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Current Pharmaceutical Design

Volumn 8, Issue 2, 2002, Pages 111-124

Quantitative structure-activity relationship studies on cholecystokinin antagonists

(1) Gupta, Satya P a

a BIRLA INSTITUTE OF TECHNOLOGY AND SCIENCE (India)

Author keywords

[No Author keywords available]

Indexed keywords

1 (2,3 DIHYDRO 1 METHYL 2 OXO 5 PHENYL 1H 1,4 BENZODIAZEPIN 3 YL) 3 (3 METHYLPHENYL)UREA; 5 PHENYL 1,4 BENZODIAZEPINE; AMINO ACID DERIVATIVE; ASPERLICIN; BENZODIAZEPINE DERIVATIVE; BENZOTRIPT; CHOLECYSTOKININ; CHOLECYSTOKININ A RECEPTOR; CHOLECYSTOKININ A RECEPTOR ANTAGONIST; CHOLECYSTOKININ B RECEPTOR; CHOLECYSTOKININ B RECEPTOR ANTAGONIST; CHOLECYSTOKININ RECEPTOR; CHOLECYSTOKININ RECEPTOR BLOCKING AGENT; CHOLECYSTOKININ RECEPTOR STIMULATING AGENT; CYCLIC NUCLEOTIDE; DEVAZEPIDE; DIAZEPAM; DIBUTYRYL CYCLIC GMP; GASTRIN; GASTRIN RECEPTOR; GASTROINTESTINAL HORMONE; GLUTAMIC ACID DERIVATIVE; MECLOQUALONE; PEPTIDE DERIVATIVE; PEPTIDE HORMONE; PROGLUMIDE; PSEUDOPEPTIDE; QUINAZOLINONE DERIVATIVE; TRYPTOPHAN DERIVATIVE; UNCLASSIFIED DRUG; UNINDEXED DRUG;

ARTICLE; CENTRAL NERVOUS SYSTEM; COMPETITIVE INHIBITION; CONTROLLED STUDY; DISPERSION; DRUG ABSORPTION; DRUG ACTIVITY; DRUG BIOAVAILABILITY; DRUG DEGRADATION; DRUG MECHANISM; DRUG POTENCY; DRUG RECEPTOR BINDING; DRUG STRUCTURE; DRUG SYNTHESIS; HUMAN; HYDROGEN BOND; HYDROPHOBICITY; MOUSE; NONHUMAN; PERIPHERAL NERVOUS SYSTEM; PRIORITY JOURNAL; PROTEIN STRUCTURE; QUANTITATIVE STRUCTURE ACTIVITY RELATION; RAT; STRUCTURE ANALYSIS;

AMINO ACID SEQUENCE; AMINO ACIDS; ANIMALS; BENZODIAZEPINES; CHOLECYSTOKININ; HUMANS; MOLECULAR SEQUENCE DATA; PEPTIDES; QUANTITATIVE STRUCTURE-ACTIVITY RELATIONSHIP; QUINAZOLINES; RECEPTORS, CHOLECYSTOKININ;

EID: 0036234364 PISSN: 13816128 EISSN: None Source Type: Journal
DOI: 10.2174/1381612023396500 Document Type: Article

Times cited : (12)

References (90)

1
- 0018101373
- (London)
- (1978) Nature , vol.274 , pp. 711
- Dockray, G.J.¹ Hutchison, R.A.² Harris, J.B.³ Gregory, R.A.⁴ Runswick, M.J.⁵

2
- 0021965981
- (1985) Neurochem , vol.44 , pp. 1
- Renfeld, J.F.¹

3
- 0022000627
- (1985) Life Sci , vol.36 , pp. 565
- Kerstens, P.J.S.M.¹ Lamers, C.B.H.W.² Jansen, J.B.M.J.³ De Jong, A.J.L.⁴

