Agents that elevate cyclic AMP induce receptor phosphorylation primarily at serine 331 in HEK 293 cells overexpressing human thromboxane receptor α

Biochemical Pharmacology

Volumn 64, Issue 3, 2002, Pages 375-383

  Yamamoto, Shuichi ^a   Yan, Fengxiang ^a   Zhou, Huiping ^a   Tai, Hsin Hsiung ^a  

^a University of Kentucky   (United States)

Author keywords

Cyclic AMP; Desensitization; Phosphorylation; Prostaglandin E1; Protein kinase A; Receptor; Thromboxane A2

Indexed keywords

(1ALPHA,2ALPHA,3BETA,4ALPHA) 7 [3 [3 HYDROXY 4 (4 INDOPHENOXY) 1 BUTENYL] 7 OXABICYCLO[2,2,1]HEPT 2 YL] 5 HEPTENOIC ACID; 7 [3 [(4 PHENYLSEMICARBAZIDO)METHYL] 7 OXABICYCLO[2.2.1]HEPT 2 YL] 5 HEPTENOIC ACID; ALANINE; ANTIBIOTIC G 418; CALCIUM CHANNEL STIMULATING AGENT; CYCLIC AMP; CYCLIC AMP DEPENDENT PROTEIN KINASE; FORSKOLIN; MUTANT PROTEIN; PROSTAGLANDIN E1; SERINE; THREONINE; THROMBOXANE RECEPTOR; THROMBOXANE RECEPTOR ALPHA; UNCLASSIFIED DRUG;

ARTICLE; CALCIUM TRANSPORT; CHEMICAL LABELING; CONCENTRATION RESPONSE; CONTROLLED STUDY; DRUG EFFECT; EMBRYO CELL; ENZYME ACTIVATION; ENZYME PURIFICATION; ENZYME SUBSTRATE; GENE OVEREXPRESSION; HUMAN; HUMAN CELL; KIDNEY CELL; PRIORITY JOURNAL; PROTEIN ANALYSIS; PROTEIN DOMAIN; PROTEIN PHOSPHORYLATION; RECEPTOR DOWN REGULATION;

ALPROSTADIL; CELLS, CULTURED; CYCLIC AMP; EPOPROSTENOL; HUMANS; PHOSPHORYLATION; PLATELET AGGREGATION INHIBITORS; PROSTAGLANDIN D2; RECEPTORS, THROMBOXANE; SERINE;

EID: 0036685195     PISSN: 00062952     EISSN: None     Source Type: Journal    
DOI: 10.1016/S0006-2952(02)01053-5     Document Type: Article

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