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Volumn 46, Issue 5, 2002, Pages 389-393

New insights into the pharmacological properties of potent antiplatelet 2-amino-benzo[d]isothiazol-3-one derivatives

Author keywords

Antiplatelet drugs; Benzoisothiazolone; Bleeding; Experimental thrombosis; Subacute treatment

Indexed keywords

15 HYDROXY 11ALPHA,9ALPHA EPOXYMETHANOPROSTA 5,13 DIENOIC ACID; ADRENALIN; ANTITHROMBOCYTIC AGENT; COLLAGEN; ISOTHIAZOLE DERIVATIVE; LYSINE ACETYLSALICYLATE; 2 AMINO BENZO(D)ISOTHIAZOL 3 ONE; 2-AMINO-BENZO(D)ISOTHIAZOL-3-ONE; CHOLINERGIC RECEPTOR BLOCKING AGENT; THIAZOLE DERIVATIVE;

EID: 0036433112     PISSN: 10436618     EISSN: None     Source Type: Journal    
DOI: 10.1016/S1043661802002086     Document Type: Article
Times cited : (7)

References (25)
  • 1
    • 0028120906 scopus 로고
    • Collaborative overview of randomized trials of platelet therapy. I. Prevention of death, infarction and stroke by prolonged antiplatelet therapy in various categories of patients
    • Antiplatelet Trialists' Collaboration. Collaborative overview of randomized trials of platelet therapy. I. Prevention of death, infarction and stroke by prolonged antiplatelet therapy in various categories of patients. Br Med J 1994; 308: 81-106.
    • (1994) Br Med J , vol.308 , pp. 81-106
  • 2
    • 0032474229 scopus 로고    scopus 로고
    • Second International Study of Infarct Survival (ISIS-2 Collaborative group): 10 years survival among patients with suspected acute myocardial infarction in randomized comparison of intravenous streptokinase, oral aspirin, both or neither
    • Baigent C, Collins R, Appleby P, Parish S, Sleight P, Peto R. Second International Study of Infarct Survival (ISIS-2 Collaborative group): 10 years survival among patients with suspected acute myocardial infarction in randomized comparison of intravenous streptokinase, oral aspirin, both or neither. Br Med J 1998; 316: 1337-43.
    • (1998) Br Med J , vol.316 , pp. 1337-1343
    • Baigent, C.1    Collins, R.2    Appleby, P.3    Parish, S.4    Sleight, P.5    Peto, R.6
  • 3
    • 0032189870 scopus 로고    scopus 로고
    • Antiplatelet therapy in coronary artery disease: Review and update of efficacy studies
    • Tisdale JE. Antiplatelet therapy in coronary artery disease: Review and update of efficacy studies. Am J Health-Syst Pharm 1998; 55(Suppl): S8-16.
    • (1998) Am J Health-Syst Pharm , vol.55 , Issue.SUPPL.
    • Tisdale, J.E.1
  • 4
    • 0028354308 scopus 로고
    • Aspirin as antiplatelet drug
    • Patrono C. Aspirin as antiplatelet drug. New Engl J Med 1994; 330: 1287-94.
    • (1994) New Engl J Med , vol.330 , pp. 1287-1294
    • Patrono, C.1
  • 5
    • 0031037170 scopus 로고    scopus 로고
    • Gastric toxicity of antiplatelet therapy with low dose aspirin
    • Guslandi M. Gastric toxicity of antiplatelet therapy with low dose aspirin. Drugs 1997; 53: 1-5.
    • (1997) Drugs , vol.53 , pp. 1-5
    • Guslandi, M.1
  • 6
    • 0030780194 scopus 로고    scopus 로고
    • Synthesis and antiplatelet effects of 2-amino-1,2-benziso-thiazolin-3-one
    • Vicini P, Manotti C, Caretta A, Amoretti L. Synthesis and antiplatelet effects of 2-amino-1,2-benziso-thiazolin-3-one. Arzneimittelforschung 1997; 47: 1218-21.
    • (1997) Arzneimittelforschung , vol.47 , pp. 1218-1221
    • Vicini, P.1    Manotti, C.2    Caretta, A.3    Amoretti, L.4
  • 7
    • 0032756925 scopus 로고    scopus 로고
