Inhibitory effect and its kinetic analysis of tyrphostin AG1478 on recombinant human protein kinase CK2 holoenzyme

Acta Pharmacologica Sinica

Volumn 23, Issue 6, 2002, Pages 556-561

  Liu, Xin Guang ^a   Liang, Nian Ci ^a  

^a GUANGDONG MEDICAL UNIVERSITY   (China)

Author keywords

Caseins; Holoenzymes; Kinetics; Protein kinases; Recombinant proteins; Tyrphostins

Indexed keywords

4 (3 CHLOROANILINO) 6,7 DIMETHOXYQUINAZOLINE; 5,6 DICHLOROBENZIMIDAZOLE RIBOSIDE; ADENOSINE TRIPHOSPHATE; CASEIN KINASE II; EPIDERMAL GROWTH FACTOR RECEPTOR; GUANOSINE TRIPHOSPHATE; HOLOENZYME; SULFONAMIDE; CASEIN; DNA BINDING PROTEIN; ENZYME INHIBITOR; PROTEIN SERINE THREONINE KINASE; RECOMBINANT PROTEIN; TYRPHOSTIN;

ARTICLE; COMPETITIVE INHIBITION; CONTROLLED STUDY; DRUG EFFECT; DRUG EFFICACY; DRUG POTENCY; DRUG STRUCTURE; ENZYME ACTIVITY; ENZYME INHIBITION; HUMAN; IC 50; KINETICS; STRUCTURE ANALYSIS; DRUG ANTAGONISM; METABOLISM;

CASEIN KINASE II; CASEINS; DNA-BINDING PROTEINS; ENZYME INHIBITORS; GUANOSINE TRIPHOSPHATE; HOLOENZYMES; HUMANS; KINETICS; PROTEIN-SERINE-THREONINE KINASES; RECOMBINANT PROTEINS; TYRPHOSTINS;

EID: 0036269027     PISSN: 16714083     EISSN: None     Source Type: Journal    
DOI: None     Document Type: Article

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