SCOPUS 정보 검색 플랫폼

Volumn 653, Issue 1-2, 2002, Pages 269-278

Investigations into the Suzuki-Miyaura coupling aiming at multikilogram synthesis of E2040 using (o-cyanophenyl)boronic esters

(5) Urawa, Yoshio a,b Naka, Hiroyuki a Miyazawa, Mamoru a Souda, Shigeru a Ogura, Katsuyuki b

a EISAI CO LTD (Japan)

b CHIBA UNIVERSITY (Japan)

Author keywords

DOE; E2040; Reductive debromination; Scale up; Suzuki Miyaura cross coupling

Indexed keywords

1 PHENYLPIPERAZINE DERIVATIVE; BORONIC ACID DERIVATIVE; BROMINE DERIVATIVE; E 2040; ESTER DERIVATIVE; PALLADIUM COMPLEX; PHOSPHINE DERIVATIVE; POTASSIUM DIHYDROGEN PHOSPHATE; SEROTONIN 2 ANTAGONIST; TOLUENE; TRIPHENYLPHOSPHINE; UNCLASSIFIED DRUG;

ARTICLE; CHEMICAL REACTION; CONTROLLED STUDY; DRUG STRUCTURE; DRUG SYNTHESIS; EXPERIMENTAL DESIGN; METHODOLOGY; SAFETY; THERMOSTABILITY;

LATEOLABRAX JAPONICUS;

EID: 0036643510 PISSN: 0022328X EISSN: None Source Type: Journal
DOI: 10.1016/S0022-328X(02)01175-0 Document Type: Article

Times cited : (38)

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