Tc and Re chelates of 8α-amino-6-methyl-ergoline: Synthesis and affinity to the dopamine D 2 receptor

Bioorganic and Medicinal Chemistry

Volumn 10, Issue 11, 2002, Pages 3523-3528

  Spies, H ^a   Noll, B ^a   Noll, St ^a   Findeisen, M ^a   Brust, P ^a   Syhre, R ^a   Berger, R ^a  

^a INSTITUTE OF ION BEAM PHYSICS AND MATERIALS RESEARCH   (Germany)

Author keywords

[No Author keywords available]

Indexed keywords

8ALPHA AMINO 6 METHYLERGOLINE; DOPAMINE 2 RECEPTOR; ERGOLINE DERIVATIVE; N (2 MERCAPTO)ACETYL 8 ALPHA AMINO 6 METHYLERGOLINE; N (2 MERCAPTO)PROPIONYL 8 ALPHA AMINO 6 METHYLERGOLINE; N (2 METHYLMERCAPTO)ACETYL 8 ALPHA AMINO 6 METHYLERGOLINE; N (2 METHYLMERCAPTO)PROPIONYL 8 ALPHA AMINO 6 METHYLERGOLINE; N 2 (BENZOYLMERCAPTO)ACETYL 8 ALPHA AMINO 6 METHYLERGOLINE; N 2 (BENZOYLMERCAPTO)PROPIONYL 8 ALPHA AMINO 6 METHYLERGOLINE; RHENIUM COMPLEX; TECHNETIUM COMPLEX; UNCLASSIFIED DRUG;

ACETYLATION; ANIMAL EXPERIMENT; ANIMAL TISSUE; ARTICLE; BRAIN; CHELATION; CONTROLLED STUDY; DOPAMINERGIC SYSTEM; DRUG SYNTHESIS; IC 50; KIDNEY; LIPOPHILICITY; LIVER; MALE; NONHUMAN; PLASMA CLEARANCE; RAT; RECEPTOR AFFINITY;

ANIMALS; BRAIN; CHELATING AGENTS; CHEMISTRY, PHYSICAL; CHROMATOGRAPHY, HIGH PRESSURE LIQUID; CLONING, MOLECULAR; DOPAMINE AGONISTS; ERGOLINES; HUMANS; INDICATORS AND REAGENTS; KIDNEY; LIVER; MAGNETIC RESONANCE SPECTROSCOPY; MALE; RADIOLIGAND ASSAY; RATS; RATS, WISTAR; RECEPTORS, DOPAMINE D2; RHENIUM; STRUCTURE-ACTIVITY RELATIONSHIP; TECHNETIUM; TISSUE DISTRIBUTION;

RATTUS NORVEGICUS;

EID: 0036836815     PISSN: 09680896     EISSN: None     Source Type: Journal    
DOI: 10.1016/S0968-0896(02)00214-6     Document Type: Article

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