Synthesis and in vitro antiprotozoal activity of 5-nitrothiophene-2-carboxaldehyde thiosemicarbazone derivatives

Bioorganic and Medicinal Chemistry Letters

Volumn 12, Issue 23, 2002, Pages 3475-3478

  Bharti, Neelam ^a   Husain, Kakul ^a   Gonzalez Garza, M T ^b   Cruz Vega, Delia E ^b   Castro Garza, J ^b   Mata Cardenas, Benito D ^b   Naqvi, Fehmida ^a   Azam, Amir ^a  

^a JAMIA MILLIA ISLAMIA CENTRAL UNIVERSITY   (India)

^b INSTITUTO MEXICANO DEL SEGURO SOCIAL   (Mexico)

Author keywords

[No Author keywords available]

Indexed keywords

5 NITROTHIOPHENE 2 CARBOXALDEHYDE; ANTITRICHOMONAL AGENT; IMINE; THIOSEMICARBAZONE DERIVATIVE; UNCLASSIFIED DRUG; ALDEHYDE; AMINE; ANTIPROTOZOAL AGENT; THIOL DERIVATIVE;

ANTIPROTOZOAL ACTIVITY; ARTICLE; DRUG SYNTHESIS; INFRARED SPECTROSCOPY; PROTON NUCLEAR MAGNETIC RESONANCE; ANIMAL; CHEMISTRY; DRUG EFFECT; DRUG SENSITIVITY; ENTAMOEBA HISTOLYTICA; GIARDIA LAMBLIA; IC 50; STRUCTURE ACTIVITY RELATION; SYNTHESIS; TRICHOMONAS VAGINALIS;

ALDEHYDES; AMINES; ANIMALS; ANTIPROTOZOAL AGENTS; ENTAMOEBA HISTOLYTICA; GIARDIA LAMBLIA; INHIBITORY CONCENTRATION 50; PARASITIC SENSITIVITY TESTS; STRUCTURE-ACTIVITY RELATIONSHIP; SULFHYDRYL COMPOUNDS; THIOSEMICARBAZONES; TRICHOMONAS VAGINALIS;

EID: 0036888378     PISSN: 0960894X     EISSN: None     Source Type: Journal    
DOI: 10.1016/S0960-894X(02)00703-5     Document Type: Article

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