    • Comparison of in vitro and ex vivo antiplatelet effects of 1,2-benzisothiazolin-3-one and its 2-amino derivative
    • Vicini P, Manotti C, Caretta A, Amoretti L. Comparison of in vitro and ex vivo antiplatelet effects of 1,2-benzisothiazolin-3-one and its 2-amino derivative. Arzneimittelforschung 1999; 49: 896-9.
    • (1999) Arzneimittelforschung , vol.49 , pp. 896-899
    • Vicini, P.1    Manotti, C.2    Caretta, A.3    Amoretti, L.4
  • 8
    • 0033868980 scopus 로고    scopus 로고
    • 2-Amino-1,2-benzisothiazolin-3-one derivatives: Synthesis and assessement of their antiplatelet/spasmolytic effects
    • Vicini P, Amoretti L, Ballabeni V, Tognolini M, Barocelli E. 2-Amino-1,2-benzisothiazolin-3-one derivatives: Synthesis and assessement of their antiplatelet/spasmolytic effects. Bioorg Med Chem 2000; 8: 2355-8.
    • (2000) Bioorg Med Chem , vol.8 , pp. 2355-2358
    • Vicini, P.1    Amoretti, L.2    Ballabeni, V.3    Tognolini, M.4    Barocelli, E.5
  • 9
    • 0026532713 scopus 로고
    • Effects of the new antiplatelet agent 2-methyl-3-(1,4,5,6-tetrahydronicotinoyl)pyrazolo[1,5-a]pyridine on platelet aggregation and thrombosis in experimental animals
    • Momo K, Someya K, Tachiiri T, Mitsuoka Y, Nakamura K, Imai S, Ino T, Ohkubo H. Effects of the new antiplatelet agent 2-methyl-3-(1,4,5,6-tetrahydronicotinoyl)pyrazolo[1,5-a]pyridine on platelet aggregation and thrombosis in experimental animals. Arzneimittelforschung 1992; 42: 32-9.
    • (1992) Arzneimittelforschung , vol.42 , pp. 32-39
    • Momo, K.1    Someya, K.2    Tachiiri, T.3    Mitsuoka, Y.4    Nakamura, K.5    Imai, S.6    Ino, T.7    Ohkubo, H.8
  • 10
    • 0020582095 scopus 로고
    • Mouse antithrombotic assay: A simple method for the evaluation of antithrombotic agents in vivo. Potentiation of antithrombotic activity by ethyl alcohol
    • DiMinno G. Mouse antithrombotic assay: A simple method for the evaluation of antithrombotic agents in vivo. Potentiation of antithrombotic activity by ethyl alcohol. J Pharmacol Exp Ther 1983; 225: 57-60.
    • (1983) J Pharmacol Exp Ther , vol.225 , pp. 57-60
    • DiMinno, G.1
  • 11
    • 0018745986 scopus 로고
    • Bleeding time in laboratory animals. II. A comparison of different assay conditions in rats
    • Dejana E, Callioni A, Quintana A, De Gaetano G. Bleeding time in laboratory animals. II. A comparison of different assay conditions in rats. Thromb Res 1979; 15: 191-7.
    • (1979) Thromb Res , vol.15 , pp. 191-197
    • Dejana, E.1    Callioni, A.2    Quintana, A.3    De Gaetano, G.4
  • 12
    • 0023228240 scopus 로고
    • Gastric ulcerogenicity of non-steroidal anti-inflammatory drugs in mice with mucosa sensitized by cholinomimetic treatment
    • Rainsford KD. Gastric ulcerogenicity of non-steroidal anti-inflammatory drugs in mice with mucosa sensitized by cholinomimetic treatment. J Pharm Pharmacol 1987; 39: 669-72.
    • (1987) J Pharm Pharmacol , vol.39 , pp. 669-672
    • Rainsford, K.D.1
  • 14
    • 0346367328 scopus 로고
    • Aggregation by ADP and its reversal
    • Born GVR. Aggregation by ADP and its reversal. Nature 1962; 194: 927-9.
    • (1962) Nature , vol.194 , pp. 927-929
    • Born, G.V.R.1
  • 15
    • 0000328674 scopus 로고
    • Blanschko H, Muscholl E, eds. New York: Springer
    • Furchgott RF. In: Blanschko H, Muscholl E, eds. Handbook of experimental pharmacology, vol. 33. New York: Springer, 1972: 283-335.