4
- 0020476561
- (1982) Life Sci , vol.30 , pp. 479
- Morley, J.E.¹

5
- 0021776085
- Neuronal Cholecystokinin
- For a general review see, Eds
- (1985) Ann. N.Y. Acad. Sci , vol.448 , pp. 1
- Vanderhaeghen, J.J.¹ Crawley, J.N.²

6
- 0017782479
- (1977) Nature (London) , vol.270 , pp. 359
- Dockray, G.J.¹ Gregory, R.A.² Hutchinson, J.B.³ Harris, J.I.⁴ Runswick, M.J.⁵

7
- 0017899221
- (1978) J. Biol. Chem , vol.253 , pp. 4022
- Renfeld, J.F.¹

8
- 0017837527
- (1978) J. Proc. Natl. Acad. Sci. U.S.A , vol.75 , pp. 524
- Robberecht, P.¹ Deschodt-Lanckman, M.² Vanderhaeghen, J.³

9
- 0014206556
- (1967) Experentia , vol.23 , pp. 699
- Anatasi, A.¹ Erspamer, V.² Endean, R.³

10
- 0003111499
- Glass, G.B.J., Ed., Raven Press, New York
- (1980) Gastrointestinal Hormones , pp. 169
- Mutt, V.¹

11
- 0023714239
- (1988) Eur. J. Pharmacol , vol.152 , pp. 371
- Vickroy, T.W.¹ Bianchi, B.R.² Kerwin, J.F.³ Kopecka, H.⁴ Nazdan, A.M.⁵

12
- 0026522625
- (1992) Am. J. Physiol , vol.262
- Moran, T.H.¹ Ameglio, P.J.² Schwartz, G.J.³ McHugh, P.R.⁴

13
- 0019222326
- (1980) Science , vol.208 , pp. 1155
- Saito, A.¹ Sankaran, H.² Goldfinde, I.D.³ Williams, J.A.⁴

14
- 2142753559
- (1989) Mol. Pharmacol , vol.46 , pp. 511
- Lin, C.W.¹ Holladay, M.W.² Barret, R.W.³ Wolfram, C.A.W.⁴ Miller, T.R.⁵ Witte, D.⁶ Kerwin J.F., Jr.⁷ Wagennar, F.⁸ Nadzan, A.M.⁹

15
- 0024412584
- (1989) Arch. Gen. Psychiatry , vol.46 , pp. 511
- de Montigny, C.¹

16
- 0025736929
- (1991) Annu. Rev. Pharmacol. Toxicol , vol.31 , pp. 469
- Woodruff, G.N.¹ Hughes, J.²

17
- 0021239236
- (1984) J. Med. Chem , vol.27 , pp. 845
- Penke, B.¹ Hajnal, F.² Lonovics, J.³ Holzinger, G.⁴ Kadar, T.⁵ Telegdy, G.⁶ Rivier, J.⁷

18
- 0021319682
- (1984) Regul. Pept , vol.8 , pp. 51
- Steigerwalt, R.W.¹ Williams, J.A.²

19
- 2142753558
- (1987) Regul. Pept , vol.18 , pp. 107
- Williams, J.A.¹ McChesney, D.J.²

20
- 0021839251
- (1985) J. Biol. Chem , vol.260 , pp. 7309
- Streb, H.¹ Heslob, J.P.² Irvine, R.F.³ Shultz, I.⁴ Berridge, M.J.⁵

21
- 0023866587
- (1988) Neurochem , vol.50 , pp. 954
- Wennogle, L.¹ Wysowskyj, H.² Steel, D.J.³ Petrack, B.J.⁴

22
- 0026559686
- (1992) Proc. Natl. Acad. Sci. U.S.A , vol.89 , pp. 3125
- Wank, S.A.¹ Harkins, R.² Jenson, R.T.³ Shapira, H.⁴ De Weerth, A.⁵ Slattery, T.⁶

23
- 0026672627
- (1992) Proc. Natl. Acad. Sci. U.S.A , vol.89 , pp. 8691
- Wank, S.A.¹ Pisegna, J.R.² De Weerth, A.³

