메뉴 건너뛰기




Volumn 5, Issue 5, 2002, Pages 793-800

New approaches to reversal of neuromuscular block

Author keywords

Acetylcholinesterase inhibitors; Anesthesia; Cyclodextrins; Muscle relaxants; Neuromuscular block; Reversal

Indexed keywords

ACETYLCHOLINE; ACETYLCHOLINESTERASE; AMINOPYRIDINE; ATROPINE; CHOLINESTERASE; CHOLINESTERASE INHIBITOR; CISATRACURIUM; CURARE DERIVATIVE; CYCLODEXTRIN; DONEPEZIL; EDROPHONIUM; GALLAMINE; GLYCOPYRRONIUM BROMIDE; MIVACURIUM; MUSCARINIC AGENT; MUSCARINIC RECEPTOR BLOCKING AGENT; MUSCLE RELAXANT AGENT; NEOSTIGMINE; NEUROMUSCULAR BLOCKING AGENT; PANCURONIUM; PHYSOSTIGMINE; PYRIDINIUM DERIVATIVE; PYRIDOSTIGMINE; RAPACURONIUM BROMIDE; ROCURONIUM; SUXAMETHONIUM; TETRYLAMMONIUM; TUBOCURARINE CHLORIDE; UNINDEXED DRUG; VECURONIUM;

EID: 0036771227     PISSN: 13676733     EISSN: None     Source Type: Journal    
DOI: None     Document Type: Review
Times cited : (14)

References (51)
  • 1
    • 0000323076 scopus 로고
    • Über die verbindung lokalanaesthesie mit der narkose, über hohe extradural anaesthesie und epidurale injektionen anaesthesierende loesungen bei tabetischen magenkriesen
    • Läwen A: Über die Verbindung Lokalanaesthesie mit der Narkose, über hohe Extradural Anaesthesie und epidurale Injektionen anaesthesierende Loesungen bei tabetischen Magenkriesen. Beitrage Klinische Chirurgie (1912) 80:168-169.
    • (1912) Beitrage Klinische Chirurgie , vol.80 , pp. 168-169
    • Läwen, A.1
  • 2
    • 0000972742 scopus 로고
    • The use of curare in general anesthesia
    • Griffith HR, Johnson GE: The use of curare in general anesthesia. Anesthesiology (1942) 3:418-420.
    • (1942) Anesthesiology , vol.3 , pp. 418-420
    • Griffith, H.R.1    Johnson, G.E.2
  • 4
    • 0001731605 scopus 로고    scopus 로고
    • Pharmacology of muscle relaxants and their antagonists
    • Miller RD (Ed), Churchill-Livingstone, Philadelphia, PA, USA
    • Savarese JJ, Caldwell JE, Lien CA, Miller RD: Pharmacology of muscle relaxants and their antagonists. In: Anesthesia, 5th Edition. Miller RD (Ed), Churchill-Livingstone, Philadelphia, PA, USA (2000):412-490. This section of the latest updated edition of this comprehensive text describes current use of AChE inhibitors in the clinic.
    • (2000) Anesthesia, 5th Edition , pp. 412-490
    • Savarese, J.J.1    Caldwell, J.E.2    Lien, C.A.3    Miller, R.D.4
  • 5
    • 0013348220 scopus 로고
    • Self-experiments with succinylcholine chloride: A new ultra-short-acting muscle relaxant
    • Mayrhofer OK: Self-experiments with succinylcholine chloride: A new ultra-short-acting muscle relaxant. Br Med J (1952) 2:1332-1334.
    • (1952) Br Med J , vol.2 , pp. 1332-1334
    • Mayrhofer, O.K.1
  • 6
    • 0013393284 scopus 로고
    • Über curare und curarealkaloide
    • Böhm R: Über Curare und Curarealkaloide. Arch Pharmacol Berlin (1897) 235:660-664.
