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Volumn 12, Issue 6, 2002, Pages 369-378

Preparation, pharmacokinetic and pharmacodynamic evaluation of carbamazepine inclusion complexes with cyclodextrins

Author keywords

CD; CD; Bioavailability and anti convulsion activity; Carbamazepine; Dissolution; DM CD; DSC; Inclusion complexes; IR spectroscopy; Solubility; X ray diffraction

Indexed keywords

ALPHA CYCLODEXTRIN; BETA CYCLODEXTRIN; CARBAMAZEPINE; CYCLODEXTRIN; DI O METHYL BETA CYCLODEXTRIN; UNCLASSIFIED DRUG;

EID: 0036857995     PISSN: 11571489     EISSN: None     Source Type: Journal    
DOI: None     Document Type: Article
Times cited : (8)

References (35)
  • 1
    • 0004144140 scopus 로고
    • Pharmaceutical Press, London
    • th Ed., Pharmaceutical Press, London, 1993, pp. 295-298.
    • (1993) th Ed. , pp. 295-298
    • Martindale1
  • 2
    • 0003576886 scopus 로고
    • The Pharmaceutical Press, London
    • nd Ed., The Pharmaceutical Press, London, 1986.
    • (1986) nd Ed.
    • Clark, C.1
  • 3
    • 0022471553 scopus 로고
    • Simultaneous first and zero-order absorption of carbamazepine tablets in human
    • Riad L.E., Chan K.K., Wagner W.E. - Simultaneous first and zero-order absorption of carbamazepine tablets in human. - J. Pharm. Sci., 75, 897-900, 1986.
    • (1986) J. Pharm. Sci. , vol.75 , pp. 897-900
    • Riad, L.E.1    Chan, K.K.2    Wagner, W.E.3
  • 4
    • 0025977852 scopus 로고
    • Dissolution and relative bioavailability of two carbamazepine preparations for children with epilepsy
    • Hartley R., Aleksandrowicz L., Bowmerc J., Cavood A., Forsythe W.J. - Dissolution and relative bioavailability of two carbamazepine preparations for children with epilepsy. - J. Pharm. Pharmacol., 43, 117-119, 1991.
    • (1991) J. Pharm. Pharmacol. , vol.43 , pp. 117-119
    • Hartley, R.1    Aleksandrowicz, L.2    Bowmerc, J.3    Cavood, A.4    Forsythe, W.J.5
  • 6
  • 7
    • 0016798977 scopus 로고
    • Bioavailability of two carbamazepine preparations during chronic administration to epileptic patients
    • Morselli P.L., Monaco F., Gerna M., Recchia M., Riccio A. - Bioavailability of two carbamazepine preparations during chronic administration to epileptic patients. - Epilepsia, 16, 759-764, 1975.
    • (1975) Epilepsia , vol.16 , pp. 759-764
    • Morselli, P.L.1    Monaco, F.2    Gerna, M.3    Recchia, M.4    Riccio, A.5
  • 8
    • 0008036592 scopus 로고
    • Drugs effective in the therapy of the epilepsies
    • M. Goodman, B. Gilman Eds., 7th ed., Macmillan, New York
    • Ball T.W., Schleifer L.S. - Drugs effective in the therapy of the epilepsies. - In: The Pharmacological Basis of Therapeutics, M. Goodman, B. Gilman Eds., 7th ed., Macmillan, New York, 1985, pp. 446-472.
    • (1985) The Pharmacological Basis of Therapeutics , pp. 446-472
    • Ball, T.W.1    Schleifer, L.S.2
  • 9
    • 0000361082 scopus 로고
    • Interaction of pharmaceuticals with Scardinger dextrins. I. Interaction with hydrobenzoic acids and p-hydroxybenzoates
    • Cohen J., Lach J.L. - Interaction of pharmaceuticals with Scardinger dextrins. I. Interaction with hydrobenzoic acids and p-hydroxybenzoates. - J. Pharm. Sci., 52, 132, 1963.
    • (1963) J. Pharm. Sci. , vol.52 , pp. 132
    • Cohen, J.1    Lach, J.L.2
  • 10
    • 0025649779 scopus 로고
    • Pharmaceutical uses of cyclodextrins and derivatives
    • Duchene D., Wouessidjewe D. - Pharmaceutical uses of cyclodextrins and derivatives. - Drug Dev. Ind. Pharm., 15, 2487-2499, 1990.
    • (1990) Drug Dev. Ind. Pharm. , vol.15 , pp. 2487-2499
    • Duchene, D.1    Wouessidjewe, D.2
  • 11
    • 0026328096 scopus 로고
    • Solubilization and stabilization of drugs through cyclodextrin complexation
    • Loftsson T., Frioriksdottir B.J. - Solubilization and stabilization of drugs through cyclodextrin complexation. - Acta Pharm. Nord., 3, 215-217, 1991.
    • (1991) Acta Pharm. Nord. , vol.3 , pp. 215-217
    • Loftsson, T.1    Frioriksdottir, B.J.2
