The rational design of drugs with phos-phonic/phinic acids as enzyme inhibitors isosteric receptor ligands

Phosphorus, Sulfur and Silicon and Related Elements

Volumn 177, Issue 6-7, 2002, Pages 1725-1729

  Ebetino, Frank H ^a   Soper, David L ^a   Dirr, Michelle J ^a   Lundy, Mark W ^a   Mieling, Glen ^a   Wos, John A ^a   DeLong, Mitchell A ^a   Liu, Xuewei ^a  

^a PROCTER AND GAMBLE PHARMACEUTICALS   (United States)

Author keywords

Isosteres; Peptidomimetic; Phosphinic phosphonic acids; Prostaglandins

Indexed keywords

ENZYME INHIBITOR; G PROTEIN COUPLED RECEPTOR; GERANYLTRANSFERASE; PHOSPHINIC ACID DERIVATIVE; PHOSPHONIC ACID DERIVATIVE; PROSTAGLANDIN;

CONFERENCE PAPER; DRUG DESIGN; DRUG SYNTHESIS; ENZYME INHIBITION;

EID: 0036404259     PISSN: 10426507     EISSN: None     Source Type: Journal    
DOI: 10.1080/10426500212317     Document Type: Conference Paper

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