    • (1897) Arch Pharmacol Berlin , vol.235 , pp. 660-664
    • Böhm, R.1
  • 7
    • 0018770642 scopus 로고
    • Residual curarization in the recovery room
    • Viby-Mogensen J, Jørgensen BC, Ørding H: Residual curarization in the recovery room. Anesthesiology (1979) 50:439-441. This paper is an early description of the problems associated with post-surgery residual curarization, revealed by detailed monitoring.
    • (1979) Anesthesiology , vol.50 , pp. 439-441
    • Viby-Mogensen, J.1    Jørgensen, B.C.2    Ørding, H.3
  • 8
    • 0000399902 scopus 로고
    • A one year prospective study of postoperative pulmonary complications after neuromuscular blockade by pancuronium and atracurium
    • Pedersen T, Viby-Mogensen J, Eliasen K, Ringsted C, Henriksen E: A one year prospective study of postoperative pulmonary complications after neuromuscular blockade by pancuronium and atracurium. Anesthesiology (1988) 69(Suppl):A902.
    • (1988) Anesthesiology , vol.69 , Issue.SUPPL.
    • Pedersen, T.1    Viby-Mogensen, J.2    Eliasen, K.3    Ringsted, C.4    Henriksen, E.5
  • 9
    • 0030828897 scopus 로고    scopus 로고
    • The impact of choice of muscle relaxant on postoperative recovery time: A retrospective study
    • Ballantyne JC, Chang Y: The impact of choice of muscle relaxant on postoperative recovery time: A retrospective study. Anesth Analg (1997) 85:476-482.
    • (1997) Anesth Analg , vol.85 , pp. 476-482
    • Ballantyne, J.C.1    Chang, Y.2
  • 10
    • 0026648625 scopus 로고
    • Reversal of neuromuscular blockade
    • Bevan DR, Donati F, Kopman AF: Reversal of neuromuscular blockade. Anesthesiology (1992) 77:785-805. A comprehensive review of the reversal of NMB.
    • (1992) Anesthesiology , vol.77 , pp. 785-805
    • Bevan, D.R.1    Donati, F.2    Kopman, A.F.3
  • 11
    • 0013401429 scopus 로고
    • Reversal of neuromuscular block
    • Edward Arnold Editions, London, UK
    • Harper NJN, Pollard MJ (Eds): Reversal of neuromuscular block. In: Muscle Relaxants in Anaesthesia. Edward Arnold Editions, London, UK (1995) 8:135-155.
    • (1995) Muscle Relaxants in Anaesthesia , vol.8 , pp. 135-155
    • Harper, N.J.N.1    Pollard, M.J.2
  • 12
    • 0000839351 scopus 로고
    • The anticurare activity of tetraethylammonium in the cat
    • Kensler CJ: The anticurare activity of tetraethylammonium in the cat. Br J Pharmacol (1950) 5:204-209.
    • (1950) Br J Pharmacol , vol.5 , pp. 204-209
    • Kensler, C.J.1
  • 14
    • 0013401430 scopus 로고
    • Pharmacology and possible clinical applications of 4-aminopyridine
    • Agoston S, Langreter D, Newton DEF: Pharmacology and possible clinical applications of 4-aminopyridine. Semin Anesth (1985) 4:81-86.
    • (1985) Semin Anesth , vol.4 , pp. 81-86
    • Agoston, S.1    Langreter, D.2    Newton, D.E.F.3
  • 15
    • 0013393439 scopus 로고
    • Physostigmin, ein gegengift des curare
    • Pal J: Physostigmin, ein Gegengift des Curare. Zeitschrift der Physiologie (1900) 14:255-258.
    • (1900) Zeitschrift der Physiologie , vol.14 , pp. 255-258
    • Pal, J.1
  • 16
    • 0013397420 scopus 로고
    • Über eine neue therapeutische verwendungs des physostigmin
    • Laquer L: Über eine neue therapeutische Verwendungs des Physostigmin. Zentr Med Wissenschaft (1876) 14:421-422.
