Pharmacological characterization of the ATP-dependent low Km guanosine 3′,5′-cyclic monophosphate (cGMP) transporter in human erythrocytes

Biochemical Pharmacology

Volumn 63, Issue 5, 2002, Pages 945-949

  Sundkvist, Elisabeth ^a   Jaeger, Ragnhild ^a   Sager, Georg ^a  

^a UNIVERSITY OF TROMSØ   (Norway)

Author keywords

cGMP; Cytotoxic drugs; Phosphodiesterase inhibitors; Purines; Steroids; Transport

Indexed keywords

4 AMINOHIPPURIC ACID; 6 MERCAPTOPURINE DERIVATIVE; 6 THIOGUANOSINE 5' MONOPHOSPHATE; ADEFOVIR; CARRIER PROTEIN; CYCLIC GMP; DAUNORUBICIN; DIPYRIDAMOLE; DOXORUBICIN; ESTRADIOL; ESTRADIOL 17 GLUCURONIDE; ESTRADIOL 3 BETA GLUCURONIDE; ESTRADIOL DERIVATIVE; GENISTEIN; GUANOSINE DERIVATIVE; MEDROXYPROGESTERONE; MEGESTROL ACETATE; MERCAPTOPURINE; METHOTREXATE; METHYLMERCAPTOPURINE; MIFEPRISTONE; ONAPRISTONE; PROGESTERONE; SILDENAFIL; SULFINPYRAZONE; TAUROCHOLIC ACID; TIOGUANINE; UNCLASSIFIED DRUG; UNINDEXED DRUG; VINCRISTINE; ZAPRINAST;

ARTICLE; BINDING AFFINITY; CELL VACUOLE; CONTROLLED STUDY; DRUG BINDING; DRUG EFFECT; DRUG POTENCY; DRUG UPTAKE; ERYTHROCYTE; HUMAN; HUMAN CELL; ION TRANSPORT; PRIORITY JOURNAL; PROTEIN ANALYSIS;

ADENOSINE TRIPHOSPHATE; ANTHRACYCLINES; BIOLOGICAL TRANSPORT; CYCLIC GMP; ERYTHROCYTES; ESTRADIOL; HUMANS; METHOTREXATE; PHOSPHODIESTERASE INHIBITORS; PROGESTINS; VINCRISTINE;

EID: 0036496833     PISSN: 00062952     EISSN: None     Source Type: Journal    
DOI: 10.1016/S0006-2952(01)00940-6     Document Type: Article

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10. 4) does not share a cellular efflux mechanism with cGMP: Characterisation of cGMP transport by uptake to inside-out vesicles from human erythrocytes
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12. 50) of an enzymatic reaction
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