Synthesis and antituberculosis activity of cycloalkylidenehydrazide and 4-aza-1-thiaspiro [4.5] decan-3-one derivatives of imidazo[2,1-b]thiazole

Arzneimittel-Forschung/Drug Research

Volumn 52, Issue 7, 2002, Pages 565-571

  Ulusoy, Nuray ^a  

^a ISTANBUL UNIVERSITY   (Turkey)

Author keywords

Antituberculosis drugs; Imidazo 2,1 b thiazolylcycloalkylidenehydrazides, antituberculosis activity, structural determination, synthesis; Spirothiazolidinones, antituberculosis activity, structural determination, synthesis

Indexed keywords

(4 CHLOROPHENYLIMIDAZO[2,1 B]THIAZOL 3 YL)ACETIC ACID; (6 PHENYLIMIDAZO [2,1 B]THIAZOL 3 YL)ACETIC ACID; 4 AZA 1 THIASPIRO[4.5]DECAN 3 ONE DERIVATIVE; 4 [[(4 CHLOROPHENYLIMIDAZO[2,1 B]THIAZOL 3 YL)ACETYL]AMINO] 4 AZA 1 THIASPIRO[4.5]DECAN 3 ONE DERIVATIVE; 4 [[(6 PHENYLIMIDAZO[2,1 B]THIAZOL 3 YL)ACETYL]AMINO] 4 AZA 1 THIASPIRO[4.5]DECAN 3 ONE DERIVATIVE; CYCLOPENTANONE DERIVATIVE; HYDRAZIDE DERIVATIVE; HYDRAZINE DERIVATIVE; IMIDAZO[2,1 B]THIAZOLE DERIVATIVE; LACTIC ACID DERIVATIVE; THIOGLYCOLIC ACID; TUBERCULOSTATIC AGENT; UNCLASSIFIED DRUG;

ANTIMICROBIAL ACTIVITY; ARTICLE; BACTERIUM CULTURE; CARBON NUCLEAR MAGNETIC RESONANCE; CHEMICAL REACTION; CONCENTRATION RESPONSE; CONTROLLED STUDY; DRUG STRUCTURE; DRUG SYNTHESIS; INFRARED SPECTROMETRY; MASS SPECTROMETRY; MINIMUM INHIBITORY CONCENTRATION; MYCOBACTERIUM TUBERCULOSIS; NONHUMAN; PROTON NUCLEAR MAGNETIC RESONANCE; REACTION ANALYSIS; STRUCTURE ACTIVITY RELATION;

EID: 0036077005     PISSN: 00044172     EISSN: None     Source Type: Journal    
DOI: 10.1055/s-0031-1299931     Document Type: Article

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