  • 12
    • 0021816582 scopus 로고
    • Solubilization of drugs by modified β-cyclodextrins
    • Haller B.W., Brauns U. - Solubilization of drugs by modified β-cyclodextrins. - Int. J. Pharm., 26, 77-88, 1985.
    • (1985) Int. J. Pharm. , vol.26 , pp. 77-88
    • Haller, B.W.1    Brauns, U.2
  • 13
    • 0032948152 scopus 로고    scopus 로고
    • Solid dispersions of hydroxypropyl-beta-cyclodextrin and carbamazepine: Study of complexation and in vitro dissolution profile
    • Londhe V. Y., Nagarsenkar M.S. - Solid dispersions of hydroxypropyl-beta-cyclodextrin and carbamazepine: Study of complexation and in vitro dissolution profile. - Indian Drugs, 36, 12-20, 1999.
    • (1999) Indian Drugs , vol.36 , pp. 12-20
    • Londhe, V.Y.1    Nagarsenkar, M.S.2
  • 14
    • 0032526833 scopus 로고    scopus 로고
    • Enhancement of carbamazepine dissolution: In vitro and in vivo evaluation
    • El-zein H., Riad L., El-Bary A.A. - Enhancement of carbamazepine dissolution: In vitro and in vivo evaluation. - Int. J. Pharm., 168, 209-220, 1998.
    • (1998) Int. J. Pharm. , vol.168 , pp. 209-220
    • El-zein, H.1    Riad, L.2    El-Bary, A.A.3
  • 15
    • 0031819170 scopus 로고    scopus 로고
    • Kneaded solid dispersions of hydroxypropyl-beta-cyclodextrin and carbamazepine: Complexation and in vitro dissolution profile
    • Nagarsenker M.S., Bhave V.M. - Kneaded solid dispersions of hydroxypropyl-beta-cyclodextrin and carbamazepine: Complexation and in vitro dissolution profile. - Pharm. Pharmacol. Comm., 4, 335-338, 1998.
    • (1998) Pharm. Pharmacol. Comm. , vol.4 , pp. 335-338
    • Nagarsenker, M.S.1    Bhave, V.M.2
  • 16
    • 0344588867 scopus 로고    scopus 로고
    • Effect of water-soluble polymers on the aqueous solubility and complexing abilities of beta-cyclodextrin
    • Loftsson T., Frioriksdottir H. - Effect of water-soluble polymers on the aqueous solubility and complexing abilities of beta-cyclodextrin. - Int. J. Pharm., 163, 115-121, 1998.
    • (1998) Int. J. Pharm. , vol.163 , pp. 115-121
    • Loftsson, T.1    Frioriksdottir, H.2
  • 17
    • 0029802020 scopus 로고    scopus 로고
    • Physicochemical characteristics of carbamazepine-beta-cyclodextrin inclusion compounds and carbamazepine-PEG solid dispersions
    • El-Nahhas S.A. - Physicochemical characteristics of carbamazepine-beta-cyclodextrin inclusion compounds and carbamazepine-PEG solid dispersions. - Pharmazie, 51, 960963, 1996.
    • (1996) Pharmazie , vol.51 , pp. 960963
    • El-Nahhas, S.A.1
  • 18
    • 15444352072 scopus 로고    scopus 로고
    • Intravenous and oral pharmacokinetic evaluation of 2-hydroxypropyl-beta-cyclodextrin based formulation of carbamazepine in the dog: Comparison with commercially available tablets and suspensions
    • Brewster M.E., Anderson W.R., Meinsma D., Moreno D., Pop E. - Intravenous and oral pharmacokinetic evaluation of 2-hydroxypropyl-beta-cyclodextrin based formulation of carbamazepine in the dog: Comparison with commercially available tablets and suspensions. - J. Pharm. Sci., 86, 335-339, 1997.
    • (1997) J. Pharm. Sci. , vol.86 , pp. 335-339
    • Brewster, M.E.1    Anderson, W.R.2    Meinsma, D.3    Moreno, D.4    Pop, E.5
  • 19
    • 0031544009 scopus 로고    scopus 로고
    • Brain delivery of carbamazepine during intravenous administration of polyethylene glycol and 2-hydroxypropylbeta-cyclodextrin formulations
    • Cheung B.W., Wang Y., Brewster M.E., Sawchuk R.J. - Brain delivery of carbamazepine during intravenous administration of polyethylene glycol and 2-hydroxypropylbeta-cyclodextrin formulations. - STP Pharma Sci., 7, 78-84, 1997.
    • (1997) STP Pharma Sci. , vol.7 , pp. 78-84
    • Cheung, B.W.1    Wang, Y.2    Brewster, M.E.3    Sawchuk, R.J.4
  • 21
    • 0027202722 scopus 로고
    • Increase in temperature enhances solubility of drugs in aqueous solutions of hydroxypropyl-beta-cyclodextrins
