Cardioselective KATP channel blockers derived from a new series of m-anisamidoethylbenzenesulfonylthioureas

Journal of Medicinal Chemistry

Volumn 44, Issue 7, 2001, Pages 1085-1098

  Englert, H C ^a   Gerlach, U ^a   Goegelein, H ^a   Hartung, J ^a   Heitsch, H ^a   Mania, D ^a   Scheidler, S ^a  

^a SANOFI AVENTIS DEUTSCHLAND GMBH   (Germany)

Author keywords

[No Author keywords available]

Indexed keywords

ADENOSINE TRIPHOSPHATASE (POTASSIUM); CLAMIKALANT; GLIBENCLAMIDE; POTASSIUM CHANNEL; POTASSIUM CHANNEL BLOCKING AGENT; SULFONYLUREA DERIVATIVE; UNCLASSIFIED DRUG;

ANIMAL TISSUE; ARTICLE; CARDIOSELECTIVITY; CORONARY ARTERY DISEASE; DRUG POTENCY; DRUG SCREENING; DRUG STRUCTURE; GENETIC TRANSFECTION; GUINEA PIG; HEART ARRHYTHMIA; HEART MUSCLE POTENTIAL; MEMBRANE DEPOLARIZATION; NONHUMAN; STRUCTURE ACTIVITY RELATION; SUDDEN DEATH;

ACTION POTENTIALS; ADENOSINE TRIPHOSPHATE; ANIMALS; ANTI-ARRHYTHMIA AGENTS; ARRHYTHMIA; ATP-BINDING CASSETTE TRANSPORTERS; CHO CELLS; CRICETINAE; DEATH, SUDDEN; ELECTRIC STIMULATION; FEMALE; GUINEA PIGS; HEART; MALE; MYOCARDIAL CONTRACTION; POTASSIUM CHANNEL BLOCKERS; POTASSIUM CHANNELS; POTASSIUM CHANNELS, INWARDLY RECTIFYING; RECEPTORS, DRUG; STRUCTURE-ACTIVITY RELATIONSHIP; SULFONAMIDES; THIOUREA;

EID: 0035966877     PISSN: 00222623     EISSN: None     Source Type: Journal    
DOI: 10.1021/jm000985v     Document Type: Article

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