24
- 0026535933
- (1992) Proc. Natl. Acad. Sci. USA , vol.89 , pp. 3605
- Kopin, A.S.¹ Lee, Y.-M.² McBride, E.W.³ Miller, L.J.⁴ Lu, M.⁵ Lin, H.Y.⁶ Kolakowski, L.F.⁷ Beinborn, M.⁸

25
- 2142814780
- Wang, R.Y., Schoenfeld, R., Eds., Alan, R. Liss, New York
- (1988) Neurology and Neurobiology , vol.47 , pp. 327
- Gertz, B.J.¹

26
- 77956808092
- (1991) Annu. Rep. Med. Chem , vol.26 , pp. 191
- Nadzan, A.M.¹ Kerwin J.F., Jr.²

27
- 0024361890
- (1989) Med. Res. Rev , vol.9 , pp. 271
- Freidinger, R.M.¹

28
- 0001373498
- (1989) Drugs Future , vol.14 , pp. 971
- Evans, B.E.¹

29
- 0001273525
- (1993) Adv. Med. Chem , vol.2 , pp. 111
- Evans, B.E.¹ Bock, M.G.²

30
- 0000205803
- Hansch, C., Sammes, P.G., Taylor, J.B., Eds., Pergamon Press, Oxford
- (1990) Comprehensive Medicinal Chemistry , vol.3 , pp. 925
- Martinez, J.¹

31
- 0022102999
- (1985) Am. J. Physiol , vol.249
- Jenson, R.T.¹ Murphy, R.B.² Trampota, M.³ Schneider, L.H.⁴ Jones, S.W.⁵ Howard, J.M.⁶ Gardner, J.D.⁷

32
- 0021436076
- (1984) Am. J. Physiol , vol.246
- Gardener, J.D.¹ Jensen, R.T.²

33
- 0022966522
- (1986) Am. J. Physiol , vol.251
- Jenson, R.T.¹ Zhou, Z.C.² Murphy, R.B.³ Jones, S.W.⁴ Setnikar, I.⁵ Rovati, L.A.⁶ Gardner, J.D.⁷

34
- 0018765587
- (1979) J. Biol. Chem , vol.254 , pp. 5321
- Peikin, S.R.¹ Costenbader, C.L.² Gardner, J.D.³

35
- 2142704836
- (1982) Am. J. Physiol , vol.242
- Barlas, N.¹ Jensen, R.T.² Beinfeld, M.C.³ Gardner, J.D.⁴

36
- 0014218864
- (1967) Minerva Med , vol.58 , pp. 3651
- Rovati, A.L.¹ Casula, P.L.² Dare, G.³

37
- 0019308879
- (1980) Hipato-Gastroenterol , vol.27 , pp. 41
- Vidal, Y.¹ Plana, R.R.² Cifarelli, A.³ Bizarri, D.⁴

38
- 0017047608
- (1976) Scand. J. Gastroenterol , vol.11 , Issue.SUPPL. 42 , pp. 113
- Rovati, A.L.¹

39
- 0001128176
- (1981) Proc. Natl. Acad. Sci. U.S.A , vol.78 , pp. 6304
- Hahne, W.F.¹ Jensen, R.T.² Lemp, G.F.³ Gardner, J.D.⁴

40
- 0022658129
- (1986) Horm. Metabol. Res , vol.18 , pp. 2
- Maton, P.N.¹ Jensen, R.T.² Gardner, J.D.³

41
- 0021041172
- (1983) Biochim. Biophys. Acta , vol.761 , pp. 269
- Jensen, R.T.¹ Jones, S.W.² Gardner, J.D.³

42
- 0022053507
- (1985) Am. J. Physiol , vol.248
- Maton, P.N.¹ Sutliff, V.E.² Jenson, R.T.³ Gardner, J.D.⁴

43
- 0002270761
- (1979) J. Med. Chem , vol.22 , pp. 2
- Sternbach, L.H.¹

44
- 0028847439
- (1995) Prog. Drug. Res , vol.45 , pp. 67
- Gupta, S.P.¹

45
- 0018835633
- (1980) Science , vol.207 , pp. 274
- Tallman, J.F.¹ Paul, S.M.² Skolnick, P.³ Gallager, D.W.⁴

