Synthesis, reactions and uses of enaminone esters

Saudi Pharmaceutical Journal

Volumn 10, Issue 1-2, 2002, Pages 1-8

  Edafiogho, Ivan O ^a  

^a KUWAIT UNIVERSITY   (Kuwait)

Author keywords

Enaminones; Reactions; Synthesis; Uses

Indexed keywords

ACETYLACETONE; AMIDE; ANTICONVULSIVE AGENT; ANTIVIRUS AGENT; ENAMINONE ESTER DERIVATIVE; ESTER DERIVATIVE; UNCLASSIFIED DRUG;

ALKYLATION; ANTICONVULSANT ACTIVITY; ANTIMALARIAL ACTIVITY; ANTIVIRAL ACTIVITY; CHEMICAL BINDING; CYCLIZATION; DRUG ACTIVITY; DRUG STRUCTURE; DRUG SYNTHESIS; ENANTIOMER; FOOD INDUSTRY; INFRARED RADIATION; INFRARED SPECTROMETRY; PROTON NUCLEAR MAGNETIC RESONANCE; REVIEW; STRUCTURE ACTIVITY RELATION; STRUCTURE ANALYSIS; ULTRAVIOLET RADIATION; ULTRAVIOLET SPECTROSCOPY;

EID: 0036096083     PISSN: 13190164     EISSN: None     Source Type: Journal    
DOI: None     Document Type: Review

References (28)

1. Enaminones
2. Synthesis, reactions and preliminary evaluations of enaminone esters
3. Aromatic enaminones. Part 1. Ultra violet absorption of N-aryl enaminones derived from dimedone
4. Reactions with aldehydes of enaminones derived from dimedone
5. Unsaturated amines. XIII. The sites of alkylation and protonation in certain enamino ketones. Substituted trimethinium compounds from O-alkylated enamino ketones
6. A study of the rates of hydrolysis of certain enaminones
7. Condensation of diethyl malonate with methyl vinyl ketone
8. Alkylation of enaminone esters
9. Some pharmacological effects of an enaminone ester on an isolated rat uterus
10. The chemotherapy of viral infections
11. Anticonvulsant enaminones: With emphasis on methyl4-[(p-chlorophenyl)-amino-6-methyl-2-oxocyclo hex -3-en-1-oate (ADD 906022)]
12. Synthesis and anticonvulsant activity of enaminones
13. Chapter 39, "Anticonvulsants"
14. Synthesis, characterization and anticonvulsant activity of enaminones. Part 6: Synthesis of substituted vinylic benzamides as potential anticonvulsants
15. Enaminones - Versatile therapeutic pharmacophores. Further advances
16. Nuclear magnetic resonance studies of anticonvulsant enaminones
17. Enaminones: Versatile intermediates for natural product synthesis
18. Stability study of an anticonvulsant enaminone (E139) using HPLC
19. Mechanism of hydrolysis and structure-stability relationship of enaminones as potential prodrugs of model primary amines
20. Chapter 35: Antiprotozoal drugs
21. Reaction of N, N-disubstituted alpha-aminomethyleneketones with tosyl isocyanate. Synthesis of amino-disubstituted 2-acyl-3-amino-N-tosylpropenamides,N,N,-(3-amino-1-alkyl-2 propeny lidene) and N,N (aminomethylene) cyclohexylidene to sylamides
22. Pharmacological studies on the centrally-acting drugs belonging to enaminone Mannich bases II. Pharmacology of MK 1-203 and 1-907, new potent analgesics
23. Synthesis and antimalarial properties of 1-imino derivatives of 7-chloro-3-substituted-3, 4-dihydro-1,9 (2H, 10H)-acridinediones and related structures
24. Synthesis and anticonvulsant activity of enaminones. 2. Further structure activity correlations
25. Synthesis, characterization, and anticonvulsant activity of enaminones. Part 5: Investigations on 3-carboalkoxy-2-methyl-2, 3-dihydro-1H-phenothiazin-[4,2] [1,2]OH-one derivatives
26. 1-Pyrrolines (3,4-dihydro-2H-pyrroles) as a template for new drugs
27. Potential anxiolytic agents. Pyrido and [2][1,2][2a] benzoimidazoles: A new structural class of ligands for the binding site on GABA-A receptors
28. Hypertensive effects and structure-activity relationships of 5-omega-aminoalkyl isoxazoles