    • (1972) Handbook of Experimental Pharmacology , vol.33 , pp. 283-335
    • Furchgott, R.F.1
  • 16
    • 0028896122 scopus 로고
    • Determination of the structure of two novel echistatin variants and comparison of the ability of echistatin variants to inhibit aggregation of platelets from different species
    • Chen YL, Huang TF, Chen SW, Tsai IH. Determination of the structure of two novel echistatin variants and comparison of the ability of echistatin variants to inhibit aggregation of platelets from different species. Biochem J 1995; 305: 513-20.
    • (1995) Biochem J , vol.305 , pp. 513-520
    • Chen, Y.L.1    Huang, T.F.2    Chen, S.W.3    Tsai, I.H.4
  • 18
    • 0029153165 scopus 로고
    • New antiplatelet agents: Platelet GPIIb/IIIa antagonists
    • Coller BS, Anderson K, Weisman HF. New antiplatelet agents: Platelet GPIIb/IIIa antagonists. Thromb Haemost 1995; 74: 302-8.
    • (1995) Thromb Haemost , vol.74 , pp. 302-308
    • Coller, B.S.1    Anderson, K.2    Weisman, H.F.3
  • 19
    • 0034038930 scopus 로고    scopus 로고
    • Antiplatelet and antithrombotic effects of a novel selective phosphodiesterase 3 inhibitor, NSP-513, in mice and rats
    • Hirose H, Kimura T, Okada M, Itoh Y, Ishida F, Mochizuki N, Nishibe T, Nishikibe M. Antiplatelet and antithrombotic effects of a novel selective phosphodiesterase 3 inhibitor, NSP-513, in mice and rats. Jpn J Pharmacol 2000; 82: 188-98.
    • (2000) Jpn J Pharmacol , vol.82 , pp. 188-198
    • Hirose, H.1    Kimura, T.2    Okada, M.3    Itoh, Y.4    Ishida, F.5    Mochizuki, N.6    Nishibe, T.7    Nishikibe, M.8
  • 20
    • 0030054350 scopus 로고    scopus 로고
    • Blood cardiolipin in haemodialysis patients. Its implication in the biological action of platelet-activating factor
    • Antonopoulou S, Demopoulos CA, Iatrou C. Blood cardiolipin in haemodialysis patients. Its implication in the biological action of platelet-activating factor. Int J Biochem Cell Biol 1996; 28: 43-51.
    • (1996) Int J Biochem Cell Biol , vol.28 , pp. 43-51
    • Antonopoulou, S.1    Demopoulos, C.A.2    Iatrou, C.3
  • 21
    • 0002920771 scopus 로고
    • Platelet thrombosis induced by adenosine diphosphate in the rat
    • Nordoy A, Chandler AB. Platelet thrombosis induced by adenosine diphosphate in the rat. Scand J Haematol 1964; 1: 16-21.
    • (1964) Scand J Haematol , vol.1 , pp. 16-21
    • Nordoy, A.1    Chandler, A.B.2
  • 24
    • 0029610590 scopus 로고
    • Triflavin, an Arg-Gly-Asp-containing peptide, prevents platelet plug formation in in vivo experiments
    • Sheu JR, Yen MH, Peng HC, Chang MC, Huang TF. Triflavin, an Arg-Gly-Asp-containing peptide, prevents platelet plug formation in in vivo experiments. Eur J Pharmacol 1995; 294: 231-7.
    • (1995) Eur J Pharmacol , vol.294 , pp. 231-237
    • Sheu, J.R.1    Yen, M.H.2    Peng, H.C.3    Chang, M.C.4    Huang, T.F.5
  • 25
    • 0028899167 scopus 로고
    • Effect of pheniramine, chlorpheniramine and brompheniramine on stimulated blood platelet: Structure-activity relationships
    • Jancinova V, Petrikova M, Majekova M, Nosal R. Effect of pheniramine, chlorpheniramine and brompheniramine on stimulated blood platelet: Structure-activity relationships. Inflamm Res 1995; 44: S38-9.
    • (1995) Inflamm Res , vol.44
    • Jancinova, V.1    Petrikova, M.2    Majekova, M.3    Nosal, R.4


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