    • (1876) Zentr Med Wissenschaft , vol.14 , pp. 421-422
    • Laquer, L.1
  • 17
    • 0000672622 scopus 로고
    • Physostigmine (Eserine)
    • Stedman E, Barger G: Physostigmine (Eserine). J Chem Soc (1925) 127:247-258.
    • (1925) J Chem Soc , vol.127 , pp. 247-258
    • Stedman, E.1    Barger, G.2
  • 18
    • 0000525340 scopus 로고
    • Studies in the indole series III: On the synthesis of physostigmine
    • Julian PL, Pikl J: Studies in the indole series III: On the synthesis of physostigmine. J Am Chem Soc (1935) 57:539-544.
    • (1935) J Am Chem Soc , vol.57 , pp. 539-544
    • Julian, P.L.1    Pikl, J.2
  • 19
    • 0001328120 scopus 로고
    • Pharmacological action of some analogues of physostigmine
    • Aeschlimann J, Reinert M: Pharmacological action of some analogues of physostigmine. J Pharmacol Exp Ther (1931) 43:413-444.
    • (1931) J Pharmacol Exp Ther , vol.43 , pp. 413-444
    • Aeschlimann, J.1    Reinert, M.2
  • 20
    • 0030886022 scopus 로고    scopus 로고
    • A comparison between chronotropic effects of neostigmine and edrophonium in isolated guinea pig right atrium
    • Endou M, Tanito Y, Okumura F: A comparison between chronotropic effects of neostigmine and edrophonium in isolated guinea pig right atrium. J Pharmacol Exp Ther (1997) 282:1480-1486.
    • (1997) J Pharmacol Exp Ther , vol.282 , pp. 1480-1486
    • Endou, M.1    Tanito, Y.2    Okumura, F.3
  • 21
    • 0034098363 scopus 로고    scopus 로고
    • Molecular modelling and QSAR of reversible acetylcholinesterase inhibitors
    • Kaur J, Zhang MQ: Molecular modelling and QSAR of reversible acetylcholinesterase inhibitors. Curr Med Chem (2000) 7:273-294.
    • (2000) Curr Med Chem , vol.7 , pp. 273-294
    • Kaur, J.1    Zhang, M.Q.2
  • 22
    • 0037147765 scopus 로고    scopus 로고
    • Oxyaniliniums as acetylcholinesterase inhibitors for the reversal of neuromuscular block
    • Grove SJ, Kaur J, Muir AW, Pow E, Tarver GJ, Zhang MQ: Oxyaniliniums as acetylcholinesterase inhibitors for the reversal of neuromuscular block. Bioorg Med Chem Lett (2002) 12:193-196.
    • (2002) Bioorg Med Chem Lett , vol.12 , pp. 193-196
    • Grove, S.J.1    Kaur, J.2    Muir, A.W.3    Pow, E.4    Tarver, G.J.5    Zhang, M.Q.6
  • 26
    • 0037119759 scopus 로고    scopus 로고
    • Novel piperidinium and pyridinium agents as water-soluble acetylcholinesterase inhibitors for the reversal of neuromuscular blockade
    • Palin R, Clark JK, Cowley P, Muir AW, Pow E, Prosser AB, Taylor R, Zhang M-Q: Novel piperidinium and pyridinium agents as water-soluble acetylcholinesterase inhibitors for the reversal of neuromuscular blockade. Bioorg Med Chem Lett (2002):12:2569-2572.
