Carbon-carbon bond construction at the 2-position of polysubstituted pyrimidinones

Tetrahedron Letters

Volumn 43, Issue 49, 2002, Pages 8901-8903

  Zhang, Dawei ^a   Sham, Kelvin ^a   Cao, Guo Qiang ^a   Hungate, Randall ^a   Dominguez, Celia ^a  

^a AMGEN INC   (United States)

Author keywords

[No Author keywords available]

Indexed keywords

CARBON; PYRIMIDINONE DERIVATIVE;

ARTICLE; CATALYST; CHEMICAL BOND; GRIGNARD REACTION; HYDROGENATION; MOLECULE; SYNTHESIS;

EID: 0037010824     PISSN: 00404039     EISSN: None     Source Type: Journal    
DOI: 10.1016/S0040-4039(02)02197-4     Document Type: Article

References (12)

1. Kondo Y., Watanabe R., Sakamoto T., Yamanka H. Chem. Pharm. Bull. 37:1989;2814-2816.
2. Gong Y., Pauls H.W. Synlett. 6:2000;829-831.
3. Schomaker J.M., Delia T.J. J. Org. Chem. 66:2001;7125-7128.
4. Ali N.M., McKillop A., Mitchell M.B., Rebelo R.A., Wallbank P.J. Tetrahedron. 48:1992;8117-8126.
5. Haider N., van der Plas H.C. J. Heterocycl. Chem. 27:1990;1095-1097.
6. McGaffin G., de Meijiere A. Synthesis. 6:1994;583-591.
7. Spohr, U. D.; Malone, M. J.; Mantlo, N. B.; Zablocky, J. A. WO9824780 (1998).
8. Wustrow D.J., Wise L.D. Synthesis. 1991;993-995.
9. Hitchcock S.A., Mayhugh D.R., Gregory G.S. Tetrahedron Lett. 36:1995;9085-9088.
10. Wolfgang, G. Eur. Pat. Appl. EP841326 (1984).
11. Schwarz W., Hartmann R.W., Schoenenberger H. Arch. Pharm. 324:1991;223-229.
12. Batori S., Messmer A. J. Heterocycl. Chem. 31:1994;1041-1046.