A stereocontrolled approach to substituted piperidones and piperidines: Flavopiridol D-ring analogs

Tetrahedron Letters

Volumn 42, Issue 9, 2001, Pages 1631-1633

  Gross, Alexandre ^a   Borcherding, David R ^a   Friedrich, Dirk ^a   Sabol, Jeffrey S ^a  

^a SANOFI   (France)

Author keywords

[No Author keywords available]

Indexed keywords

ANTINEOPLASTIC AGENT; FLAVONE DERIVATIVE; FLAVOPIRIDOL; FLAVOPIRIDOL DERIVATIVE; PIPERIDINE DERIVATIVE; PIPERIDONE DERIVATIVE; UNCLASSIFIED DRUG;

ARTICLE; DRUG STRUCTURE; DRUG SYNTHESIS; REACTION ANALYSIS; STEREOCHEMISTRY;

EID: 0035951928     PISSN: 00404039     EISSN: None     Source Type: Journal    
DOI: 10.1016/S0040-4039(00)02350-9     Document Type: Article

References (9)

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5. 3), 2.40 m (H-6β), 1.54 m (H-5β), 1.26 d (3H; J=6.5 Hz; H-7), NOEs between axial H-4β and axial H-2β, H-6β.
6. The authors thank Drs. Philip Weintraub and Ronald Bernotas for helpful discussions.
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