    • (2002) Bioorg Med Chem Lett , vol.12 , pp. 2569-2572
    • Palin, R.1    Clark, J.K.2    Cowley, P.3    Muir, A.W.4    Pow, E.5    Prosser, A.B.6    Taylor, R.7    Zhang, M.-Q.8
  • 27
    • 0022625010 scopus 로고
    • Elimination of atracurium in humans: Contribution of Hofmann elimination and ester hydrolysis versus organ-based elimination
    • Fisher DM, Canfell PC, Fahey MR, Rosen JI, Rupp SM, Sheiner LB, Miller RD: Elimination of atracurium in humans: Contribution of Hofmann elimination and ester hydrolysis versus organ-based elimination. Anesthesiology (1986) 65:6-12.
    • (1986) Anesthesiology , vol.65 , pp. 6-12
    • Fisher, D.M.1    Canfell, P.C.2    Fahey, M.R.3    Rosen, J.I.4    Rupp, S.M.5    Sheiner, L.B.6    Miller, R.D.7
  • 28
    • 0017153543 scopus 로고
    • Suxamethonium apnoea terminated with commercial serumcholinesterase
    • Stovner J, Stadskleiv K: Suxamethonium apnoea terminated with commercial serumcholinesterase. Acta Anaesthesiol Scand (1976) 20:211-215.
    • (1976) Acta Anaesthesiol Scand , vol.20 , pp. 211-215
    • Stovner, J.1    Stadskleiv, K.2
  • 29
    • 0029032329 scopus 로고
    • Human plasma cholinesterase for antagonism of prolonged mivacurium-induced neuromuscular blockade
    • Naguib M, el-Gammal M, Daoud W, Ammar A, Moukhtar H, Turkistani A: Human plasma cholinesterase for antagonism of prolonged mivacurium-induced neuromuscular blockade. Anesthesiology (1995) 82:1288-1292.
    • (1995) Anesthesiology , vol.82 , pp. 1288-1292
    • Naguib, M.1    El-Gammal, M.2    Daoud, W.3    Ammar, A.4    Moukhtar, H.5    Turkistani, A.6
  • 30
    • 0029740796 scopus 로고    scopus 로고
    • Edrophonium and human plasma cholinesterase combination for antagonism of mivacurium-induced neuromuscular block
    • Naguib M, Samarkandi AH, Bakhamees HS, Turkistani A, Alharby SW: Edrophonium and human plasma cholinesterase combination for antagonism of mivacurium-induced neuromuscular block. Br J Anaesth (1996) 77:424-426.
    • (1996) Br J Anaesth , vol.77 , pp. 424-426
    • Naguib, M.1    Samarkandi, A.H.2    Bakhamees, H.S.3    Turkistani, A.4    Alharby, S.W.5
  • 31
    • 0029962859 scopus 로고    scopus 로고
    • Enzymatic versus pharmacologic antagonism of profound mivacurium-induced neuromuscular blockade
    • Naguib M, Selim M, Bakhamees HS, Samarkandi AH, Turkistani A: Enzymatic versus pharmacologic antagonism of profound mivacurium-induced neuromuscular blockade. Anesthesiology (1996) 84:1051-1059.
    • (1996) Anesthesiology , vol.84 , pp. 1051-1059
    • Naguib, M.1    Selim, M.2    Bakhamees, H.S.3    Samarkandi, A.H.4    Turkistani, A.5
  • 33
    • 0032500864 scopus 로고    scopus 로고
    • Neuromuscular blocking N,N′-polymethylene bistropanium, 3αhydroxytropanium and bis-3-oxotropanium compounds
    • Gyermek L, Cho YM, Nguyen N, Lee C: Neuromuscular blocking N,N′-polymethylene bistropanium, 3αhydroxytropanium and bis-3-oxotropanium compounds. Life Sci (1998) 63:PL303-PL309.
    • (1998) Life Sci , vol.63
    • Gyermek, L.1    Cho, Y.M.2    Nguyen, N.3    Lee, C.4
  • 34
    • 0001375146 scopus 로고    scopus 로고
    • Neuromuscular blocking bis tropinium glutarate diesters: Optimisation of the benzyl quaternary groups
    • Gyermek L, Cho YM, Nguyen N: Neuromuscular blocking bis tropinium glutarate diesters: Optimisation of the benzyl quaternary groups. Anesth Analg (2001) 92:S199.
