Differences in signal transduction of two 5-HT4 receptor splice variants: Compound specificity and dual coupling with Gαs- and Gαi/o-proteins

Molecular Pharmacology

Volumn 61, Issue 1, 2002, Pages 85-96

  Pindon, Armelle ^a   Van Hecke, Geert ^a   Van Gompel, Paul ^a   Lesage, Anne S ^a   Leysen, Josée E ^a   Jurzak, Mirek ^a  

^a JANSSEN RESEARCH FOUNDATION   (Belgium)

Author keywords

[No Author keywords available]

Indexed keywords

8 AMINO 7 CHLORO 1,4 BENZODIOXAN 5 CARBOXYLIC ACID 1 BUTYL 4 PIPERIDINYLMETHYL ESTER; CYCLIC AMP; FORSKOLIN; GUANINE NUCLEOTIDE BINDING PROTEIN; GUANOSINE 5' O (3 THIOTRIPHOSPHATE); INDOLEAMINE; ISOBUTYLMETHYLXANTHINE; PERTUSSIS TOXIN; PRUCALOPRIDE; SEROTONIN 4 RECEPTOR; TEGASEROD;

ARTICLE; BINDING AFFINITY; BINDING SITE; CALCIUM CELL LEVEL; CALCIUM TRANSPORT; CARBOXY TERMINAL SEQUENCE; HUMAN; HUMAN CELL; LIGAND BINDING; PRIORITY JOURNAL; PROTEIN BINDING; PROTEIN EXPRESSION; RECEPTOR AFFINITY; SIGNAL TRANSDUCTION;

ADENYLATE CYCLASE; ALTERNATIVE SPLICING; CALCIUM; CELL LINE; ENZYME ACTIVATION; GTP-BINDING PROTEIN ALPHA SUBUNITS, GI-GO; GTP-BINDING PROTEIN ALPHA SUBUNITS, GS; GUANOSINE 5'-O-(3-THIOTRIPHOSPHATE); HUMANS; INDOLES; INOSITOL PHOSPHATES; PERTUSSIS TOXIN; RECEPTORS, SEROTONIN; RECEPTORS, SEROTONIN, 5-HT4; SEROTONIN ANTAGONISTS; SIGNAL TRANSDUCTION; SULFONAMIDES; SULFUR RADIOISOTOPES; TRANSFECTION; VIRULENCE FACTORS, BORDETELLA;

EID: 0036140947     PISSN: 0026895X     EISSN: None     Source Type: Journal    
DOI: 10.1124/mol.61.1.85     Document Type: Article

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