    • Hoshino T., Uekama K., Pitha J. - Increase in temperature enhances solubility of drugs in aqueous solutions of hydroxypropyl-beta-cyclodextrins. - Int. J. Pharm., 98,239-242, 1993.
    • (1993) Int. J. Pharm. , vol.98 , pp. 239-242
    • Hoshino, T.1    Uekama, K.2    Pitha, J.3
  • 22
    • 85047693676 scopus 로고
    • Oral pharmacokinetics of carbamazepine: In dogs from commercial tablets and a cyclodextrin complex
    • Bettach C.J., Gonzalez M.A., McHiernan B.C., Neff-Davis C., Bodor N. - Oral pharmacokinetics of carbamazepine: In dogs from commercial tablets and a cyclodextrin complex. J. Pharm. Sci., 82, 1058-1060, 1993.
    • (1993) J. Pharm. Sci. , vol.82 , pp. 1058-1060
    • Bettach, C.J.1    Gonzalez, M.A.2    McHiernan, B.C.3    Neff-Davis, C.4    Bodor, N.5
  • 23
    • 0026672498 scopus 로고
    • Improvement of oral bioavailability of carbamazepine by inclusion in 2-hydroxypropylbeta-cyclodextrin
    • Choudhury S., Nelson K.F. - Improvement of oral bioavailability of carbamazepine by inclusion in 2-hydroxypropylbeta-cyclodextrin. - Int. J. Pharm., 85, 175-180, 1992.
    • (1992) Int. J. Pharm. , vol.85 , pp. 175-180
    • Choudhury, S.1    Nelson, K.F.2
  • 24
    • 0025810218 scopus 로고
    • Development of aqueous parenteral formulations for carbamazepine through the use of modified cyclodextrins
    • Brewster M.E., Anderson W.R., Estes K.S., Bodor N. - Development of aqueous parenteral formulations for carbamazepine through the use of modified cyclodextrins. - J. Pharm. Sci., 80, 380-383, 1991.
    • (1991) J. Pharm. Sci. , vol.80 , pp. 380-383
    • Brewster, M.E.1    Anderson, W.R.2    Estes, K.S.3    Bodor, N.4
  • 26
    • 0021984767 scopus 로고
    • Simultaneous determination of carbamazepine and its epixide metabolite in plasma and urine by high performance liquid chromatography
    • Chan K.K.H. - Simultaneous determination of carbamazepine and its epixide metabolite in plasma and urine by high performance liquid chromatography. - J. Chromatogr., 342, 341-346, 1985.
    • (1985) J. Chromatogr. , vol.342 , pp. 341-346
    • Chan, K.K.H.1
  • 29
    • 0020692951 scopus 로고
    • The evaluation of different types of anti-convulsant drug activity against leptazol-induced epileptogenic activity in the anaesthetized rat
    • Kent A.P., Webster R.A. - The evaluation of different types of anti-convulsant drug activity against leptazol-induced epileptogenic activity in the anaesthetized rat. - Br. J. Pharmacol., 78, 553-559, 1983.
    • (1983) Br. J. Pharmacol. , vol.78 , pp. 553-559
    • Kent, A.P.1    Webster, R.A.2
  • 31
    • 0021321230 scopus 로고
    • A new type of anticonvulsant, Stiripentol: Pharmacological profile and neurochemical study
    • No. 2
    • Poisson M., Huguet A., Bakri-Logeais F., Narcisse G. - A new type of anticonvulsant, Stiripentol: Pharmacological profile and neurochemical study. - Drug Res., 34 (1), No. 2, 1984.
    • (1984) Drug Res. , vol.34 , Issue.1
    • Poisson, M.1    Huguet, A.2    Bakri-Logeais, F.3    Narcisse, G.4
  • 32
    • 0018846940 scopus 로고
    • Convulsant drugs: Mechanisms of action
    • Woodbury D.M. - Convulsant drugs: Mechanisms of action. - Adv. Neurol., 27, 249-303, 1980.
    • (1980) Adv. Neurol. , vol.27 , pp. 249-303
    • Woodbury, D.M.1
  • 33
    • 0011889492 scopus 로고
    • Experimental evaluation of anticonvulsants
    • J.A. Vida Ed., Academic Press, New York
    • Reinhard J.F., Reinhard J.F. Jr. - Experimental evaluation of anticonvulsants. - In: Anticonvulsants, J.A. Vida Ed., Academic Press, New York, 1977, pp. 581112.
    • (1977) Anticonvulsants , pp. 581112
    • Reinhard, J.F.1    Reinhard J.F., Jr.2
  • 34
    • 84951384024 scopus 로고
    • A simplified method of evaluating dose-effect experiments
    • Litcfield, J.T. Jr., Wilcoxon F. - A simplified method of evaluating dose-effect experiments. - J. Pharmacol. Exp. Ther., 96, 99-113, 1994.
    • (1994) J. Pharmacol. Exp. Ther. , vol.96 , pp. 99-113
    • Litcfield J.T., Jr.1    Wilcoxon, F.2


* 이 정보는 Elsevier사의 SCOPUS DB에서 KISTI가 분석하여 추출한 것입니다.