메뉴 건너뛰기




Volumn 164, Issue 1, 2002, Pages 115-120

Comparison of the discriminative and neuroendocrine effects of centrally penetrating κ-opioid agonists in rhesus monkeys

Author keywords

Opioids; Biomarker; Drug discrimination; Prolactin

Indexed keywords

3,4 DICHLORO N METHYL N [2 (1 PYRROLIDINYL)CYCLOHEXYL]BENZENEACETAMIDE; 4 [ALPHA (4 ALLYL 2,5 DIMETHYL 1 PIPERAZINYL) 3 METHOXYBENZYL] N,N DIETHYLBENZAMIDE; BREMAZOCINE; FENTANYL; KAPPA OPIATE RECEPTOR AGONIST; N METHYL N [7 (1 PYRROLIDINYL) 1 OXASPIRO[4.5]DEC 8 YL]BENZENEACETAMIDE; NALBUPHINE; NALMEFENE; PROLACTIN; R 84760; SPIRADOLINE; UNCLASSIFIED DRUG;

EID: 0036402146     PISSN: 00333158     EISSN: None     Source Type: Journal    
DOI: 10.1007/s00213-002-1195-y     Document Type: Article
Times cited : (20)

References (41)
  • 1
    • 0023521010 scopus 로고
    • Early ontogeny of kappa-opioid receptor regulation of prolactin secretion in the rat
    • Bero LA, Lurie SN, Kuhn CM (1987) Early ontogeny of kappa-opioid receptor regulation of prolactin secretion in the rat. Brain Res 465:189-196
    • (1987) Brain Res , vol.465 , pp. 189-196
    • Bero, L.A.1    Lurie, S.N.2    Kuhn, C.M.3
  • 2
    • 0036162288 scopus 로고    scopus 로고
    • The effects of heroin on prolactin levels in male rhesus monkeys: Use of cumulative dosing procedures
    • Bowen CA, Negus SS, Kelly M, Mello NK (2002) The effects of heroin on prolactin levels in male rhesus monkeys: use of cumulative dosing procedures. Psychoneuroendocrinology 27:319-336
    • (2002) Psychoneuroendocrinology , vol.27 , pp. 319-336
    • Bowen, C.A.1    Negus, S.S.2    Kelly, M.3    Mello, N.K.4
  • 4
    • 0032764055 scopus 로고    scopus 로고
    • Apparent efficacy of kappa-opioid receptor ligands on serum prolactin levels in rhesus monkeys
    • Butelman ER, Harris TJ, Kreek M (1999) Apparent efficacy of kappa-opioid receptor ligands on serum prolactin levels in rhesus monkeys. Eur J Pharmacol 383:305-309
    • (1999) Eur J Pharmacol , vol.383 , pp. 305-309
    • Butelman, E.R.1    Harris, T.J.2    Kreek, M.3
  • 6
    • 0035087089 scopus 로고    scopus 로고
    • Enadoline discrimination in squirrel monkeys: Effects of opioid agonists and antagonists
    • Carey GJ, Bergman J (2001) Enadoline discrimination in squirrel monkeys: effects of opioid agonists and antagonists. J Pharmacol Exp Ther 297:215-223
    • (2001) J Pharmacol Exp Ther , vol.297 , pp. 215-223
    • Carey, G.J.1    Bergman, J.2
  • 8
    • 0028911130 scopus 로고
    • Cocaine binges differentially alter striatal preprodynorphin and zif/268 mRNAs
    • Daunais JB, McGinty JF (1995) Cocaine binges differentially alter striatal preprodynorphin and zif/268 mRNAs. Brain Res Mol Brain Res 29:201-210
    • (1995) Brain Res Mol Brain Res , vol.29 , pp. 201-210
    • Daunais, J.B.1    McGinty, J.F.2
  • 10
    • 0023836656 scopus 로고
    • Opposite effects of mu and kappa opiate agonists on dopamine release in the nucleus accumbens and in the dorsal caudate of freely moving rats
    • Di Chiara G, Imperato A (1988) Opposite effects of mu and kappa opiate agonists on dopamine release in the nucleus accumbens and in the dorsal caudate of freely moving rats. J Pharmacol Exp Ther 244:1067-1080