    • (2001) Anesth Analg , vol.92
    • Gyermek, L.1    Cho, Y.M.2    Nguyen, N.3
  • 35
    • 0036201675 scopus 로고    scopus 로고
    • Neuromuscular pharmacology of TAAC3, a new nondepolarizing muscle relaxant with rapid onset and ultrashort duration of action
    • Gyermek L, Lee C, Cho YM, Nguyen N, Tsai SK: Neuromuscular pharmacology of TAAC3, a new nondepolarizing muscle relaxant with rapid onset and ultrashort duration of action. Anesth Analg (2002) 94:879-885. The paper presents the most recent results in the quest for ultra-short acting neuromuscular blockers, discovered after optimization of the bistropaninium series of compounds.
    • (2002) Anesth Analg , vol.94 , pp. 879-885
    • Gyermek, L.1    Lee, C.2    Cho, Y.M.3    Nguyen, N.4    Tsai, S.K.5
  • 38
    • 0013348866 scopus 로고    scopus 로고
    • American Society of Anesthesiologist 1999 Annual Meeting (Part II)
    • October 9-13
    • Gotta AW: American Society of Anesthesiologist 1999 Annual Meeting (Part II). Dallas, TX, USA IDdb3 Meeting Report (1999) October 9-13. www.iddb3.com
    • (1999) Dallas, TX, USA IDdb3 Meeting Report
    • Gotta, A.W.1
  • 39
    • 0013348653 scopus 로고    scopus 로고
    • Legal information
    • Barcelona, Spain
    • Legal information. Prous Science, Barcelona, Spain. www.prous.com/legal.html
    • Prous Science
  • 40
    • 0037127108 scopus 로고    scopus 로고
    • A novel concept of reversing neuromuscular block: Chemical encapsulation of rocuronium bromide by a cyclodextrin-based synthetic host
    • Bom A, Bradley M, Cameron K, Clark JK, Egmond J van, Feilden H, MacLean EJ, Muir AW, Palin R, Rees DC, Zhang M-Q: A novel concept of reversing neuromuscular block: Chemical encapsulation of rocuronium bromide by a cyclodextrin-based synthetic host. Angew Chem Int Ed (2002) 41:265-270. This is the first report demonstrating that host-guest chemistry can provide a potent pharmacological agent, both in vitro and in vivo.
    • (2002) Angew Chem Int Ed , vol.41 , pp. 265-270
    • Bom, A.1    Bradley, M.2    Cameron, K.3    Clark, J.K.4    Egmond, J.5    Van Feilden, H.6    MacLean, E.J.7    Muir, A.W.8    Palin, R.9    Rees, D.C.10    Zhang, M.-Q.11
  • 41
    • 0037171790 scopus 로고    scopus 로고
    • Cyclodextrin-derived host molecules as reversal agents for the neuromuscular blocker rocuronium bromide: Synthesis and structure-activity relationships
    • Adam JM, Bennett DJ, Bom A, Clark JK, Feilden H, Hutchinson EJ, Palin R, Prosser A, Rees DC, Rosair GM, Stevenson D et al: Cyclodextrin-derived host molecules as reversal agents for the neuromuscular blocker rocuronium bromide: Synthesis and structure-activity relationships. J Med Chem (2002) 45:1806-1816. This paper describes the structure-activity of functionalized cyclodextrin derivatives with high binding affinity for rocuronium bromide, and the resultant rapid reversal of NMB.
    • (2002) J Med Chem , vol.45 , pp. 1806-1816
    • Adam, J.M.1    Bennett, D.J.2    Bom, A.3    Clark, J.K.4    Feilden, H.5    Hutchinson, E.J.6    Palin, R.7    Prosser, A.8    Rees, D.C.9    Rosair, G.M.10    Stevenson, D.11
  • 42
    • 0015290518 scopus 로고
    • The effects of germine-3-acetate on neuromuscular transmission
    • Detwiler PB: The effects of germine-3-acetate on neuromuscular transmission. J Pharmacol Exp Ther (1972) 180:244-254.