46
- 0022365699
- (1985) J. Antibiot , vol.38 , pp. 1633
- Goetz, M.A.¹ Lopez, M.² Monaghan, R.L.³ Chang, R.S.L.⁴ Lotti, V.J.⁵ Chen, T.B.⁶

47
- 0022373437
- (1985) Science , vol.230 , pp. 177
- Chang, R.S.L.¹ Lotti, V.J.² Monaghan, R.L.³ Birnbaum, J.⁴ Stapley, E.O.⁵ Goetz, M.A.⁶ Albers-Schonberg, G.⁷ Patchett, A.A.⁸ Liesch, J.M.⁹ Hensens, O.D.¹⁰ Springer, J.P.¹¹

48
- 0023786383
- (1988) J. Antibiot , vol.41 , pp. 875
- Goetz, M.A.¹ Monaghan, R.L.² Chang, R.S.L.³ Ondeyka, J.⁴ Chen, T.B.⁵ Lotti, V.J.⁶

49
- 0023793422
- (1988) J. Antibiot , vol.41 , pp. 878
- Liesch, J.M.¹ Hensens, O.D.² Zink, D.L.³ Goetz, M.A.⁴

50
- 0022345752
- (1985) J. Antibiot , vol.38 , pp. 1638
- Liesch, J.M.¹ Hensens, O.D.² Springer, J.P.³ Chang, R.S.L.⁴ Lotti, V.⁵

51
- 0001151817
- (1983) Proc. Natl. Acad. Sci. U.S.A , vol.80 , pp. 3531
- Guidotti, A.¹ Furchetti, C.M.² Corda, M.G.³ Konkel, D.⁴ Bennet, C.D.⁵ Costa, E.⁶

52
- 0022363286
- (1985) Science , vol.229 , pp. 179
- Alho, H.¹ Costa, E.² Ferrero, P.³ Fujimoto, M.⁴ Cosenza-Murphy, D.⁵ Guidotti, A.⁶

53
- 0010401679
- (1986) Proc. Natl. Acad. Sci. U.S.A , vol.83 , pp. 4918
- Evans, B.E.¹ Bock, M.G.² Rittle, K.E.³ Di Pardo, R.M.⁴ Whitter, W.L.⁵ Veber, D.F.⁶ Anderson, P.S.⁷ Freidinger, R.M.⁸

54
- 0001603410
- (1986) Proc. Natl. Acad. Sci. U.S.A , vol.83 , pp. 4923
- Chang, R.S.L.¹ Lotti, V.J.²

55
- 0024239320
- (1988) J. Med. Chem , vol.31 , pp. 2235
- Evans, B.E.¹ Rittle, K.E.² Bock, M.G.³ Di Pardo, R.M.⁴ Freidinger, R.M.⁵ Whitter, W.L.⁶ Lunden, G.F.⁷ Veber, D.F.⁸ Anderson, P.S.⁹ Chang, R.S.L.¹⁰ Lotti, V.J.¹¹ Cerino, D.J.¹² Chen, T.B.¹³ Kling, P.J.¹⁴ Kunkel, K.A.¹⁵ Springer, J.P.¹⁶ Hirshfield, J.J.¹⁷

56
- 2142649762
- (1989) J. Med. Chem , vol.32 , pp. 13
- Boc, M.G.¹ Di Pardo, R.M.² Evans, B.E.³ Rittle, K.E.⁴ Whitter, W.L.⁵ Veber, D.F.⁶ Anderson, P.F.⁷ Freidinger, R.M.⁸

57
- 0024520619
- (1989) Eur. J. Pharmacol , vol.162 , pp. 273
- Lotti, V.J.¹ Chang, R.S.L.²