    • (1988) J Pharmacol Exp Ther , vol.244 , pp. 1067-1080
    • Di Chiara, G.1    Imperato, A.2
  • 11
    • 0034111174 scopus 로고    scopus 로고
    • Maximum tolerated dose of nalmefene in patients receiving epidural fentanyl and dilute bupivacaine for postoperative analgesia
    • Dougherty TB, Porche VH, Thall PF (2000) Maximum tolerated dose of nalmefene in patients receiving epidural fentanyl and dilute bupivacaine for postoperative analgesia. Anesthesiology 92:1010-1016
    • (2000) Anesthesiology , vol.92 , pp. 1010-1016
    • Dougherty, T.B.1    Porche, V.H.2    Thall, P.F.3
  • 12
    • 0023626436 scopus 로고
    • Kappa opioids in rhesus monkeys. II. Analysis of the antagonistic actions of quadazocine and beta-funaltrexamine
    • Dykstra LA, Gmerek DE, Winger G, Woods JH (1987a) Kappa opioids in rhesus monkeys. II. Analysis of the antagonistic actions of quadazocine and beta-funaltrexamine. J Pharmacol Exp Ther 242:421-427
    • (1987) J Pharmacol Exp Ther , vol.242 , pp. 421-427
    • Dykstra, L.A.1    Gmerek, D.E.2    Winger, G.3    Woods, J.H.4
  • 13
    • 0023637786 scopus 로고
    • Kappa opioids in rhesus monkeys. I. Diuresis, sedation, analgesia and discriminative stimulus effects
    • Dykstra LA, Gmerek DE, Winger G, Woods JH (1987b) Kappa opioids in rhesus monkeys. I. Diuresis, sedation, analgesia and discriminative stimulus effects. J Pharmacol Exp Ther 242:413-420
    • (1987) J Pharmacol Exp Ther , vol.242 , pp. 413-420
    • Dykstra, L.A.1    Gmerek, D.E.2    Winger, G.3    Woods, J.H.4
  • 14
    • 0028109622 scopus 로고
    • Binding affinity and selectivity of opioids at mu, delta and kappa receptors in monkey brain membranes
    • Emmerson PJ, Liu MR, Woods JH, Medzihradsky F (1994) Binding affinity and selectivity of opioids at mu, delta and kappa receptors in monkey brain membranes. J Pharmacol Exp Ther 271:1630-1637
    • (1994) J Pharmacol Exp Ther , vol.271 , pp. 1630-1637
    • Emmerson, P.J.1    Liu, M.R.2    Woods, J.H.3    Medzihradsky, F.4
  • 15
    • 0028072518 scopus 로고
    • Behavioral effects of 6-methylene naltrexone (nalmefene) in rhesus monkeys
    • France CP, Gerak LR (1994) Behavioral effects of 6-methylene naltrexone (nalmefene) in rhesus monkeys. J Pharmacol Exp Ther 270:992-999
    • (1994) J Pharmacol Exp Ther , vol.270 , pp. 992-999
    • France, C.P.1    Gerak, L.R.2
  • 16
    • 0024414685 scopus 로고
    • Pharmacological characterization of supersensitivity to naltrexone in squirrel monkeys
    • France CP, Morse WH (1989) Pharmacological characterization of supersensitivity to naltrexone in squirrel monkeys. J Pharmacol Exp Ther 250:937-943
    • (1989) J Pharmacol Exp Ther , vol.250 , pp. 937-943
    • France, C.P.1    Morse, W.H.2
  • 17
    • 0028013439 scopus 로고
    • Comparison of kappa opioids in rhesus monkeys: Behavioral effects and receptor binding affinities
    • France CP, Medzihradsky F, Woods JH (1994) Comparison of kappa opioids in rhesus monkeys: behavioral effects and receptor binding affinities. J Pharmacol Exp Ther 268:47-58
    • (1994) J Pharmacol Exp Ther , vol.268 , pp. 47-58
    • France, C.P.1    Medzihradsky, F.2    Woods, J.H.3
  • 18
    • 0028142488 scopus 로고
