS; MAGNETIC RESONANCE SPECTROSCOPY; MICRODIALYSIS; RADIOLIGAND ASSAY; RATS; RECEPTORS, DOPAMINE D2; RECEPTORS, DOPAMINE D3; STRUCTURE-ACTIVITY RELATIONSHIP; THIOPHENES;

EID: 0037019274 PISSN: 00222623 EISSN: None Source Type: Journal
DOI: 10.1021/jm001015a Document Type: Article

Times cited : (22)

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