Desensitization of the mouse thromboxane A2 receptor (TP) by G protein-coupled receptor kinases (GRKs)

Prostaglandins and Other Lipid Mediators

Volumn 70, Issue 1-2, 2002, Pages 79-90

  Flannery, Patrick J ^a   Spurney, Robert F ^a  

^a DURHAM VA MEDICAL CENTER   (United States)

Author keywords

Desensitization; Eicosanoid; G protein coupled receptor kinase; Thromboxane

Indexed keywords

15 HYDROXY 11ALPHA,9ALPHA EPOXYMETHANOPROSTA 5,13 DIENOIC ACID; 7 [3 [(4 PHENYLSEMICARBAZIDO)METHYL] 7 OXABICYCLO[2.2.1]HEPT 2 YL] 5 HEPTENOIC ACID; ALANINE; G PROTEIN COUPLED RECEPTOR; G PROTEIN COUPLED RECEPTOR KINASE; MUTANT PROTEIN; THREONINE; THROMBOXANE A2; THROMBOXANE A2 RECEPTOR; THROMBOXANE A2 RECEPTOR BLOCKING AGENT; THROMBOXANE A2 RECEPTOR STIMULATING AGENT;

AMINO ACID SUBSTITUTION; ANIMAL CELL; ARTICLE; BINDING AFFINITY; CELL CULTURE; COLUMN CHROMATOGRAPHY; CONTROLLED STUDY; DESENSITIZATION; DRUG EFFECT; EMBRYO; ENZYME ACTIVITY; HUMAN; HUMAN CELL; MOLECULAR CLONING; MOUSE; NONHUMAN; PHOSPHORYLATION; PROTEIN EXPRESSION; PROTEIN MOTIF; RAT; REVERSE TRANSCRIPTION POLYMERASE CHAIN REACTION; SEQUENCE HOMOLOGY; WILD TYPE;

15-HYDROXY-11 ALPHA,9 ALPHA-(EPOXYMETHANO)PROSTA-5,13-DIENOIC ACID; AMINO ACID SEQUENCE; AMINO ACID SUBSTITUTION; ANIMALS; BETA-ADRENERGIC RECEPTOR KINASE; CELL LINE; CYCLIC AMP-DEPENDENT PROTEIN KINASES; GLOMERULAR MESANGIUM; MICE; MICE, TRANSGENIC; PHORBOL 12,13-DIBUTYRATE; PHOSPHORYLATION; PROTEIN KINASE C; RECEPTORS, THROMBOXANE; THREONINE; THROMBOXANE A2;

EID: 0036744127     PISSN: 00906980     EISSN: None     Source Type: Journal    
DOI: 10.1016/S0090-6980(02)00013-8     Document Type: Article

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