58
- 0001128176
- (1981) Proc. Natl. Acad. Sci. U.S.A , vol.78 , pp. 6304
- Hahne, W.F.¹ Jensen, R.T.² Lemp, G.F.³ Gardner, J.D.⁴

59
- 0025770236
- (1991) J. Med. Chem , vol.34 , pp. 1505
- Yu, M.J.¹ Thrasher, K.J.² McCowan, J.R.³ Mason, N.R.⁴ Mendelsohn, L.G.⁵

60
- 0026718844
- (1992) J. Med. Chem , vol.35 , pp. 2534
- Yu, M.J.¹ McCowan, J.R.² Mason, N.R.³ Deter, J.B.⁴ Mendelsohn, L.G.⁵

61
- 0020644532
- (1983) J. Biol. Chem , vol.258 , pp. 6746
- Spanarkel, M.¹ Martinez, J.² Briet, C.³ Jensen, R.T.⁴ Gardener, J.D.⁵

62
- 0022996585
- (1986) J. Med. Chem , vol.29 , pp. 2201
- Martinez, J.¹ Rodriguez, M.² Castro, B.³ Bali, J.-P.⁴ Laur, J.⁵

63
- 0022405729
- (1985) J. Med. Chem , vol.28 , pp. 1874
- Martinez, J.¹ Bali, J.-P.² Rodriguez, M.³ Castro, B.⁴ Magous, R.⁵ Laur, J.⁶ Lignon, M.-F.⁷

64
- 0022480008
- (1988) Int. J. Pept. Prot. Res , vol.27 , pp. 293
- Rodriguez, M.¹ Bali, J.-P.² Magous, R.³ Castro, B.⁴ Martinez, J.⁵

65
- 0023235968
- (1987) J. Med. Chem , vol.30 , pp. 1366
- Rodriguez, M.¹ Lignon, M.-F.² Galas, J.C.³ Fulcrand, P.⁴ Mendro, C.⁵ Aumelas, A.⁶ Laur, J.⁷ Martinez, J.⁸

66
- 0023696163
- (1988) J. Biol. Chem , vol.263 , pp. 10641
- Mendre, C.¹ Rodriguez, M.² Gueudet, C.³ Lignon, M.-F.⁴ Galas, M.-C.⁵ Laur, J.⁶ Worms, P.⁷ Martinez, J.⁸

67
- 0008947877
- Kuchar, M., Ed., J.R. Prous Science Publishers, Barcelona, Spain
- (1992) QSAR in Design of Bioactive Compounds , pp. 285
- Gupta, S.P.¹ Saha, R.N.²

68
- 0028004476
- (1994) J. Med. Chem , vol.37 , pp. 3639
- Tokarski, J.¹ Hopfinger, A.J.²

69
- 2142821920
- (1988) J. Mol. Struc , vol.453 , pp. 97
- Huché, M.¹ Cense, J.-M.² Legendre, J.-J.³

70
- 0033051468
- (1999) Bioorg. Med. Chem , vol.7 , pp. 1127
- Sinha, J.¹ Kurup, A.² Paleti, A.³ Gupta, S.P.⁴

71
- 0021039340
- (1983) Neuropeptides , vol.3 , pp. 411
- Beinfeld, M.C.¹

72
- 0029565241
- (1995) Quant. Struct.-Act. Relat , vol.14 , pp. 437
- Gupta, S.P.¹ Mulchandani, V.² Das, S.³ Subbiah, A.⁴ Narsimha Reddy, D.⁵ Sinha, J.⁶

73
- 0023222021
- (1987) J. Med. Chem , vol.30 , pp. 1229
- Evans, B.E.¹ Rittle, K.E.² Bock, M.G.³ Di Pardo, R.M.⁴ Freidinger, R.M.⁵ Whitter, W.L.⁶ Gould, N.P.⁷ Lundell, P.S.⁸ Chang, R.S.L.⁹ Lotti, V.J.¹⁰ Chen, T.B.¹¹ Kling, P.J.¹² Kunkel, K.A.¹³ Springer, J.P.¹⁴ Hirshfield, J.J.¹⁵

