4-N-aryl(benzyl)amino-4-hetaryl-1-butenes as building blocks in heterocyclic synthesis. 3. A simple synthesis of fluorinated 4-methyl-2-(3-pyridyl)-1,2,3,4-tetrahydroquinolines and their respective quinolines

Heterocyclic Communications

Volumn 8, Issue 6, 2002, Pages 583-586

  Vargas Méndez, Leonor Y ^a   Kouznetsov, Vladimir ^b  

^a UNIVERSIDAD INDUSTRIAL DE SANTANDER   (Colombia)

^b UNIVERSIDAD DE TALCA   (Chile)

Author keywords

[No Author keywords available]

Indexed keywords

2,4 DIFLUOROANILINE; 4 FLUOROANILINE; ALDEHYDE DERIVATIVE; ALKENE DERIVATIVE; NICOTINALDEHYDE; QUINOLINE DERIVATIVE; UNCLASSIFIED DRUG;

ARTICLE; CARBON NUCLEAR MAGNETIC RESONANCE; DRUG SYNTHESIS; FLUORINATION; GRIGNARD REACTION;

EID: 0036976540     PISSN: 07930283     EISSN: None     Source Type: Journal    
DOI: None     Document Type: Article

References (23)

1. Andriole, V.T., The Quinolines, Academic Press, New York, 1988.
2. Siporin, C., The New Generation of Quinolones, Basel, New York, 1990.
3. Strekowski, L., Kiselov, A.S., Hojjat, M., J. Org. Chem., 59, 5886, (1994).
4. Strekowski, L., Gulevich, Yu., van Aken, K., Wilson, D.W., Tetrahedron Lett., 36, 225, (1995).
5. Fluorine in Bioorganic Chemistry, Welch, J.T., Eswarakrishnan, S., eds., Wiley, New York, 1991.
6. Chemistry of Organic Fluorine Compounds II, Huddlicky, M., Pavlath, A.E., eds., American Chemical Society, Washington, DC, 1995.
7. Manske, R.H.F., Kulka, M, Org. React., 7, 59, (1953).
8. Oleynik, I.I., Shteingarts, V.D., J. Fluorine Chem., 91, 25, (1998).
9. Hromatka, O., Sauter, F., Knollmüller, M., Stütz, P., Monatsh. Chem., 97, 1763, (1966).
10. Communication No.1 of this series : Vargas Méndez, L.Y., Kouznetsov, V., Stashenko, E., Bahsas, A., Amaro-Luis, J., Heterocycl. Commun., 7, 323, (2001).
11. Kouznetsov, V.V., Palma, A.R., Aliev, A.E., Anales de Química. Int. Ed., 94, 132, (1998).
12. Kouznetsov, V., Turgut, Z., Zubkov, F., Kaban, S., Varlamov, A., Monatsh. Chem., 129, 671 (1998).
13. Vargas, L.Y., Rozo, W., Kouznetsov, V., Heterocycles, 53, 785, (2000).
14. Bloch, R., Chem. Rev., 98, 1407, (1998).
15. Brown, R.C.C., Fisher, M., J. Chem. Soc., Chem. Commun., 1547, (1999).
16. Voigtmann, V., Blechert, S., Synthesis, 893, (2000).
17. Wright, D.L., Schulte II, J.P., Page, M. A., Org. Lett., 2, 1847, (2000).
18. Oraa, H., Stagies, R., van der Marel, G.A., van Boom, J.H., Blechert, S., J. Chem. Soc., Chem. Commun., 1501, (2000).
19. Kuznetsov, V.V., Aliev, A.E., Prostakov, N.S., Khim. Geterotsikl. Soedin., 73, (1994) (C.A. 1994, 121, 300733p).
20. The detailed results from these studies will be published elsewhere.
21. FH = 8.9 Hz).
22. The detailed results from these studies will be published elsewhere.
23. Methods for the Oxidation of Organic Compounds, Haines, A.H., ed., Academic Press, New York, 1985, pp 16.