Cloned human EP1 prostanoid receptor pharmacology characterized using radioligand binding techniques

Journal of Pharmacy and Pharmacology

Volumn 54, Issue 4, 2002, Pages 539-547

  Sharif, Najam A ^a   Davis, Terry L ^a  

^a ALCON RESEARCH LTD   (United States)

Author keywords

[No Author keywords available]

Indexed keywords

17 PHENYL OMEGA TRINORPROSTAGLANDIN E2; 6 ISOPROPOXY 9 OXO 2 XANTHENECARBOXYLIC ACID; 7 [3 [(4 PHENYLSEMICARBAZIDO)METHYL] 7 OXABICYCLO[2.2.1]HEPT 2 YL] 5 HEPTENOIC ACID; 7 [5 (4 BIPHENYLYLMETHOXY) 2 MORPHOLINO 3 OXOCYCLOPENTYL] 4 HEPTENOIC ACID; 9BETA CHLORO 15 CYCLOHEXYL 9 DEOXY 16,17,18,19,20 PENTANOR 3 OXAPROSTAGLANDIN F2 ALPHA; 9BETA CHLORO 15 CYCLOHEXYL 9 DEOXY 16,17,18,19,20 PENTANORPROSTAGLANDIN F2 ALPHA; AL 24615; AL 24620; AL 6556; AL 6598; BW 868C; BWA 245C; CLOPROSTENOL; ENPROSTIL; FLUPROSTENOL; ILOPROST; LATANOPROST; MISOPROSTOL; PROSTACYCLIN; PROSTAGLANDIN; PROSTAGLANDIN D2; PROSTAGLANDIN E1; PROSTAGLANDIN E2; PROSTAGLANDIN F2; PROSTANOID RECEPTOR; RADIOLIGAND; RECEPTOR SUBTYPE; RECOMBINANT PROSTANOID EP1 RECEPTOR; RECOMBINANT RECEPTOR; RS 93520; S 1033; SC 19920; SQ 27986; SULPROSTONE; TRAVOPROST; UNCLASSIFIED DRUG; UNINDEXED DRUG; UNOPROSTONE ISOPROPYL ESTER; DIAGNOSTIC AGENT; LIGAND; PROSTAGLANDIN E; PROSTAGLANDIN E RECEPTOR; PROSTAGLANDIN F2 ALPHA; PROSTANOID RECEPTOR EP1; RECOMBINANT DNA; TRITIUM;

ARTICLE; BINDING AFFINITY; BINDING COMPETITION; CELL MEMBRANE; CONCENTRATION (PARAMETERS); DRUG RECEPTOR BINDING; DRUG SPECIFICITY; EMBRYO CELL; HUMAN; HUMAN CELL; KIDNEY CELL; LIGAND BINDING; MOLECULAR CLONING; PROTEIN EXPRESSION; RECEPTOR AFFINITY; RECEPTOR BINDING; RECEPTOR INTRINSIC ACTIVITY; SCATCHARD PLOT; ALGORITHM; CELL LINE; DOSE RESPONSE; DRUG EFFECT; GENETICS; METABOLISM; RADIOASSAY;

ALGORITHMS; ALPROSTADIL; BINDING, COMPETITIVE; CELL LINE; CELL MEMBRANE; CLONING, MOLECULAR; DINOPROST; DINOPROSTONE; DNA, RECOMBINANT; DOSE-RESPONSE RELATIONSHIP, DRUG; EPOPROSTENOL; HUMANS; LIGANDS; PROSTAGLANDIN D2; PROSTAGLANDINS E; RADIOLIGAND ASSAY; RECEPTORS, PROSTAGLANDIN E; TRITIUM;

EID: 0036010492     PISSN: 00223573     EISSN: None     Source Type: Journal    
DOI: 10.1211/0022357021778655     Document Type: Article

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