Indexed keywords
2 (2,3 DIHYDRO 2 PENTYLBENZOFURAN 2 YL) 2 IMIDAZOLINE;
ADRENERGIC RECEPTOR STIMULATING AGENT;
GUANINE NUCLEOTIDE BINDING PROTEIN;
LIGAND;
PARTIAL AGONIST;
PROTEIN SUBUNIT;
UNCLASSIFIED DRUG;
BINDING AFFINITY;
CELL TYPE;
CHO CELL;
DRUG RECEPTOR BINDING;
GENETIC TRANSFECTION;
LETTER;
LIGAND BINDING;
MOLECULAR MODEL;
PRIORITY JOURNAL;
PROTEIN CONFORMATION;
SIGNAL TRANSDUCTION;
1
0029162109
Pharmacological proteus?
T. Kenakin Pharmacological proteus? Trends Pharmacol. Sci. 16 1995 256 258
(1995)
Trends Pharmacol. Sci. , vol.16
, pp. 256-258
Kenakin, T.1
2
0035083109
Inverse, protean, and ligand-selective agonism: matters of receptor conformation
T. Kenakin Inverse, protean, and ligand-selective agonism: matters of receptor conformation FASEB J. 15 2001 598 611
(2001)
FASEB J. , vol.15
, pp. 598-611
Kenakin, T.1
3
0034792326
Considerations in the evaluation of inverse agonism and protean agonism at G protein-coupled receptors
P. Chidiac Considerations in the evaluation of inverse agonism and protean agonism at G protein-coupled receptors Methods Enzymol. 343 2002 3 16
(2002)
Methods Enzymol. , vol.343
, pp. 3-16
Chidiac, P.1
4
0036094811
Evidence for protean agonism of RX 831003 at α2A-adrenoceptors by co-expression with different Gα protein subunits
α protein subunits Neuropharmacology 42 2002 855 863
(2002)
Neuropharmacology , vol.42
, pp. 855-863
Pauwels, P.J.1
5
0029054965
Agonist-receptor efficacy II: agonist trafficking of receptor signals
T. Kenakin Agonist-receptor efficacy II: agonist trafficking of receptor signals Trends Pharmacol. Sci. 16 1995 232 238
(1995)
Trends Pharmacol. Sci. , vol.16
, pp. 232-238
Kenakin, T.1
6
0032819108
Influence of G protein type on agonist efficacy
G. Lang S.M. Lanier Influence of G protein type on agonist efficacy Mol. Pharmacol. 56 1999 651 656
(1999)
Mol. Pharmacol. , vol.56
, pp. 651-656
Lang, G.1
Lanier, S.M.2
7
0033929371
Agonist-directed trafficking of porcine α2A-adrenergic receptor signaling in CHO cells. l-Isoproterenol selectively activates Gs
s J. Pharmacol. Exp. Ther. 294 2000 539 547
(2000)
J. Pharmacol. Exp. Ther. , vol.294
, pp. 539-547
Brink, C.B.1
8
0031815337
Effector pathway-dependent R.e. at serotonin type 2A and 2C receptors: evidence for agonist-directed trafficking of receptor stimulus
K.A. Berg Effector pathway-dependent R. e . at serotonin type 2A and 2C receptors: evidence for agonist-directed trafficking of receptor stimulus Mol. Pharmacol. 54 1998 94 104
(1998)
Mol. Pharmacol. , vol.54
, pp. 94-104
Berg, K.A.1
9
0030823303
A three-state model of agonist action
P. Leff A three-state model of agonist action Trends Pharmacol. Sci. 18 1997 355 362
(1997)
Trends Pharmacol. Sci. , vol.18
, pp. 355-362
Leff, P.1
10
0034791894
Theoretical implications of receptor coupling to multiple G proteins based on analysis of a three-state model
C. Scaramellini P. Leff Theoretical implications of receptor coupling to multiple G proteins based on analysis of a three-state model Methods Enzymol. 343 2002 17 29
(2002)
Methods Enzymol. , vol.343
, pp. 17-29
Scaramellini, C.1
Leff, P.2