    • Pharmacological properties of R-84760, a novel kappa-opioid receptor agonist
    • Fujibayashi K, Sakamoto K, Watanabe M, Iizuka Y (1994) Pharmacological properties of R-84760, a novel kappa-opioid receptor agonist. Eur J Pharmacol 261:133-140
    • (1994) Eur J Pharmacol , vol.261 , pp. 133-140
    • Fujibayashi, K.1    Sakamoto, K.2    Watanabe, M.3    Iizuka, Y.4
  • 19
    • 0027223531 scopus 로고
    • The kappa-opioid receptor agonist U-69593 attenuates cocaine-induced behavioral sensitization in the rat
    • Heidbreder CA, Goldberg SR, Shippenberg TS (1993) The kappa-opioid receptor agonist U-69593 attenuates cocaine-induced behavioral sensitization in the rat. Brain Res 616:335-338
    • (1993) Brain Res , vol.616 , pp. 335-338
    • Heidbreder, C.A.1    Goldberg, S.R.2    Shippenberg, T.S.3
  • 20
    • 0023808040 scopus 로고
    • Human studies on the mu opiate receptor agonist fentanyl: Neuroendocrine and behavioral responses
    • Hoehe M, Duka T, Doenicke A (1988) Human studies on the mu opiate receptor agonist fentanyl: neuroendocrine and behavioral responses. Psychoneuroendocrinology 13:397-408
    • (1988) Psychoneuroendocrinology , vol.13 , pp. 397-408
    • Hoehe, M.1    Duka, T.2    Doenicke, A.3
  • 23
    • 0033025795 scopus 로고    scopus 로고
    • Quantitative analysis of R-84760, a selective kappa-opioid receptor agonist, in plasma by liquid chromatography with electrospray ionization tandem mass spectrometry
    • Kobayashi N, Naganuma H (1999) Quantitative analysis of R-84760, a selective kappa-opioid receptor agonist, in plasma by liquid chromatography with electrospray ionization tandem mass spectrometry. J Pharm Biomed Anal 19:829-836
    • (1999) J Pharm Biomed Anal , vol.19 , pp. 829-836
    • Kobayashi, N.1    Naganuma, H.2
  • 24
    • 0034723054 scopus 로고    scopus 로고
    • Opioid receptor and peptide gene polymorphisms: Potential implications for addictions
    • LaForge KS, Yuferov V, Kreek MJ (2000) Opioid receptor and peptide gene polymorphisms: potential implications for addictions. Eur J Pharmacol 410:249-268
    • (2000) Eur J Pharmacol , vol.410 , pp. 249-268
    • LaForge, K.S.1    Yuferov, V.2    Kreek, M.J.3
  • 25
    • 0034045604 scopus 로고    scopus 로고
    • Acute effects of nalmefene on LH, prolactin, and testosterone in male rhesus monkeys
    • Mello NK, Mendelson JH, Kelly M (2000) Acute effects of nalmefene on LH, prolactin, and testosterone in male rhesus monkeys. Pharmacol Biochem Behav 66:275-283
    • (2000) Pharmacol Biochem Behav , vol.66 , pp. 275-283
    • Mello, N.K.1    Mendelson, J.H.2    Kelly, M.3
  • 26
    • 0025742665 scopus 로고
    • Neurons with access to the general circulation in the central nervous system of the rat: A retrograde tracing study with fluoro-gold
    • Merchenthaler I (1991) Neurons with access to the general circulation in the central nervous system of the rat: a retrograde tracing study with fluoro-gold. Neuroscience 44:655-662
    • (1991) Neuroscience , vol.44 , pp. 655-662
    • Merchenthaler, I.1
  • 27
    • 0002131424 scopus 로고
    • Dopaminergic neuronal systems in the hypothalamus
    • Bloom FE, Kupfer DJ (eds). Raven Press, New York