    • (1972) J Pharmacol Exp Ther , vol.180 , pp. 244-254
    • Detwiler, P.B.1
  • 43
    • 0014743746 scopus 로고
    • The neuromuscular pharmacology of germine-3-acetate and germine-3,16diacetate
    • Standaert FG, Detwiler PB: The neuromuscular pharmacology of germine-3-acetate and germine-3,16diacetate. J Pharmacol Exp Ther (1970) 171:223-241.
    • (1970) J Pharmacol Exp Ther , vol.171 , pp. 223-241
    • Standaert, F.G.1    Detwiler, P.B.2
  • 45
    • 0023819511 scopus 로고
    • 2purinoceptor antagonist in the mouse vas deferens
    • 2purinoceptor antagonist in the mouse vas deferens. Br J Pharmacol (1988) 93:243-245.
    • (1988) Br J Pharmacol , vol.93 , pp. 243-245
    • Dunn, P.M.1    Blakely, A.G.2
  • 47
    • 0027407137 scopus 로고
    • Reversal by suramin of neuromuscular block produced by pancuronium in the anaesthetized rat
    • Henning RH, Nelemans A, Houwertjes M, Agoston S: Reversal by suramin of neuromuscular block produced by pancuronium in the anaesthetized rat. Br J Pharmacol (1993) 108:717-720.
    • (1993) Br J Pharmacol , vol.108 , pp. 717-720
    • Henning, R.H.1    Nelemans, A.2    Houwertjes, M.3    Agoston, S.4
  • 48
    • 0029992807 scopus 로고    scopus 로고
    • The prejunctional inhibitory effect of suramin on neuromuscular transmission in vitro
    • Henning RH, Rowan EG, Braga MF, Nelemans A, Harvey AL: The prejunctional inhibitory effect of suramin on neuromuscular transmission in vitro. Eur J Pharmacol (1996) 301:91-97.
    • (1996) Eur J Pharmacol , vol.301 , pp. 91-97
    • Henning, R.H.1    Rowan, E.G.2    Braga, M.F.3    Nelemans, A.4    Harvey, A.L.5
  • 49
    • 0025832625 scopus 로고
    • Reversibility of the neuromuscular blocking effects of active components of the malayan cobra (naja naja sputatrix) venom in the presence of heparin
    • Geh SL: Reversibility of the neuromuscular blocking effects of active components of the malayan cobra (naja naja sputatrix) venom in the presence of heparin. Asia Pacif J Pharmacol (1991) 6:81-85.
    • (1991) Asia Pacif J Pharmacol , vol.6 , pp. 81-85
    • Geh, S.L.1
  • 50
    • 0013393440 scopus 로고    scopus 로고
    • drug-induced neuromuscular block. WO-00112202 (2001)
    • ORGANON LABORATORIES LTD (Bom A, Muir A, Rees DC): drug-induced neuromuscular block. WO-00112202 (2001).
    • Bom, A.1    Muir, A.2    Rees, D.C.3
  • 51
    • 0013398129 scopus 로고    scopus 로고
    • 6-Mercapto-cyclodextrin derivatives: Reversal agents for drug-induced neuromuscular block. WO-00140316 (2001)
    • ORGANON LABORATORIES LTD (Zhang M-Q, Palin R, Bennet JD): 6-Mercapto-cyclodextrin derivatives: Reversal agents for drug-induced neuromuscular block. WO-00140316 (2001).
    • Zhang, M.-Q.1    Palin, R.2    Bennet, J.D.3


* 이 정보는 Elsevier사의 SCOPUS DB에서 KISTI가 분석하여 추출한 것입니다.