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Volumn 10, Issue 2, 2002, Pages 437-448

5-Phenyl substituted 1-methyl-2-pyridones and 4′-substituted biphenyl-4-carboxylic acids. synthesis and evaluation as inhibitors of steroid-5α-reductase type 1 and 2

(3) Picard, Franck a Schulz, Tobias a Hartmann, Rolf W a

a SAARLAND UNIVERSITY (Germany)

Author keywords

[No Author keywords available]

Indexed keywords

1 METHYL 2 PYRIDONE DERIVATIVE; ANDROSTANOLONE; BIPHENYL 4 CARBOXYLIC ACID DERIVATIVE; MEMBRANE ENZYME; STEROID 5ALPHA REDUCTASE; STEROID 5ALPHA REDUCTASE INHIBITOR; TESTOSTERONE; UNCLASSIFIED DRUG;

ANIMAL CELL; ARTICLE; COLUMN CHROMATOGRAPHY; CONTROLLED STUDY; CRYSTALLIZATION; DRUG SYNTHESIS; ENZYME INHIBITION; ENZYME ISOLATION; HUMAN; HUMAN CELL; NONHUMAN; OXIDATION; POWDER; PROSTATE; PROSTATE HYPERTROPHY; RAT; STRUCTURE ACTIVITY RELATION; TEMPERATURE;

ANIMALS; CARBOXYLIC ACIDS; DRUG EVALUATION, PRECLINICAL; ENZYME INHIBITORS; HUMANS; INHIBITORY CONCENTRATION 50; ISOENZYMES; MALE; PROSTATE; RATS; TESTOSTERONE 5-ALPHA-REDUCTASE;

EID: 0036132203 PISSN: 09680896 EISSN: None Source Type: Journal
DOI: 10.1016/S0968-0896(01)00293-0 Document Type: Article

Times cited : (53)

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