    • Moore KE, Lookingland KJ (1995) Dopaminergic neuronal systems in the hypothalamus. In: Bloom FE, Kupfer DJ (eds) Psychopharmacology: the fourth generation of progress. Raven Press, New York, pp 245-256
    • (1995) Psychopharmacology: The Fourth Generation of Progress , pp. 245-256
    • Moore, K.E.1    Lookingland, K.J.2
  • 28
    • 0027495926 scopus 로고
    • Effects of opioid agonists selective for mu, kappa and delta opioid receptors on schedule-controlled responding in rhesus monkeys: Antagonism by quadazocine
    • Negus SS, Burke TF, Medzihradsky F, Woods JH (1993) Effects of opioid agonists selective for mu, kappa and delta opioid receptors on schedule-controlled responding in rhesus monkeys: antagonism by quadazocine. J Pharmacol Exp Ther 267:896-903
    • (1993) J Pharmacol Exp Ther , vol.267 , pp. 896-903
    • Negus, S.S.1    Burke, T.F.2    Medzihradsky, F.3    Woods, J.H.4
  • 29
    • 0003285230 scopus 로고    scopus 로고
    • Biomarkers and surrogate endpoints in clinical research: Definitions and conceptual model
    • Downing GJ (ed). Elsevier, Amsterdam
    • NIH Definitions Working Group (2000) Biomarkers and surrogate endpoints in clinical research: definitions and conceptual model. In: Downing GJ (ed) Biomarkers and surrogate endpoints: clinical research and applications. Elsevier, Amsterdam
    • (2000) Biomarkers and Surrogate Endpoints: Clinical Research and Applications
  • 30
    • 0022494591 scopus 로고
    • Psychotomimesis mediated by kappa opiate receptors
    • Pfeiffer A, Brantl V, Herz A, Emrich HM (1986a) Psychotomimesis mediated by kappa opiate receptors. Science 233:774-776
    • (1986) Science , vol.233 , pp. 774-776
    • Pfeiffer, A.1    Brantl, V.2    Herz, A.3    Emrich, H.M.4
  • 32
    • 0027940660 scopus 로고
    • Drug discrimination assessment of agonist-antagonist opioids in humans: A three-choice saline-hydromorphone-butorphanol procedure
    • Preston KL, Bigelow GE (1994) Drug discrimination assessment of agonist-antagonist opioids in humans: a three-choice saline-hydromorphone-butorphanol procedure. J Pharmacol Exp Ther 271:48-60
    • (1994) J Pharmacol Exp Ther , vol.271 , pp. 48-60
    • Preston, K.L.1    Bigelow, G.E.2
  • 33
    • 0028297606 scopus 로고
    • The cardiovascular and central nervous system effects in the human of U-62066E. A selective opioid receptor agonist
    • Rimoy GH, Wright DM, Bhaskar NK, Rubin PC (1994) The cardiovascular and central nervous system effects in the human of U-62066E. A selective opioid receptor agonist. Eur J Clin Pharmacol 46:203-207
    • (1994) Eur J Clin Pharmacol , vol.46 , pp. 203-207
    • Rimoy, G.H.1    Wright, D.M.2    Bhaskar, N.K.3    Rubin, P.C.4
  • 34
    • 0034545699 scopus 로고    scopus 로고
    • A double blind, placebo controlled study of the tolerability and efficacy of a new kappa-opioid receptor agonist (R-84760) in patients with pain after dental surgery
    • Seymour RA, Stassen L, Moore U, Hawkesford JE, Oshima T, Suggi M, Nimmo WS (2000) A double blind, placebo controlled study of the tolerability and efficacy of a new kappa-opioid receptor agonist (R-84760) in patients with pain after dental surgery. Clin Drug Invest 20:409-414
    • (2000) Clin Drug Invest , vol.20 , pp. 409-414
