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Bioorganic and Medicinal Chemistry Letters

Volumn 11, Issue 8, 2001, Pages 1065-1068

Design, synthesis and stability of N-acyloxymethyl- and N-aminocarbonyloxymethyl-2-azetidinones as human leukocyte elastase inhibitors

(9) Clemente, A a Domingos, A a Grancho, A P a Iley, J b Moreira, R c Neres, J c Palma, N d,e Santana, A B c Valente, E c

a INETI (Portugal)

b OPEN UNIVERSITY (United Kingdom)

c RESEARCH INSTITUTE FOR MEDICINES IMED ULISBOA (Portugal)

d UNIVERSIDADE NOVA DE LISBOA (Portugal)

e INSTITUTO SUPERIOR DE CIÊNCIAS DA SAÚDE EGAS MONIZ (Portugal)

Author keywords

[No Author keywords available]

Indexed keywords

AZETIDINONE DERIVATIVE; LEUKOCYTE ELASTASE INHIBITOR; N ACYLOXYMETHYL 2 AZETIDINONE DERIVATIVE; N AMINOCARBONYLOXYMETHYL 2 AZETIDINONE DERIVATIVE; UNCLASSIFIED DRUG;

ARTICLE; DRUG DESIGN; DRUG POTENCY; DRUG SELECTIVITY; DRUG STABILITY; DRUG SYNTHESIS; ENZYME INHIBITION; HUMAN; MOLECULAR MODEL;

AZETIDINES; DRUG DESIGN; DRUG STABILITY; ENZYME INHIBITORS; HUMANS; LEUKOCYTE ELASTASE; MODELS, MOLECULAR; SENSITIVITY AND SPECIFICITY;

EID: 0035938401 PISSN: 0960894X EISSN: None Source Type: Journal
DOI: 10.1016/S0960-894X(01)00131-7 Document Type: Article

Times cited : (52)

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