75
- 0027026407
- (1992) J. Comput.-Aided Molec. Des , vol.6 , pp. 553
- Rault, S.¹ Burea, R.² Pilo, J.C.³ Robba, M.⁴

76
- 0020514512
- (1983) Arzneim.-Forsch , vol.33 , pp. 1086
- Borea, P.A.¹

77
- 0028077890
- (1944) Drug Des. Discov , vol.12 , pp. 129
- van der Bent, A.¹ Ijzerman, A.P.² Soudijn, W.³

78
- 0032537618
- (1998) Bioorg. Med. Chem , vol.8 , pp. 1449
- Tabuchi, S.¹ Nakanishi, I.² Satoh, Y.³

79
- 0026515186
- (1992) J. Med. Chem , vol.35 , pp. 28
- Makovec, F.¹ Peris, W.² Revel, L.³ Giovanetti, R.⁴ Mennuni, L.⁵ Rovati, L.C.⁶

80
- 0028379870
- (1994) Indian J. Biochem. Biophys , vol.31 , pp. 55
- Singh, P.¹ Tiwari, S.² Sharma, R.C.³ Ojha, T.N.⁴

81
- 0022648286
- (1986) Eur. J. Med. Chem , vol.21 , pp. 9
- Makovec, F.¹ Chisté, R.² Bani, M.³ Revel, L.⁴ Setnikar, I.⁵ Rovati, A.L.⁶

82
- 0025152919
- (1990) Quant. Struct.-Act. Relat , vol.9 , pp. 94
- Coats, E.A.¹ Knittel, J.J.²

83
- 0025066135
- (1990) J. Med. Chem , vol.33 , pp. 2950
- Shiosaki, K.¹ Lin, C.W.² Kopecka, H.³ Craig, R.⁴ Wagenaar, F.⁵ Bianchi, B.⁶ Miller, T.⁷ Witte, D.⁸ Nazdan, A.M.⁹

84
- 0026017959
- (1991) J. Med. Chem , vol.34 , pp. 2837
- Shiosaki, K.¹ Lin, C.W.² Kopecka, H.³ Tufano, M.D.⁴ Bianchi, B.⁵ Miller, T.⁶ Witte, D.⁷ Nazdan, A.M.⁸

85
- 0030972940
- (1997) J. Med. Chem , vol.40 , pp. 1169
- Shiosaki, K.¹ Lin, C.W.² Kopecka, H.³ Bianchi, B.⁴ Miller, T.⁵ Stashko, M.⁶ Witte, D.⁷

86
- 0026623087
- (1992) J. Med. Chem , vol.35 , pp. 2007
- Shiosaki, K.¹ Lin, C.W.² Kopecka, H.³ Craig, R.A.⁴ Bianchi, B.⁵ Miller, T.⁶ Witte, D.⁷ Stashko, M.⁸ Nazdan, A.M.⁹

87
- 0026092714
- (1991) J. Med. Chem , vol.34 , pp. 404
- Horwell, D.C.¹ Hughes, J.² Hunter, J.C.³ Pritchard, M.C.⁴ Richardson, R.S.⁵ Roberts, E.⁶ Woodruff, G.N.⁷

88
- 0344230147
- (1996) Bioorg. Med. Chem , vol.4 , pp. 1733
- Augelli-Szafran, C.E.¹ Horwell, D.C.² Kneen, C.³ Ortwine, D.F.⁴ Pritchard, M.C.⁵ Purchase, T.S.⁶ Roth, B.D.⁷ Trivedi, B.K.⁸ Hill, D.⁹ Suman-Chauhan, N.¹⁰ Webdale, L.¹¹

89
- 0003537140
- The STERIMOL Approach to Drug Design
- Marcell Dekker, New York
- (1987)
- Verloop, A.¹

90
- 0026753127
- (1992) J. Med. Chem , vol.35 , pp. 1572
- Higginbottom, M.¹ Kneen, C.² Ratcliffe, G.S.³

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