    • Seymour, R.A.1    Stassen, L.2    Moore, U.3    Hawkesford, J.E.4    Oshima, T.5    Suggi, M.6    Nimmo, W.S.7
  • 35
    • 0026559951 scopus 로고
    • Opposing tonically active endogenous opioid systems modulate the mesolimbic dopaminergic pathway
    • Spanagel R, Herz A, Shippenberg TS (1992) Opposing tonically active endogenous opioid systems modulate the mesolimbic dopaminergic pathway. Proc Natl Acad Sci USA 89:2046-2050
    • (1992) Proc Natl Acad Sci USA , vol.89 , pp. 2046-2050
    • Spanagel, R.1    Herz, A.2    Shippenberg, T.S.3
  • 36
    • 0030612008 scopus 로고    scopus 로고
    • Kappa2 opioid receptors in limbic areas of the human brain are upregulated by cocaine in fatal overdose victims
    • Staley JK, Rothman RB, Rice KC, Partilla J, Mash DC (1997) Kappa2 opioid receptors in limbic areas of the human brain are upregulated by cocaine in fatal overdose victims. J Neurosci 17:8225-8233
    • (1997) J Neurosci , vol.17 , pp. 8225-8233
    • Staley, J.K.1    Rothman, R.B.2    Rice, K.C.3    Partilla, J.4    Mash, D.C.5
  • 37
    • 0032949540 scopus 로고    scopus 로고
    • U50,488 and the kappa-receptor: A personalized account covering 1973 to 1990
    • Jucker E (ed). Birkhauser, Basel
    • Szmuszkovicz J (1999) U50,488 and the kappa-receptor: a personalized account covering 1973 to 1990. In: Jucker E (ed) Progress in drug research. Birkhauser, Basel, pp 168-195
    • (1999) Progress in Drug Research , pp. 168-195
    • Szmuszkovicz, J.1
  • 38
    • 0035805085 scopus 로고    scopus 로고
    • The frequency of cocaine administration impacts cocaine-induced receptor alterations
    • Unterwald EM, Kreek MJ, Cuntapay M (2001) The frequency of cocaine administration impacts cocaine-induced receptor alterations. Brain Res 900:103-109
    • (2001) Brain Res , vol.900 , pp. 103-109
    • Unterwald, E.M.1    Kreek, M.J.2    Cuntapay, M.3
  • 39
    • 0030972607 scopus 로고    scopus 로고
    • The effects of spiradoline (U-62066E), a kappa-opioid receptor agonist, on neuroendocrine function in man
    • Ur E, Wright DM, Bouloux PM, Grossman A (1997) The effects of spiradoline (U-62066E), a kappa-opioid receptor agonist, on neuroendocrine function in man. Br J Pharmacol 120:781-784
    • (1997) Br J Pharmacol , vol.120 , pp. 781-784
    • Ur, E.1    Wright, D.M.2    Bouloux, P.M.3    Grossman, A.4
  • 40
    • 0034873586 scopus 로고    scopus 로고
    • Enadoline, a selective kappa opioid agonist: Comparison with butorphanol and hydromorphone in humans
    • Walsh SL, Strain EC, Abreu ME, Bigelow GE (2001) Enadoline, a selective kappa opioid agonist: comparison with butorphanol and hydromorphone in humans. Psychopharmacology 157:151-162
    • (2001) Psychopharmacology , vol.157 , pp. 151-162
    • Walsh, S.L.1    Strain, E.C.2    Abreu, M.E.3    Bigelow, G.E.4
  • 41
    • 0032076332 scopus 로고    scopus 로고
    • Nalmefene: A long-acting opioid antagonist. Clinical applications in emergency medicine
    • Wang DS, Sternbach G, Varon J (1998) Nalmefene: a long-acting opioid antagonist. Clinical applications in emergency medicine. J Emerg Med 16:471-475
    • (1998) J Emerg Med , vol.16 , pp. 471-475
    • Wang, D.S.1    Sternbach, G.2    Varon, J.3


* 이 정보는 Elsevier사의 SCOPUS DB에서 KISTI가 분석하여 추출한 것입니다.