Prenylamine block of Nav1.5 channel is mediated via a receptor distinct from that of local anesthetics

Molecular Pharmacology

Volumn 62, Issue 2, 2002, Pages 415-422

  Mujtaba, Mustafa G ^b   Wang, Sho Ya ^a   Wang, Ging Kuo ^b  

^a STATE UNIVERSITY OF NEW YORK   (United States)

^b BRIGHAM AND WOMEN S HOSPITAL   (United States)

Author keywords

[No Author keywords available]

Indexed keywords

BUPIVACAINE; COMPLEMENTARY DNA; LOCAL ANESTHETIC AGENT; LYSINE; PRENYLAMINE; SODIUM CHANNEL; SODIUM CHANNEL BLOCKING AGENT;

AMINO ACID SUBSTITUTION; ARTICLE; CONTROLLED STUDY; DEPOLARIZATION; DRUG BINDING SITE; EMBRYO; HEART; HUMAN; HUMAN CELL; HYPERPOLARIZATION; KIDNEY CELL; LOCAL ANESTHESIA; PRIORITY JOURNAL; SITE DIRECTED MUTAGENESIS; VOLTAGE CLAMP;

ANESTHETICS, LOCAL; ANILINE COMPOUNDS; BUPIVACAINE; CELLS, CULTURED; DRUG INTERACTIONS; HUMANS; MUTAGENESIS, SITE-DIRECTED; MYOCARDIUM; SODIUM CHANNEL BLOCKERS; SODIUM CHANNELS; TRANSFECTION;

EID: 0036070820     PISSN: 0026895X     EISSN: None     Source Type: Journal    
DOI: 10.1124/mol.62.2.415     Document Type: Article

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